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PDB: 1 件

8RIY
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Human NUDT5 with ibrutinib derivative
分子名称: 1-(1-methylpiperidin-4-yl)-3-(4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-4-amine, ADP-sugar pyrophosphatase
著者Balikci-Akil, E, Elkins, J.M, Huber, K.V.M.
登録日2023-12-19
公開日2024-05-01
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (2.288 Å)
主引用文献Unexpected Noncovalent Off-Target Activity of Clinical BTK Inhibitors Leads to Discovery of a Dual NUDT5/14 Antagonist.
J.Med.Chem., 67, 2024

221716

件を2024-06-26に公開中

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