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PDB: 1 results

8ATZ
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BU of 8atz by Molmil
Crystal structure of PPAR gamma (PPARG) in complex with SA112 (compound 2).
Descriptor: 2-[4-chloranyl-6-[[3-(2-phenylethoxy)phenyl]amino]pyrimidin-2-yl]sulfanylethanoic acid, GLYCEROL, Peroxisome proliferator-activated receptor gamma
Authors:Chaikuad, A, Arifi, S, Merk, D, Knapp, S, Structural Genomics Consortium (SGC)
Deposit date:2022-08-24
Release date:2023-07-12
Last modified:2024-02-07
Method:X-RAY DIFFRACTION (1.95 Å)
Cite:Targeting the Alternative Vitamin E Metabolite Binding Site Enables Noncanonical PPAR gamma Modulation.
J.Am.Chem.Soc., 145, 2023

222926

數據於2024-07-24公開中

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