4IBM
| Crystal structure of insulin receptor kinase domain in complex with an inhibitor Irfin-1 | Descriptor: | 5-(2-phenylpyrazolo[1,5-a]pyridin-3-yl)-3H-pyrazolo[3,4-c]pyridazin-3-one, Insulin receptor | Authors: | Wu, J, Anastassiadis, T, Duong-Ly, K.C, Peterson, J.R. | Deposit date: | 2012-12-08 | Release date: | 2013-08-21 | Last modified: | 2024-02-28 | Method: | X-RAY DIFFRACTION (1.8 Å) | Cite: | A highly selective dual insulin receptor (IR)/insulin-like growth factor 1 receptor (IGF-1R) inhibitor derived from an extracellular signal-regulated kinase (ERK) inhibitor. J.Biol.Chem., 288, 2013
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