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PDB: 1 件

4IBM
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Crystal structure of insulin receptor kinase domain in complex with an inhibitor Irfin-1
分子名称: 5-(2-phenylpyrazolo[1,5-a]pyridin-3-yl)-3H-pyrazolo[3,4-c]pyridazin-3-one, Insulin receptor
著者Wu, J, Anastassiadis, T, Duong-Ly, K.C, Peterson, J.R.
登録日2012-12-08
公開日2013-08-21
最終更新日2024-02-28
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献A highly selective dual insulin receptor (IR)/insulin-like growth factor 1 receptor (IGF-1R) inhibitor derived from an extracellular signal-regulated kinase (ERK) inhibitor.
J.Biol.Chem., 288, 2013

221716

件を2024-06-26に公開中

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