1ST7
| Solution structure of Acyl Coenzyme A Binding Protein from yeast | 分子名称: | Acyl-CoA-binding protein | 著者 | Teilum, K, Thormann, T, Caterer, N.R, Poulsen, H.I, Jensen, P.H, Knudsen, J, Kragelund, B.B, Poulsen, F.M. | 登録日 | 2004-03-25 | 公開日 | 2005-03-01 | 最終更新日 | 2022-03-02 | 実験手法 | SOLUTION NMR | 主引用文献 | Different secondary structure elements as scaffolds for protein folding transition states of two homologous four-helix bundles Proteins, 59, 2005
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4W1O
| PDE4D complexed with inhibitor | 分子名称: | N-(3,5-dichloropyridin-4-yl)-3-[(3-ethyl-1,2-oxazol-5-yl)methoxy]-4-methoxybenzamide, ZINC ION, cAMP-specific 3',5'-cyclic phosphodiesterase 4D | 著者 | Sorensen, M.D. | 登録日 | 2014-08-14 | 公開日 | 2014-11-05 | 最終更新日 | 2020-03-11 | 実験手法 | X-RAY DIFFRACTION (2.2 Å) | 主引用文献 | Discovery and Early Clinical Development of 2-{6-[2-(3,5-Dichloro-4-pyridyl)acetyl]-2,3-dimethoxyphenoxy}-N-propylacetamide (LEO 29102), a Soft-Drug Inhibitor of Phosphodiesterase 4 for Topical Treatment of Atopic Dermatitis J.Med.Chem, 57, 2014
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4WCU
| PDE4 complexed with inhibitor | 分子名称: | MAGNESIUM ION, N-benzyl-2-{6-[(3,5-dichloropyridin-4-yl)acetyl]-2,3-dimethoxyphenoxy}acetamide, ZINC ION, ... | 著者 | Sorensen, M.D. | 登録日 | 2014-09-05 | 公開日 | 2014-10-08 | 実験手法 | X-RAY DIFFRACTION (2.35 Å) | 主引用文献 | Discovery and Early Clinical Development of 2-{6-[2-(3,5-Dichloro-4-pyridyl)acetyl]-2,3-dimethoxyphenoxy}-N-propylacetamide (LEO 29102), a Soft-Drug Inhibitor of Phosphodiesterase 4 for Topical Treatment of Atopic Dermatitis. J. Med. Chem., 57, 2014
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