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1ST7
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BU of 1st7 by Molmil
Solution structure of Acyl Coenzyme A Binding Protein from yeast
分子名称: Acyl-CoA-binding protein
著者Teilum, K, Thormann, T, Caterer, N.R, Poulsen, H.I, Jensen, P.H, Knudsen, J, Kragelund, B.B, Poulsen, F.M.
登録日2004-03-25
公開日2005-03-01
最終更新日2022-03-02
実験手法SOLUTION NMR
主引用文献Different secondary structure elements as scaffolds for protein folding transition states of two homologous four-helix bundles
Proteins, 59, 2005
4W1O
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BU of 4w1o by Molmil
PDE4D complexed with inhibitor
分子名称: N-(3,5-dichloropyridin-4-yl)-3-[(3-ethyl-1,2-oxazol-5-yl)methoxy]-4-methoxybenzamide, ZINC ION, cAMP-specific 3',5'-cyclic phosphodiesterase 4D
著者Sorensen, M.D.
登録日2014-08-14
公開日2014-11-05
最終更新日2020-03-11
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Discovery and Early Clinical Development of 2-{6-[2-(3,5-Dichloro-4-pyridyl)acetyl]-2,3-dimethoxyphenoxy}-N-propylacetamide (LEO 29102), a Soft-Drug Inhibitor of Phosphodiesterase 4 for Topical Treatment of Atopic Dermatitis
J.Med.Chem, 57, 2014
4WCU
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BU of 4wcu by Molmil
PDE4 complexed with inhibitor
分子名称: MAGNESIUM ION, N-benzyl-2-{6-[(3,5-dichloropyridin-4-yl)acetyl]-2,3-dimethoxyphenoxy}acetamide, ZINC ION, ...
著者Sorensen, M.D.
登録日2014-09-05
公開日2014-10-08
実験手法X-RAY DIFFRACTION (2.35 Å)
主引用文献Discovery and Early Clinical Development of 2-{6-[2-(3,5-Dichloro-4-pyridyl)acetyl]-2,3-dimethoxyphenoxy}-N-propylacetamide (LEO 29102), a Soft-Drug Inhibitor of Phosphodiesterase 4 for Topical Treatment of Atopic Dermatitis.
J. Med. Chem., 57, 2014

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件を2024-04-24に公開中

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