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4P24
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BU of 4p24 by Molmil
pore forming toxin
分子名称: (4S)-2-METHYL-2,4-PENTANEDIOL, Alpha-hemolysin
著者Sugawara, T, Yamashita, D, Tanaka, Y, Tanaka, I, Yao, M.
登録日2014-03-01
公開日2015-03-11
最終更新日2023-12-27
実験手法X-RAY DIFFRACTION (3.1 Å)
主引用文献Structural basis for pore-forming mechanism of staphylococcal alpha-hemolysin.
Toxicon, 108, 2015
4YHD
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BU of 4yhd by Molmil
Staphylococcal alpha-hemolysin H35A mutant monomer
分子名称: Alpha-hemolysin, CHLORIDE ION
著者Sugawara, T, Kato, K, Tanaka, Y, Yao, M.
登録日2015-02-27
公開日2015-10-21
最終更新日2024-03-20
実験手法X-RAY DIFFRACTION (2.801 Å)
主引用文献Structural basis for pore-forming mechanism of staphylococcal alpha-hemolysin
Toxicon, 108, 2015
5N49
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BU of 5n49 by Molmil
BRPF2 in complex with Compound 7
分子名称: 2-(1,3,6-trimethyl-2-oxidanylidene-benzimidazol-5-yl)benzo[de]isoquinoline-1,3-dione, Bromodomain-containing protein 1
著者Bouche, L, Christ, C.D, Siegel, S, Fernandez-Montalvan, A.E, Holton, S.J, Fedorov, O, ter Laak, A, Sugawara, T, Stoeckigt, D, Tallant, C, Bennett, J, Monteiro, O, Saez, L.D, Siejka, P, Meier, J, Puetter, V, Weiske, J, Mueller, S, Huber, K.V.M, Hartung, I.V, Haendler, B.
登録日2017-02-10
公開日2017-05-03
最終更新日2017-05-24
実験手法X-RAY DIFFRACTION (1.94 Å)
主引用文献Benzoisoquinolinediones as Potent and Selective Inhibitors of BRPF2 and TAF1/TAF1L Bromodomains.
J. Med. Chem., 60, 2017
5XUV
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BU of 5xuv by Molmil
Crystal structure of DNA duplex containing 4-thiothymine-2Ag(I)-4-thiothymine base pairs
分子名称: DNA (5'-D(*CP*GP*CP*GP*AP*(8RO)P*(8RO)P*TP*CP*GP*CP*G)-3'), POTASSIUM ION, SILVER ION
著者Kondo, J, Sugawara, T, Saneyoshi, H, Ono, A.
登録日2017-06-26
公開日2017-09-20
最終更新日2023-11-22
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Crystal structure of a DNA duplex containing four Ag(i) ions in consecutive dinuclear Ag(i)-mediated base pairs: 4-thiothymine-2Ag(i)-4-thiothymine
Chem. Commun. (Camb.), 53, 2017
5MG2
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BU of 5mg2 by Molmil
Crystal structure of the second bromodomain of human TAF1 in complex with BAY-299 chemical probe
分子名称: 1,2-ETHANEDIOL, 6-(3-oxidanylpropyl)-2-(1,3,6-trimethyl-2-oxidanylidene-benzimidazol-5-yl)benzo[de]isoquinoline-1,3-dione, Transcription initiation factor TFIID subunit 1
著者Tallant, C, Bouche, L, Holton, S.J, Fedorov, O, Siejka, P, Picaud, S, Krojer, T, Srikannathasan, V, von Delft, F, Arrowsmith, C.H, Edwards, A.M, Bountra, C, Hartung, I.V, Haendler, B, Muller, S, Huber, K.V.M, Structural Genomics Consortium (SGC)
登録日2016-11-20
公開日2017-05-03
最終更新日2024-01-17
実験手法X-RAY DIFFRACTION (1.75 Å)
主引用文献Benzoisoquinolinediones as Potent and Selective Inhibitors of BRPF2 and TAF1/TAF1L Bromodomains.
J. Med. Chem., 60, 2017
4P1Y
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BU of 4p1y by Molmil
Crystal structure of staphylococcal gamma-hemolysin prepore
分子名称: Gamma-hemolysin component A, Gamma-hemolysin component B
著者Yamashita, D, Tanaka, Y, Tanaka, I, Yao, M.
登録日2014-02-28
公開日2014-10-01
最終更新日2023-12-27
実験手法X-RAY DIFFRACTION (2.992 Å)
主引用文献Molecular basis of transmembrane beta-barrel formation of staphylococcal pore-forming toxins.
Nat Commun, 5, 2014
4P1X
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BU of 4p1x by Molmil
Crystal structure of staphylococcal LUK prepore
分子名称: (4S)-2-METHYL-2,4-PENTANEDIOL, Gamma-hemolysin component B, Gamma-hemolysin component C
著者Yamashita, D, Tanaka, Y, Tanaka, I, Yao, M.
登録日2014-02-28
公開日2014-10-01
最終更新日2023-12-27
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献Molecular basis of transmembrane beta-barrel formation of staphylococcal pore-forming toxins.
Nat Commun, 5, 2014

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件を2024-04-24に公開中

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