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ORIENTATION OF PEPTIDE FRAGMENTS FROM SOS PROTEINS BOUND TO THE N-TERMINAL SH3 DOMAIN OF GRB2 DETERMINED BY NMR SPECTROSCOPY
分子名称:	GROWTH FACTOR RECEPTOR-BOUND PROTEIN 2, SOS-A PEPTIDE
著者	Wittekind, M, Mapelli, C, Farmer, B.T, Suen, K.-L, Goldfarb, V, Tsao, J, Lavoie, T, Barbacid, M, Meyers, C.A, Mueller, L.
登録日	1994-08-12
公開日	1995-01-26
最終更新日	2022-02-23
実験手法	SOLUTION NMR
主引用文献	Orientation of peptide fragments from Sos proteins bound to the N-terminal SH3 domain of Grb2 determined by NMR spectroscopy. Biochemistry, 33, 1994

MMP-13 in complex with a non zinc-chelating inhibitor
分子名称:	5-(4-chlorophenyl)-N-[(1S)-1-cyclohexyl-2-(methylamino)-2-oxoethyl]furan-2-carboxamide, CALCIUM ION, Collagenase 3, ...
著者	Farrow, N.A.
登録日	2009-07-08
公開日	2009-09-01
最終更新日	2024-02-21
実験手法	X-RAY DIFFRACTION (1.95 Å)
主引用文献	Improving potency and selectivity of a new class of non-Zn-chelating MMP-13 inhibitors. Bioorg.Med.Chem.Lett., 19, 2009

MMP-13 in complex with a non zinc-chelating inhibitor
分子名称:	CALCIUM ION, Collagenase 3, N-[4-(5-{[(1S)-1-cyclohexyl-2-(methylamino)-2-oxoethyl]carbamoyl}furan-2-yl)phenyl]-1-benzofuran-2-carboxamide, ...
著者	Farrow, N.A, Margarit, S.M.
登録日	2009-07-08
公開日	2009-09-01
最終更新日	2024-02-21
実験手法	X-RAY DIFFRACTION (2.208 Å)
主引用文献	Improving potency and selectivity of a new class of non-Zn-chelating MMP-13 inhibitors. Bioorg.Med.Chem.Lett., 19, 2009

Crystal structure of human Pim-1 in complex with DAPPA
分子名称:	(2E)-3-{3-[6-(4-methyl-1,4-diazepan-1-yl)pyrazin-2-yl]phenyl}prop-2-enoic acid, MAGNESIUM ION, Proto-oncogene serine/threonine-protein kinase Pim-1
著者	Qian, K.
登録日	2008-10-29
公開日	2009-03-10
最終更新日	2023-12-27
実験手法	X-RAY DIFFRACTION (1.9 Å)
主引用文献	Hit to lead account of the discovery of a new class of inhibitors of Pim kinases and crystallographic studies revealing an unusual kinase binding mode. J.Med.Chem., 52, 2009