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4PNZ
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BU of 4pnz by Molmil
Human dipeptidyl peptidase IV/CD26 in complex with the long-acting inhibitor Omarigliptin (MK-3102)
分子名称: (2R,3S,5R)-5-[2-(methylsulfonyl)-2,6-dihydropyrrolo[3,4-c]pyrazol-5(4H)-yl]-2-(2,4,5-trifluorophenyl)tetrahydro-2H-pyran-3-amine, 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, ...
著者Scapin, G, Yan, Y.
登録日2014-02-22
公開日2014-04-09
最終更新日2023-09-20
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Omarigliptin (MK-3102): A Novel Long-Acting DPP-4 Inhibitor for Once-Weekly Treatment of Type 2 Diabetes.
J.Med.Chem., 57, 2014
5IEA
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BU of 5iea by Molmil
TRIM5 B-box2 and coiled-coil chimera
分子名称: Tripartite motif-containing protein 5, Serine--tRNA ligase Chimera, ZINC ION
著者Wagner, J.M, Doss, G, Pornillos, O.
登録日2016-02-25
公開日2016-06-15
最終更新日2024-03-06
実験手法X-RAY DIFFRACTION (3.258 Å)
主引用文献Mechanism of B-box 2 domain-mediated higher-order assembly of the retroviral restriction factor TRIM5 alpha.
Elife, 5, 2016
5EIU
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BU of 5eiu by Molmil
Mini TRIM5 B-box 2 dimer C2 crystal form
分子名称: TRIM protein-E3 ligase Chimera, ZINC ION
著者Wagner, J.M, Doss, G, Pornillos, O.
登録日2015-10-30
公開日2016-06-15
最終更新日2024-03-06
実験手法X-RAY DIFFRACTION (1.908 Å)
主引用文献Mechanism of B-box 2 domain-mediated higher-order assembly of the retroviral restriction factor TRIM5 alpha.
Elife, 5, 2016
5F7T
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BU of 5f7t by Molmil
TRIM5 B-box2 and coiled-coil chimera
分子名称: Tripartite motif-containing protein 5,Serine--tRNA ligase,Tripartite motif-containing protein 5, ZINC ION
著者Wagner, J.M, Doss, G, Pornillos, O.
登録日2015-12-08
公開日2016-06-15
最終更新日2024-03-06
実験手法X-RAY DIFFRACTION (2.292 Å)
主引用文献Mechanism of B-box 2 domain-mediated higher-order assembly of the retroviral restriction factor TRIM5 alpha.
Elife, 5, 2016

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件を2024-04-24に公開中

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