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5I97
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BU of 5i97 by Molmil
Structural analysis and inhibition of TraE from the pKM101 type IV secretion system
分子名称: Conjugal transfer protein
著者Casu, B, Sygusch, J, Baron, C.
登録日2016-02-19
公開日2016-09-28
最終更新日2023-09-27
実験手法X-RAY DIFFRACTION (2.441 Å)
主引用文献Structural Analysis and Inhibition of TraE from the pKM101 Type IV Secretion System.
J.Biol.Chem., 291, 2016
8BKY
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BU of 8bky by Molmil
Cryo-EM structure of a contractile injection system in Streptomyces coelicolor, the contracted sheath shell.
分子名称: Phage tail sheath protein
著者Casu, B, Sallmen, J.W, Schlimpert, S, Pilhofer, M.
登録日2022-11-09
公開日2023-03-15
最終更新日2023-04-12
実験手法ELECTRON MICROSCOPY (3.6 Å)
主引用文献Cytoplasmic contractile injection systems mediate cell death in Streptomyces.
Nat Microbiol, 8, 2023
8BL4
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BU of 8bl4 by Molmil
Cryo-EM structure of a contractile injection system in Streptomyces coelicolor, the sheath-tube module in extended state.
分子名称: Phage tail protein, Phage tail sheath family protein
著者Casu, B, Sallmen, J.W, Schlimpert, S, Pilhofer, M.
登録日2022-11-09
公開日2023-03-15
最終更新日2023-04-12
実験手法ELECTRON MICROSCOPY (3.9 Å)
主引用文献Cytoplasmic contractile injection systems mediate cell death in Streptomyces.
Nat Microbiol, 8, 2023
5WIO
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BU of 5wio by Molmil
TraE protein in complex with 4-(1H-pyrrol-1-yl)pyridine-2-carboxylic acid
分子名称: 4-(1H-pyrrol-1-yl)pyridine-2-carboxylic acid, Conjugal transfer protein
著者Casu, B, Arya, T, Bessette, B, Baron, C.
登録日2017-07-19
公開日2017-11-15
最終更新日2023-10-04
実験手法X-RAY DIFFRACTION (2.52 Å)
主引用文献Fragment-based screening identifies novel targets for inhibitors of conjugative transfer of antimicrobial resistance by plasmid pKM101.
Sci Rep, 7, 2017
5WIC
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BU of 5wic by Molmil
TraE protein in complex with 2-Furoic Acid (FOA)
分子名称: 2-FUROIC ACID, Conjugal transfer protein
著者Casu, B, Arya, T, Bessette, B, Baron, C.
登録日2017-07-19
公開日2017-11-15
最終更新日2023-10-04
実験手法X-RAY DIFFRACTION (2.55 Å)
主引用文献Fragment-based screening identifies novel targets for inhibitors of conjugative transfer of antimicrobial resistance by plasmid pKM101.
Sci Rep, 7, 2017
5WII
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BU of 5wii by Molmil
TraE protein in complex with 2-Chloroisonicotinic Acid
分子名称: 2-chloropyridine-4-carboxylic acid, Conjugal transfer protein
著者Casu, B, Arya, T, Bessette, B, Baron, C.
登録日2017-07-19
公開日2017-11-15
最終更新日2023-10-04
実験手法X-RAY DIFFRACTION (2.79 Å)
主引用文献Fragment-based screening identifies novel targets for inhibitors of conjugative transfer of antimicrobial resistance by plasmid pKM101.
Sci Rep, 7, 2017
5WIP
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BU of 5wip by Molmil
TraE protein in complex with 2-(2-furyl)isonicotinic acid
分子名称: 2-(furan-2-yl)pyridine-4-carboxylic acid, Conjugal transfer protein
著者Casu, B, Arya, T, Bessette, B, Baron, C.
登録日2017-07-19
公開日2017-11-15
最終更新日2023-10-04
実験手法X-RAY DIFFRACTION (2.62 Å)
主引用文献Fragment-based screening identifies novel targets for inhibitors of conjugative transfer of antimicrobial resistance by plasmid pKM101.
Sci Rep, 7, 2017
6BGE
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BU of 6bge by Molmil
HELICOBACTER PYLORI ATPASE, HP0525, IN COMPLEX WITH 1G2 COMPOUND
分子名称: 4-(2-HYDROXYETHYL)-1-PIPERAZINE ETHANESULFONIC ACID, 4-[(pyridin-2-yl)oxy]benzoic acid, GLYCEROL, ...
著者Arya, T, Casu, B, Baron, C.
登録日2017-10-27
公開日2018-10-31
最終更新日2023-12-27
実験手法X-RAY DIFFRACTION (2.9 Å)
主引用文献CagAlpha in complex with hexamer inhibitor
To Be Published

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件を2024-05-01に公開中

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