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1XUF
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BU of 1xuf by Molmil
TRYPSIN-BABIM-ZN+2, PH 8.2
Descriptor: BIS(5-AMIDINO-BENZIMIDAZOLYL)METHANE ZINC, CALCIUM ION, TRYPSIN
Authors:Katz, B.A, Clark, J.M, Finer-Moore, J.S, Jenkins, T.E, Johnson, C.R, Rose, M.J, Luong, C, Moore, W.R, Stroud, R.M.
Deposit date:1997-10-10
Release date:1998-12-16
Last modified:2024-06-05
Method:X-RAY DIFFRACTION (1.9 Å)
Cite:Design of potent selective zinc-mediated serine protease inhibitors.
Nature, 391, 1998
1XUH
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BU of 1xuh by Molmil
TRYPSIN-KETO-BABIM-CO+2, PH 8.2
Descriptor: BIS(5-AMIDINO-2-BENZIMIDAZOLYL)METHANONE, CALCIUM ION, COBALT (II) ION, ...
Authors:Katz, B.A, Clark, J.M, Finer-Moore, J.S, Jenkins, T.E, Johnson, C.R, Rose, M.J, Luong, C, Moore, W.R, Stroud, R.M.
Deposit date:1997-10-10
Release date:1998-11-11
Last modified:2011-07-13
Method:X-RAY DIFFRACTION (2.2 Å)
Cite:Design of potent selective zinc-mediated serine protease inhibitors.
Nature, 391, 1998
1XUJ
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BU of 1xuj by Molmil
TRYPSIN-KETO-BABIM-ZN+2, PH 8.2
Descriptor: BIS(5-AMIDINO-BENZIMIDAZOLYL)METHANONE ZINC, CALCIUM ION, SULFATE ION, ...
Authors:Katz, B.A, Clark, J.M, Finer-Moore, J.S, Jenkins, T.E, Johnson, C.R, Rose, M.J, Luong, C, Moore, W.R, Stroud, R.M.
Deposit date:1997-10-10
Release date:1998-11-11
Last modified:2011-07-13
Method:X-RAY DIFFRACTION (1.92 Å)
Cite:Design of potent selective zinc-mediated serine protease inhibitors.
Nature, 391, 1998
1XUK
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BU of 1xuk by Molmil
TRYPSIN-BABIM-SULFATE, PH 5.9
Descriptor: BIS(5-AMIDINO-BENZIMIDAZOLYL)METHANE, CALCIUM ION, SULFATE ION, ...
Authors:Katz, B.A, Clark, J.M, Finer-Moore, J.S, Jenkins, T.E, Johnson, C.R, Rose, M.J, Luong, C, Moore, W.R, Stroud, R.M.
Deposit date:1997-10-10
Release date:1998-11-11
Last modified:2024-06-05
Method:X-RAY DIFFRACTION (1.8 Å)
Cite:Design of potent selective zinc-mediated serine protease inhibitors.
Nature, 391, 1998
1XUI
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BU of 1xui by Molmil
TRYPSIN-KETO-BABIM, ZN+2-FREE, PH 8.2
Descriptor: BIS(5-AMIDINO-2-BENZIMIDAZOLYL)METHANONE, CALCIUM ION, SODIUM ION, ...
Authors:Katz, B.A, Clark, J.M, Finer-Moore, J.S, Jenkins, T.E, Johnson, C.R, Rose, M.J, Luong, C, Moore, W.R, Stroud, R.M.
Deposit date:1997-10-10
Release date:1998-11-11
Last modified:2024-06-05
Method:X-RAY DIFFRACTION (1.5 Å)
Cite:Design of potent selective zinc-mediated serine protease inhibitors.
Nature, 391, 1998
1XUG
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BU of 1xug by Molmil
TRYPSIN-BABIM-ZN+2, PH 8.2
Descriptor: BIS(5-AMIDINO-BENZIMIDAZOLYL)METHANE, CALCIUM ION, TRYPSIN, ...
Authors:Katz, B.A, Clark, J.M, Finer-Moore, J.S, Jenkins, T.E, Johnson, C.R, Rose, M.J, Luong, C, Moore, W.R, Stroud, R.M.
Deposit date:1997-10-10
Release date:1998-12-16
Last modified:2024-06-05
Method:X-RAY DIFFRACTION (1.5 Å)
Cite:Design of potent selective zinc-mediated serine protease inhibitors.
Nature, 391, 1998
1VWA
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BU of 1vwa by Molmil
STREPTAVIDIN-FSHPQNT
Descriptor: PEPTIDE LIGAND CONTAINING HPQ, STREPTAVIDIN
Authors:Katz, B.A, Cass, R.T.
Deposit date:1997-03-03
Release date:1998-03-18
Last modified:2024-02-14
Method:X-RAY DIFFRACTION (1.85 Å)
Cite:In crystals of complexes of streptavidin with peptide ligands containing the HPQ sequence the pKa of the peptide histidine is less than 3.0.
J.Biol.Chem., 272, 1997
2RTL
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BU of 2rtl by Molmil
STREPTAVIDIN-2-IMINOBIOTIN-SULFATE COMPLEX, PH 2.50, SPACE GROUP I4122
Descriptor: 2-IMINOBIOTIN, STREPTAVIDIN, SULFATE ION
Authors:Katz, B.A.
Deposit date:1997-09-11
Release date:1998-10-14
Last modified:2024-02-21
Method:X-RAY DIFFRACTION (1.41 Å)
Cite:Binding of biotin to streptavidin stabilizes intersubunit salt bridges between Asp61 and His87 at low pH.
J.Mol.Biol., 274, 1997
1VWF
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BU of 1vwf by Molmil
STREPTAVIDIN COMPLEXED WITH CYCLO-AC-[CHPQGPPC]-NH2 MONOMER, PH 3.67
Descriptor: PEPTIDE LIGAND CONTAINING HPQ, STREPTAVIDIN
Authors:Katz, B.A, Cass, R.T.
Deposit date:1997-03-03
Release date:1998-03-18
Last modified:2024-06-05
Method:X-RAY DIFFRACTION (1.92 Å)
Cite:In crystals of complexes of streptavidin with peptide ligands containing the HPQ sequence the pKa of the peptide histidine is less than 3.0.
J.Biol.Chem., 272, 1997
1VWK
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BU of 1vwk by Molmil
STREPTAVIDIN-CYCLO-[5-S-VALERAMIDE-HPQGPPC]K-NH2
Descriptor: PENTANOIC ACID, PEPTIDE LIGAND CONTAINING HPQ, STREPTAVIDIN
Authors:Katz, B.A, Cass, R.T.
Deposit date:1997-03-03
Release date:1998-03-18
Last modified:2024-06-05
Method:X-RAY DIFFRACTION (1.45 Å)
Cite:In crystals of complexes of streptavidin with peptide ligands containing the HPQ sequence the pKa of the peptide histidine is less than 3.0.
J.Biol.Chem., 272, 1997
1VWH
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BU of 1vwh by Molmil
STREPTAVIDIN COMPLEXED WITH THE HEAD-TO-TAIL DISULFIDE-BONDED PEPTIDE DIMER OF CYCLO-AC-[CHPQGPPC]-NH2, PH 3.5
Descriptor: PEPTIDE LIGAND CONTAINING HPQ, STREPTAVIDIN
Authors:Katz, B.A, Cass, R.T.
Deposit date:1997-03-03
Release date:1998-03-18
Last modified:2024-06-05
Method:X-RAY DIFFRACTION (1.48 Å)
Cite:In crystals of complexes of streptavidin with peptide ligands containing the HPQ sequence the pKa of the peptide histidine is less than 3.0.
J.Biol.Chem., 272, 1997
1VWR
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BU of 1vwr by Molmil
STREPTAVIDIN-CYCLO-[5-S-VALERAMIDE-HPQGPPC]K-NH2, PH 3.5, I4122 COMPLEX
Descriptor: PENTANOIC ACID, PEPTIDE LIGAND CONTAINING HPQ, STREPTAVIDIN
Authors:Katz, B.A, Cass, R.T.
Deposit date:1997-03-03
Release date:1998-03-18
Last modified:2024-06-05
Method:X-RAY DIFFRACTION (1.5 Å)
Cite:In crystals of complexes of streptavidin with peptide ligands containing the HPQ sequence the pKa of the peptide histidine is less than 3.0.
J.Biol.Chem., 272, 1997
1VWI
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BU of 1vwi by Molmil
STREPTAVIDIN-CYCLO-[5-S-VALERAMIDE-HPQGPPC]K-NH2, PH 1.5, I222 COMPLEX
Descriptor: PENTANOIC ACID, PEPTIDE LIGAND CONTAINING HPQ, STREPTAVIDIN
Authors:Katz, B.A, Cass, R.T.
Deposit date:1997-03-03
Release date:1998-03-18
Last modified:2024-06-05
Method:X-RAY DIFFRACTION (1.5 Å)
Cite:In crystals of complexes of streptavidin with peptide ligands containing the HPQ sequence the pKa of the peptide histidine is less than 3.0.
J.Biol.Chem., 272, 1997
1VWP
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BU of 1vwp by Molmil
STREPTAVIDIN COMPLEXED WITH CYCLO-AC-[CHPQGPPC]-NH2 MONOMER, PH 2.5
Descriptor: PEPTIDE LIGAND CONTAINING HPQ, STREPTAVIDIN
Authors:Katz, B.A, Cass, R.T.
Deposit date:1997-03-03
Release date:1998-03-18
Last modified:2024-06-05
Method:X-RAY DIFFRACTION (1.75 Å)
Cite:In crystals of complexes of streptavidin with peptide ligands containing the HPQ sequence the pKa of the peptide histidine is less than 3.0.
J.Biol.Chem., 272, 1997
1VWQ
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BU of 1vwq by Molmil
STREPTAVIDIN-CYCLO-[5-S-VALERAMIDE-HPQGPPC]K-NH2, PH 2.5, I4122 COMPLEX
Descriptor: PENTANOIC ACID, PEPTIDE LIGAND CONTAINING HPQ, STREPTAVIDIN
Authors:Katz, B.A, Cass, R.T.
Deposit date:1997-03-03
Release date:1998-03-18
Last modified:2024-06-05
Method:X-RAY DIFFRACTION (1.7 Å)
Cite:In crystals of complexes of streptavidin with peptide ligands containing the HPQ sequence the pKa of the peptide histidine is less than 3.0.
J.Biol.Chem., 272, 1997
1VWN
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BU of 1vwn by Molmil
STREPTAVIDIN-CYCLO-AC-[CHPQFC]-NH2, PH 4.8
Descriptor: PEPTIDE LIGAND CONTAINING HPQ, STREPTAVIDIN
Authors:Katz, B.A, Cass, R.T.
Deposit date:1997-03-03
Release date:1998-03-18
Last modified:2024-06-05
Method:X-RAY DIFFRACTION (1.85 Å)
Cite:In crystals of complexes of streptavidin with peptide ligands containing the HPQ sequence the pKa of the peptide histidine is less than 3.0.
J.Biol.Chem., 272, 1997
1VWM
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BU of 1vwm by Molmil
STREPTAVIDIN-CYCLO-AC-[CHPQFC]-NH2, PH 4.2
Descriptor: PEPTIDE LIGAND CONTAINING HPQ, STREPTAVIDIN
Authors:Katz, B.A, Cass, R.T.
Deposit date:1997-03-03
Release date:1998-03-18
Last modified:2024-06-05
Method:X-RAY DIFFRACTION (1.6 Å)
Cite:In crystals of complexes of streptavidin with peptide ligands containing the HPQ sequence the pKa of the peptide histidine is less than 3.0.
J.Biol.Chem., 272, 1997
1VWG
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BU of 1vwg by Molmil
STREPTAVIDIN COMPLEXED WITH THE HEAD-TO-TAIL DISULFIDE-BONDED PEPTIDE DIMER OF CYCLO-AC-[CHPQGPPC]-NH2, PH 2.5
Descriptor: PEPTIDE LIGAND CONTAINING HPQ, STREPTAVIDIN
Authors:Katz, B.A, Cass, R.T.
Deposit date:1997-03-03
Release date:1998-03-18
Last modified:2024-06-05
Method:X-RAY DIFFRACTION (1.46 Å)
Cite:In crystals of complexes of streptavidin with peptide ligands containing the HPQ sequence the pKa of the peptide histidine is less than 3.0.
J.Biol.Chem., 272, 1997
1VWJ
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BU of 1vwj by Molmil
STREPTAVIDIN-CYCLO-[5-S-VALERAMIDE-HPQGPPC]K-NH2, PH 2.5, I222 COMPLEX
Descriptor: PENTANOIC ACID, PEPTIDE LIGAND CONTAINING HPQ, STREPTAVIDIN
Authors:Katz, B.A, Cass, R.T.
Deposit date:1997-03-03
Release date:1998-03-18
Last modified:2024-06-05
Method:X-RAY DIFFRACTION (1.45 Å)
Cite:In crystals of complexes of streptavidin with peptide ligands containing the HPQ sequence the pKa of the peptide histidine is less than 3.0.
J.Biol.Chem., 272, 1997
1VWE
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BU of 1vwe by Molmil
STREPTAVIDIN-CYCLO-AC-[CHPQFC]-NH2, PH 3.6
Descriptor: PEPTIDE LIGAND CONTAINING HPQ, STREPTAVIDIN
Authors:Katz, B.A, Cass, R.T.
Deposit date:1997-03-03
Release date:1998-03-18
Last modified:2024-06-05
Method:X-RAY DIFFRACTION (1.5 Å)
Cite:In crystals of complexes of streptavidin with peptide ligands containing the HPQ sequence the pKa of the peptide histidine is less than 3.0.
J.Biol.Chem., 272, 1997
1VWO
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BU of 1vwo by Molmil
STREPTAVIDIN COMPLEXED WITH CYCLO-AC-[CHPQGPPC]-NH2 MONOMER, PH 2.85
Descriptor: PEPTIDE LIGAND CONTAINING HPQ, STREPTAVIDIN
Authors:Katz, B.A, Cass, R.T.
Deposit date:1997-03-03
Release date:1998-03-18
Last modified:2024-06-05
Method:X-RAY DIFFRACTION (1.65 Å)
Cite:In crystals of complexes of streptavidin with peptide ligands containing the HPQ sequence the pKa of the peptide histidine is less than 3.0.
J.Biol.Chem., 272, 1997
2RTI
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BU of 2rti by Molmil
STREPTAVIDIN-GLYCOLURIL COMPLEX, PH 2.50, SPACE GROUP I222
Descriptor: FORMIC ACID, GLYCOLURIL, STREPTAVIDIN
Authors:Katz, B.A.
Deposit date:1997-09-11
Release date:1998-10-14
Last modified:2024-02-21
Method:X-RAY DIFFRACTION (1.4 Å)
Cite:Binding of biotin to streptavidin stabilizes intersubunit salt bridges between Asp61 and His87 at low pH.
J.Mol.Biol., 274, 1997
2RTD
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BU of 2rtd by Molmil
STREPTAVIDIN-BIOTIN COMPLEX, PH 1.39, SPACE GROUP I222
Descriptor: BIOTIN, STREPTAVIDIN
Authors:Katz, B.A.
Deposit date:1997-09-11
Release date:1998-10-14
Last modified:2024-02-21
Method:X-RAY DIFFRACTION (1.65 Å)
Cite:Binding of biotin to streptavidin stabilizes intersubunit salt bridges between Asp61 and His87 at low pH.
J.Mol.Biol., 274, 1997
2RTR
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BU of 2rtr by Molmil
STREPTAVIDIN-2-IMINOBIOTIN COMPLEX, PH 4.0, SPACE GROUP I222
Descriptor: 2-IMINOBIOTIN, STREPTAVIDIN
Authors:Katz, B.A.
Deposit date:1997-09-11
Release date:1998-10-14
Last modified:2024-02-21
Method:X-RAY DIFFRACTION (1.62 Å)
Cite:Binding of biotin to streptavidin stabilizes intersubunit salt bridges between Asp61 and His87 at low pH.
J.Mol.Biol., 274, 1997
1C1T
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BU of 1c1t by Molmil
RECRUITING ZINC TO MEDIATE POTENT, SPECIFIC INHIBITION OF SERINE PROTEASES
Descriptor: BIS(5-AMIDINO-BENZIMIDAZOLYL)METHANE, CALCIUM ION, MAGNESIUM ION, ...
Authors:Katz, B.A, Luong, C.
Deposit date:1999-07-21
Release date:2000-07-26
Last modified:2023-12-27
Method:X-RAY DIFFRACTION (1.37 Å)
Cite:Design of potent selective zinc-mediated serine protease inhibitors.
Nature, 391, 1998

 

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數據於2024-07-17公開中

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