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6VGL
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BU of 6vgl by Molmil
JAK2 JH1 in complex with ruxolitinib
Descriptor: (3R)-3-cyclopentyl-3-[4-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)-1H-pyrazol-1-yl]propanenitrile, Tyrosine-protein kinase JAK2
Authors:Davis, R.R, Schonbrunn, E.
Deposit date:2020-01-08
Release date:2021-01-13
Last modified:2023-11-15
Method:X-RAY DIFFRACTION (1.9 Å)
Cite:Structural Insights into JAK2 Inhibition by Ruxolitinib, Fedratinib, and Derivatives Thereof.
J.Med.Chem., 64, 2021
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數據於2024-07-24公開中

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