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8F4B
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Bovine multidrug resistance protein 1 (MRP1) bound to cyclic peptide inhibitor 1 (CPI1)
Descriptor: Cyclic peptide inhibitor 1 (CPI1), Multidrug resistance-associated protein 1
Authors:Pietz, H.L, Chen, J.
Deposit date:2022-11-10
Release date:2023-03-22
Method:ELECTRON MICROSCOPY (3.27 Å)
Cite:A macrocyclic peptide inhibitor traps MRP1 in a catalytically incompetent conformation.
Proc.Natl.Acad.Sci.USA, 120, 2023

222415

数据于2024-07-10公开中

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