English
日本語
简体中文
繁體中文
한국어
✖
Menu
RCSB PDB
PDBe
BMRB
Adv. Search
Search help
Search by PDB author
6GE0
Fragment-based discovery of a highly potent, orally bioavailable inhibitor which modulates the phosphorylation and catalytic activity of ERK1/2
Descriptor:
2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{H}-isoindol-2-yl]-~{N}-[(1~{R})-1-(3-methoxyphenyl)ethyl]ethanamide, DIMETHYL SULFOXIDE, Mitogen-activated protein kinase 1, ...
Authors:
O'Reilly, M.
Deposit date:
2018-04-25
Release date:
2018-05-30
Last modified:
2018-06-27
Method:
X-RAY DIFFRACTION (1.82 Å)
Cite:
Fragment-Based Discovery of a Potent, Orally Bioavailable Inhibitor That Modulates the Phosphorylation and Catalytic Activity of ERK1/2.
J. Med. Chem., 61, 2018
<
1
2
3
Home
首页
统计数据
帮助
FAQ
联系我们
引用PDBj / 使用条款
相关链接
Settings
数据登记 (OneDep)
帮助
Deposition to PDB, EMDB or BMRB
下载
下载PDB存档 / 快照存档
标准格式
PDBx/mmCIF Resources
格式转换
PDBx/mmCIF editor
Quick links
帮助
PDB格式不兼容数据
Group Depositions
Chemical Component entries
Latest entries
搜索
帮助
Search PDB (PDBj Mine)
Search PDBj RDB
Chemie search
Search BMRB
Sequence-Navigator
DASH
EM Navigator
Omokage search
Omokage搜索
wwPDB/RDF
RDF Portal
Status search
Molecular Viewers
帮助
jV: Graphic Viewer
Molmil: WebGL Mol. Viewer
服务&软件
帮助
Yorodumi
ASH
MAFFTash
NMRToolBox
gmfit
CRNPRED
Spanner
SFAS
HOMCOS
衍生数据库
帮助
eF-site
eF-seek
eF-surf
ProMode Elastic
hGTOP
教材
帮助
eProtS
本月的分子
Previous workshop
Games
Papermodels
关于PDBj
帮助
出版物
新闻发布 / 公共关系资源
PDBj成员
PDBj咨询委员会
个人信息保护方针
222415
数据于2024-07-10公开中