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7HN8
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BU of 7hn8 by Molmil
PanDDA analysis group deposition -- Crystal Structure of TRIM21 in complex with Z1318110042
Descriptor: 1,2-ETHANEDIOL, 4-[(but-2-yn-1-yl)(methyl)amino]-1lambda~6~-thiane-1,1-dione, E3 ubiquitin-protein ligase TRIM21, ...
Authors:Kim, Y, Marples, P, Fearon, D, von Delft, F, Knapp, S, Kraemer, A, Structural Genomics Consortium (SGC)
Deposit date:2024-11-04
Release date:2024-11-27
Method:X-RAY DIFFRACTION (1.23 Å)
Cite:PanDDA analysis group deposition
To Be Published
7HNN
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BU of 7hnn by Molmil
PanDDA analysis group deposition -- Crystal Structure of TRIM21 in complex with Z31432226
Descriptor: (azepan-1-yl)(2H-1,3-benzodioxol-5-yl)methanone, 1,2-ETHANEDIOL, E3 ubiquitin-protein ligase TRIM21, ...
Authors:Kim, Y, Marples, P, Fearon, D, von Delft, F, Knapp, S, Kraemer, A, Structural Genomics Consortium (SGC)
Deposit date:2024-11-04
Release date:2024-11-27
Method:X-RAY DIFFRACTION (1.31 Å)
Cite:PanDDA analysis group deposition
To Be Published
7HO0
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BU of 7ho0 by Molmil
PanDDA analysis group deposition -- Crystal Structure of TRIM21 in complex with Z363071686
Descriptor: 1,2-ETHANEDIOL, E3 ubiquitin-protein ligase TRIM21, N-methyl-N-[2-oxo-2-(piperidin-1-yl)ethyl]methanesulfonamide, ...
Authors:Kim, Y, Marples, P, Fearon, D, von Delft, F, Knapp, S, Kraemer, A, Structural Genomics Consortium (SGC)
Deposit date:2024-11-04
Release date:2024-11-27
Method:X-RAY DIFFRACTION (1.15 Å)
Cite:PanDDA analysis group deposition
To Be Published
7HLK
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BU of 7hlk by Molmil
PanDDA analysis group deposition -- Crystal Structure of TRIM21 in complex with Z285642082
Descriptor: 1,2-ETHANEDIOL, 4-(2-HYDROXYETHYL)-1-PIPERAZINE ETHANESULFONIC ACID, E3 ubiquitin-protein ligase TRIM21, ...
Authors:Kim, Y, Marples, P, Fearon, D, von Delft, F, Knapp, S, Kraemer, A, Structural Genomics Consortium (SGC)
Deposit date:2024-11-04
Release date:2024-11-27
Method:X-RAY DIFFRACTION (1.39 Å)
Cite:PanDDA analysis group deposition
To Be Published
7HLY
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BU of 7hly by Molmil
PanDDA analysis group deposition -- Crystal Structure of TRIM21 in complex with Z235449082
Descriptor: 1,2-ETHANEDIOL, E3 ubiquitin-protein ligase TRIM21, SULFATE ION, ...
Authors:Kim, Y, Marples, P, Fearon, D, von Delft, F, Knapp, S, Kraemer, A, Structural Genomics Consortium (SGC)
Deposit date:2024-11-04
Release date:2024-11-27
Method:X-RAY DIFFRACTION (1.32 Å)
Cite:PanDDA analysis group deposition
To Be Published
7HNA
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BU of 7hna by Molmil
PanDDA analysis group deposition -- Crystal Structure of TRIM21 in complex with Z1929757385
Descriptor: (3S)-1-(3-fluoropyridin-2-yl)-4,4-dimethylpyrrolidin-3-ol, 1,2-ETHANEDIOL, E3 ubiquitin-protein ligase TRIM21, ...
Authors:Kim, Y, Marples, P, Fearon, D, von Delft, F, Knapp, S, Kraemer, A, Structural Genomics Consortium (SGC)
Deposit date:2024-11-04
Release date:2024-11-27
Method:X-RAY DIFFRACTION (1.29 Å)
Cite:PanDDA analysis group deposition
To Be Published
7HNQ
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BU of 7hnq by Molmil
PanDDA analysis group deposition -- Crystal Structure of TRIM21 in complex with Z30620520
Descriptor: 1,2-ETHANEDIOL, 4-(2-HYDROXYETHYL)-1-PIPERAZINE ETHANESULFONIC ACID, E3 ubiquitin-protein ligase TRIM21, ...
Authors:Kim, Y, Marples, P, Fearon, D, von Delft, F, Knapp, S, Kraemer, A, Structural Genomics Consortium (SGC)
Deposit date:2024-11-04
Release date:2024-11-27
Method:X-RAY DIFFRACTION (1.37 Å)
Cite:PanDDA analysis group deposition
To Be Published
7HO4
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BU of 7ho4 by Molmil
PanDDA analysis group deposition -- Crystal Structure of TRIM21 in complex with Z1003146540
Descriptor: 1,2-ETHANEDIOL, 2-(difluoromethoxy)benzene-1-sulfonamide, E3 ubiquitin-protein ligase TRIM21, ...
Authors:Kim, Y, Marples, P, Fearon, D, von Delft, F, Knapp, S, Kraemer, A, Structural Genomics Consortium (SGC)
Deposit date:2024-11-04
Release date:2024-11-27
Method:X-RAY DIFFRACTION (1.21 Å)
Cite:PanDDA analysis group deposition
To Be Published
7HLN
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BU of 7hln by Molmil
PanDDA analysis group deposition -- Crystal Structure of TRIM21 in complex with Z26823525
Descriptor: (2S)-N-(5-ethyl-1,3,4-thiadiazol-2-yl)oxolane-2-carboxamide, 1,2-ETHANEDIOL, E3 ubiquitin-protein ligase TRIM21, ...
Authors:Kim, Y, Marples, P, Fearon, D, von Delft, F, Knapp, S, Kraemer, A, Structural Genomics Consortium (SGC)
Deposit date:2024-11-04
Release date:2024-11-27
Method:X-RAY DIFFRACTION (1.2 Å)
Cite:PanDDA analysis group deposition
To Be Published
7HLZ
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BU of 7hlz by Molmil
PanDDA analysis group deposition -- Crystal Structure of TRIM21 in complex with Z256709358
Descriptor: 1,2-ETHANEDIOL, E3 ubiquitin-protein ligase TRIM21, SULFATE ION, ...
Authors:Kim, Y, Marples, P, Fearon, D, von Delft, F, Knapp, S, Kraemer, A, Structural Genomics Consortium (SGC)
Deposit date:2024-11-04
Release date:2024-11-27
Method:X-RAY DIFFRACTION (1.29 Å)
Cite:PanDDA analysis group deposition
To Be Published
7HMA
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BU of 7hma by Molmil
PanDDA analysis group deposition -- Crystal Structure of TRIM21 in complex with Z291279160
Descriptor: 1,2-ETHANEDIOL, 1-[2-(trifluoromethyloxy)phenyl]thiourea, E3 ubiquitin-protein ligase TRIM21, ...
Authors:Kim, Y, Marples, P, Fearon, D, von Delft, F, Knapp, S, Kraemer, A, Structural Genomics Consortium (SGC)
Deposit date:2024-11-04
Release date:2024-11-27
Method:X-RAY DIFFRACTION (1.15 Å)
Cite:PanDDA analysis group deposition
To Be Published
7HMP
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BU of 7hmp by Molmil
PanDDA analysis group deposition -- Crystal Structure of TRIM21 in complex with Z1530301542
Descriptor: 1,2-ETHANEDIOL, 4-(2-HYDROXYETHYL)-1-PIPERAZINE ETHANESULFONIC ACID, 4-ethyl-2-(1H-imidazol-5-yl)-1,3-thiazole, ...
Authors:Kim, Y, Marples, P, Fearon, D, von Delft, F, Knapp, S, Kraemer, A, Structural Genomics Consortium (SGC)
Deposit date:2024-11-04
Release date:2024-11-27
Method:X-RAY DIFFRACTION (1.15 Å)
Cite:PanDDA analysis group deposition
To Be Published
7HN5
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BU of 7hn5 by Molmil
PanDDA analysis group deposition -- Crystal Structure of TRIM21 in complex with Z45617795
Descriptor: 1,2-ETHANEDIOL, E3 ubiquitin-protein ligase TRIM21, N-(2-phenylethyl)methanesulfonamide, ...
Authors:Kim, Y, Marples, P, Fearon, D, von Delft, F, Knapp, S, Kraemer, A, Structural Genomics Consortium (SGC)
Deposit date:2024-11-04
Release date:2024-11-27
Method:X-RAY DIFFRACTION (1.32 Å)
Cite:PanDDA analysis group deposition
To Be Published
7HNL
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BU of 7hnl by Molmil
PanDDA analysis group deposition -- Crystal Structure of TRIM21 in complex with Z1251207602
Descriptor: 1,2-ETHANEDIOL, 1-(5-methyl-1,3,4-thiadiazol-2-yl)piperidine, 4-(2-HYDROXYETHYL)-1-PIPERAZINE ETHANESULFONIC ACID, ...
Authors:Kim, Y, Marples, P, Fearon, D, von Delft, F, Knapp, S, Kraemer, A, Structural Genomics Consortium (SGC)
Deposit date:2024-11-04
Release date:2024-11-27
Method:X-RAY DIFFRACTION (1.44 Å)
Cite:PanDDA analysis group deposition
To Be Published
7HME
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BU of 7hme by Molmil
PanDDA analysis group deposition -- Crystal Structure of TRIM21 in complex with Z319545618
Descriptor: 1,2-ETHANEDIOL, 3-[(2-methyl-1H-imidazol-1-yl)methyl]benzonitrile, E3 ubiquitin-protein ligase TRIM21, ...
Authors:Kim, Y, Marples, P, Fearon, D, von Delft, F, Knapp, S, Kraemer, A, Structural Genomics Consortium (SGC)
Deposit date:2024-11-04
Release date:2024-11-27
Method:X-RAY DIFFRACTION (1.51 Å)
Cite:PanDDA analysis group deposition
To Be Published
5HFR
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BU of 5hfr by Molmil
Crystal structure of the second bromodomain H395R mutant of human BRD3
Descriptor: 1,2-ETHANEDIOL, Bromodomain-containing protein 3, NITRATE ION
Authors:Tallant, C, Lori, C, Pasquo, A, Chiaraluce, R, Consalvi, V, Fonseca, M, von Delft, F, Arrowsmith, C.H, Edwards, A.M, Bountra, C, Knapp, S.
Deposit date:2016-01-07
Release date:2016-01-20
Last modified:2024-01-10
Method:X-RAY DIFFRACTION (1.7 Å)
Cite:Crystal structure of the second bromodomain H395R mutant of human BRD3
To Be Published
7HMR
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BU of 7hmr by Molmil
PanDDA analysis group deposition -- Crystal Structure of TRIM21 in complex with Z1267882044
Descriptor: 1,2-ETHANEDIOL, 4-(2-HYDROXYETHYL)-1-PIPERAZINE ETHANESULFONIC ACID, E3 ubiquitin-protein ligase TRIM21, ...
Authors:Kim, Y, Marples, P, Fearon, D, von Delft, F, Knapp, S, Kraemer, A, Structural Genomics Consortium (SGC)
Deposit date:2024-11-04
Release date:2024-11-27
Method:X-RAY DIFFRACTION (1.15 Å)
Cite:PanDDA analysis group deposition
To Be Published
7HN7
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BU of 7hn7 by Molmil
PanDDA analysis group deposition -- Crystal Structure of TRIM21 in complex with Z198194396
Descriptor: 1,2-ETHANEDIOL, 4-(furan-2-carbonyl)piperazine-1-carboxamide, E3 ubiquitin-protein ligase TRIM21, ...
Authors:Kim, Y, Marples, P, Fearon, D, von Delft, F, Knapp, S, Kraemer, A, Structural Genomics Consortium (SGC)
Deposit date:2024-11-04
Release date:2024-11-27
Method:X-RAY DIFFRACTION (1.31 Å)
Cite:PanDDA analysis group deposition
To Be Published
7HNO
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BU of 7hno by Molmil
PanDDA analysis group deposition -- Crystal Structure of TRIM21 in complex with Z57450788
Descriptor: 1,2-ETHANEDIOL, E3 ubiquitin-protein ligase TRIM21, N-{4-[(morpholin-4-yl)methyl]phenyl}acetamide, ...
Authors:Kim, Y, Marples, P, Fearon, D, von Delft, F, Knapp, S, Kraemer, A, Structural Genomics Consortium (SGC)
Deposit date:2024-11-04
Release date:2024-11-27
Method:X-RAY DIFFRACTION (1.33 Å)
Cite:PanDDA analysis group deposition
To Be Published
7HO1
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BU of 7ho1 by Molmil
PanDDA analysis group deposition -- Crystal Structure of TRIM21 in complex with Z369263636
Descriptor: 1,2-ETHANEDIOL, E3 ubiquitin-protein ligase TRIM21, N-[(1R)-1-(1,5-dimethyl-1H-pyrazol-4-yl)ethyl]methanesulfonamide, ...
Authors:Kim, Y, Marples, P, Fearon, D, von Delft, F, Knapp, S, Kraemer, A, Structural Genomics Consortium (SGC)
Deposit date:2024-11-04
Release date:2024-11-27
Method:X-RAY DIFFRACTION (1.17 Å)
Cite:PanDDA analysis group deposition
To Be Published
7HO7
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BU of 7ho7 by Molmil
PanDDA analysis group deposition -- Crystal Structure of TRIM21 in complex with Z30820160
Descriptor: 1,2-ETHANEDIOL, E3 ubiquitin-protein ligase TRIM21, N-(4-methyl-1,3-thiazol-2-yl)propanamide, ...
Authors:Kim, Y, Marples, P, Fearon, D, von Delft, F, Knapp, S, Kraemer, A, Structural Genomics Consortium (SGC)
Deposit date:2024-11-04
Release date:2024-11-27
Method:X-RAY DIFFRACTION (1.3 Å)
Cite:PanDDA analysis group deposition
To Be Published
7HLM
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BU of 7hlm by Molmil
PanDDA analysis group deposition -- Crystal Structure of TRIM21 in complex with Z29077827
Descriptor: 1,2-ETHANEDIOL, E3 ubiquitin-protein ligase TRIM21, SULFATE ION, ...
Authors:Kim, Y, Marples, P, Fearon, D, von Delft, F, Knapp, S, Kraemer, A, Structural Genomics Consortium (SGC)
Deposit date:2024-11-04
Release date:2024-11-27
Method:X-RAY DIFFRACTION (1.15 Å)
Cite:PanDDA analysis group deposition
To Be Published
7HM2
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BU of 7hm2 by Molmil
PanDDA analysis group deposition -- Crystal Structure of TRIM21 in complex with Z32400357
Descriptor: 1,2-ETHANEDIOL, 1-(3-methylbenzene-1-carbonyl)piperidine-4-carboxamide, E3 ubiquitin-protein ligase TRIM21, ...
Authors:Kim, Y, Marples, P, Fearon, D, von Delft, F, Knapp, S, Kraemer, A, Structural Genomics Consortium (SGC)
Deposit date:2024-11-04
Release date:2024-11-27
Method:X-RAY DIFFRACTION (1.15 Å)
Cite:PanDDA analysis group deposition
To Be Published
7HMH
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BU of 7hmh by Molmil
PanDDA analysis group deposition -- Crystal Structure of TRIM21 in complex with Z1636723439
Descriptor: (2R)-N-methylmorpholine-2-carboxamide, 1,2-ETHANEDIOL, E3 ubiquitin-protein ligase TRIM21, ...
Authors:Kim, Y, Marples, P, Fearon, D, von Delft, F, Knapp, S, Kraemer, A, Structural Genomics Consortium (SGC)
Deposit date:2024-11-04
Release date:2024-11-27
Method:X-RAY DIFFRACTION (1.5 Å)
Cite:PanDDA analysis group deposition
To Be Published
7HLL
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BU of 7hll by Molmil
PanDDA analysis group deposition -- Crystal Structure of TRIM21 in complex with Z1328968520
Descriptor: 1,2-ETHANEDIOL, 4-[(2-methylsulfonylimidazol-1-yl)methyl]-1,3-thiazole, E3 ubiquitin-protein ligase TRIM21, ...
Authors:Kim, Y, Marples, P, Fearon, D, von Delft, F, Knapp, S, Kraemer, A, Structural Genomics Consortium (SGC)
Deposit date:2024-11-04
Release date:2024-11-27
Method:X-RAY DIFFRACTION (1.15 Å)
Cite:PanDDA analysis group deposition
To Be Published

238582

数据于2025-07-09公开中

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