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6VSN
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JAK2 JH1 in complex with BL2-110
Descriptor: (3S)-3-cyclopentyl-3-[4-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)-1H-pyrazol-1-yl]propanenitrile, Tyrosine-protein kinase JAK2
Authors:Davis, R.R, Schonbrunn, E.
Deposit date:2020-02-11
Release date:2021-02-17
Last modified:2023-11-15
Method:X-RAY DIFFRACTION (2.5 Å)
Cite:Structural Insights into JAK2 Inhibition by Ruxolitinib, Fedratinib, and Derivatives Thereof.
J.Med.Chem., 64, 2021
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数据于2024-08-28公开中

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