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2YJX
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BU of 2yjx by Molmil
Tricyclic series of Hsp90 inhibitors
Descriptor: 1-(3H-imidazo[4,5-c]pyridin-2-yl)-3,4-dihydropyrido[2,1-a]isoindol-6(2H)-one, HEAT SHOCK PROTEIN HSP 90-ALPHA
Authors:Dupuy, A, Vallee, F.
Deposit date:2011-05-24
Release date:2011-10-19
Last modified:2024-05-08
Method:X-RAY DIFFRACTION (1.83 Å)
Cite:Tricyclic Series of Heat Shock Protein 90 (Hsp90) Inhibitors Part I: Discovery of Tricyclic Imidazo[4,5-C]Pyridines as Potent Inhibitors of the Hsp90 Molecular Chaperone.
J.Med.Chem., 54, 2011
1JVG
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BU of 1jvg by Molmil
CRYSTAL STRUCTURE OF HUMAN AGX2 COMPLEXED WITH UDPGALNAC
Descriptor: GLCNAC1P URIDYLTRANSFERASE, URIDINE-DIPHOSPHATE-N-ACETYLGALACTOSAMINE
Authors:Peneff, C, Bourne, Y.
Deposit date:2001-08-30
Release date:2002-08-30
Last modified:2023-10-25
Method:X-RAY DIFFRACTION (2.3 Å)
Cite:Crystal structures of two human pyrophosphorylase isoforms in complexes with UDPGlc(Gal)NAc: role of the alternatively spliced insert in the enzyme oligomeric assembly and active site architecture.
EMBO J., 20, 2001
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