1FM0
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![BU of 1fm0 by Molmil](/molmil-images/mine/1fm0) | MOLYBDOPTERIN SYNTHASE (MOAD/MOAE) | Descriptor: | CHLORIDE ION, MOLYBDOPTERIN CONVERTING FACTOR, SUBUNIT 1, ... | Authors: | Rudolph, M.J, Wuebbens, M.M, Rajagolpalan, K.V, Schindelin, H. | Deposit date: | 2000-08-15 | Release date: | 2001-01-17 | Last modified: | 2024-02-07 | Method: | X-RAY DIFFRACTION (1.45 Å) | Cite: | Crystal structure of molybdopterin synthase and its evolutionary relationship to ubiquitin activation. Nat.Struct.Biol., 8, 2001
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1FMA
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![BU of 1fma by Molmil](/molmil-images/mine/1fma) | MOLYBDOPTERIN SYNTHASE (MOAD/MOAE) | Descriptor: | CHLORIDE ION, MOLYBDOPTERIN CONVERTING FACTOR, SUBUNIT 1, ... | Authors: | Rudolph, M.J, Wuebbens, M.M, Rajagolpalan, K.V, Schindelin, H. | Deposit date: | 2000-08-16 | Release date: | 2001-01-17 | Last modified: | 2024-02-07 | Method: | X-RAY DIFFRACTION (1.58 Å) | Cite: | Crystal structure of molybdopterin synthase and its evolutionary relationship to ubiquitin activation. Nat.Struct.Biol., 8, 2001
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2Q5W
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![BU of 2q5w by Molmil](/molmil-images/mine/2q5w) | |
4EYI
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![BU of 4eyi by Molmil](/molmil-images/mine/4eyi) | |
4OYU
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![BU of 4oyu by Molmil](/molmil-images/mine/4oyu) | Crystal structure of the N-terminal domains of muskelin | Descriptor: | 1,2-ETHANEDIOL, GLYCEROL, Muskelin | Authors: | Delto, C, Kuper, J, Schindelin, H. | Deposit date: | 2014-02-13 | Release date: | 2015-02-11 | Last modified: | 2023-12-27 | Method: | X-RAY DIFFRACTION (1.8 Å) | Cite: | The LisH Motif of Muskelin Is Crucial for Oligomerization and Governs Intracellular Localization. Structure, 23, 2015
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3QQ8
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![BU of 3qq8 by Molmil](/molmil-images/mine/3qq8) | |
4D81
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![BU of 4d81 by Molmil](/molmil-images/mine/4d81) | Metallosphera sedula Vps4 crystal structure | Descriptor: | AAA ATPase, central domain protein, ADENOSINE-5'-DIPHOSPHATE | Authors: | Caillat, C, Macheboeuf, P, Wu, Y, McCarthy, A.A, Boeri-Erba, E, Effantin, G, Gottlinger, H.G, Weissenhorn, W, Renesto, P. | Deposit date: | 2014-12-02 | Release date: | 2015-11-25 | Last modified: | 2024-05-08 | Method: | X-RAY DIFFRACTION (2.4 Å) | Cite: | Asymmetric Ring Structure of Vps4 Required for Escrt-III Disassembly. Nat.Commun., 6, 2015
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4GLJ
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![BU of 4glj by Molmil](/molmil-images/mine/4glj) | Crystal structure of methylthioadenosine phosphorylase in complex with rhodamine B | Descriptor: | CHLORIDE ION, N-[9-(2-carboxyphenyl)-6-(diethylamino)-3H-xanthen-3-ylidene]-N-ethylethanaminium, PHOSPHATE ION, ... | Authors: | Bujacz, A, Bujacz, G, Cieslinski, H, Bartasun, P. | Deposit date: | 2012-08-14 | Release date: | 2013-02-20 | Last modified: | 2023-09-13 | Method: | X-RAY DIFFRACTION (1.9 Å) | Cite: | A study on the interaction of rhodamine B with methylthioadenosine phosphorylase protein sourced from an antarctic soil metagenomic library. Plos One, 8, 2013
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5T14
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![BU of 5t14 by Molmil](/molmil-images/mine/5t14) | DNA polymerase kappa extending beyond a bulky major benzo[a]pyrene adduct | Descriptor: | 2'-deoxy-5'-O-[(R)-hydroxy{[(R)-hydroxy(phosphonooxy)phosphoryl]amino}phosphoryl]adenosine, DNA, DNA polymerase kappa, ... | Authors: | Jha, V.K, Ling, H. | Deposit date: | 2016-08-17 | Release date: | 2016-12-21 | Last modified: | 2024-03-06 | Method: | X-RAY DIFFRACTION (3 Å) | Cite: | Structural basis of accurate replication beyond a bulky major benzo[a]pyrene adduct by human DNA polymerase kappa. DNA Repair (Amst.), 49, 2017
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5T27
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![BU of 5t27 by Molmil](/molmil-images/mine/5t27) | mPI3Kd IN COMPLEX WITH 5d | Descriptor: | 3-(benzotriazol-1-yl)-5-[1-methyl-5-[(1~{S})-1-morpholin-4-ylethyl]-1,2,4-triazol-3-yl]pyrazin-2-amine, Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform | Authors: | Petersen, J, Terstige, I, Perry, M, Svensson, T, Tyrchan, C, Lindmark, H, Oster, L. | Deposit date: | 2016-08-23 | Release date: | 2017-04-19 | Last modified: | 2024-05-08 | Method: | X-RAY DIFFRACTION (2.6 Å) | Cite: | Discovery of triazole aminopyrazines as a highly potent and selective series of PI3K delta inhibitors. Bioorg. Med. Chem. Lett., 27, 2017
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5T23
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![BU of 5t23 by Molmil](/molmil-images/mine/5t23) | PI3Kg IN COMPLEX WITH 5d | Descriptor: | 3-(benzotriazol-1-yl)-5-[1-methyl-5-[(1~{S})-1-morpholin-4-ylethyl]-1,2,4-triazol-3-yl]pyrazin-2-amine, Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform | Authors: | Petersen, J, Terstige, I, Perry, M, Svensson, T, Tyrchan, C, Lindmark, H, Oster, L. | Deposit date: | 2016-08-23 | Release date: | 2017-04-19 | Last modified: | 2024-05-08 | Method: | X-RAY DIFFRACTION (2.78 Å) | Cite: | Discovery of triazole aminopyrazines as a highly potent and selective series of PI3K delta inhibitors. Bioorg. Med. Chem. Lett., 27, 2017
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5T2I
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![BU of 5t2i by Molmil](/molmil-images/mine/5t2i) | mPI3Kd IN COMPLEX WITH 7k | Descriptor: | 1-[3-azanyl-6-[1-methyl-5-(1-phenylcyclopropyl)-1,2,4-triazol-3-yl]pyrazin-2-yl]pyrazole-4-carboxamide, Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform | Authors: | Petersen, J, Terstige, I, Perry, M, Svensson, T, Tyrchan, C, Lindmark, H, Oster, L. | Deposit date: | 2016-08-23 | Release date: | 2017-04-19 | Last modified: | 2024-05-08 | Method: | X-RAY DIFFRACTION (2.3 Å) | Cite: | Discovery of triazole aminopyrazines as a highly potent and selective series of PI3K delta inhibitors. Bioorg. Med. Chem. Lett., 27, 2017
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5T2D
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![BU of 5t2d by Molmil](/molmil-images/mine/5t2d) | mPI3Kd IN COMPLEX WITH 7j | Descriptor: | 4-[3-azanyl-6-[1-methyl-5-(1-phenylcyclopropyl)-1,2,4-triazol-3-yl]pyrazin-2-yl]-~{N},~{N}-dimethyl-pyrazole-1-sulfonamide, Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform | Authors: | Petersen, J, Terstige, I, Perry, M, Svensson, T, Tyrchan, C, Lindmark, H, Oster, L. | Deposit date: | 2016-08-23 | Release date: | 2017-04-19 | Last modified: | 2024-05-08 | Method: | X-RAY DIFFRACTION (2.9 Å) | Cite: | Discovery of triazole aminopyrazines as a highly potent and selective series of PI3K delta inhibitors. Bioorg. Med. Chem. Lett., 27, 2017
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5T2M
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![BU of 5t2m by Molmil](/molmil-images/mine/5t2m) | mPI3Kd IN COMPLEX WITH 7m | Descriptor: | 4-[3-azanyl-6-[1-methyl-5-(1-phenylcyclopropyl)-1,2,4-triazol-3-yl]pyrazin-2-yl]benzamide, Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform | Authors: | Petersen, J, Terstige, I, Perry, M, Svensson, T, Tyrchan, C, Lindmark, H, Oster, L. | Deposit date: | 2016-08-23 | Release date: | 2017-04-19 | Last modified: | 2024-05-08 | Method: | X-RAY DIFFRACTION (2.8 Å) | Cite: | Discovery of triazole aminopyrazines as a highly potent and selective series of PI3K delta inhibitors. Bioorg. Med. Chem. Lett., 27, 2017
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4GLF
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![BU of 4glf by Molmil](/molmil-images/mine/4glf) | |
5T2G
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![BU of 5t2g by Molmil](/molmil-images/mine/5t2g) | mPI3Kd IN COMPLEX WITH 7i | Descriptor: | 4-[3-azanyl-6-[1-methyl-5-(1-phenylcyclopropyl)-1,2,4-triazol-3-yl]pyrazin-2-yl]pyrazole-1-carboxamide, Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform | Authors: | Petersen, J, Terstige, I, Perry, M, Svensson, T, Tyrchan, C, Lindmark, H, Oster, L. | Deposit date: | 2016-08-23 | Release date: | 2017-04-19 | Last modified: | 2024-05-08 | Method: | X-RAY DIFFRACTION (2.55 Å) | Cite: | Discovery of triazole aminopyrazines as a highly potent and selective series of PI3K delta inhibitors. Bioorg. Med. Chem. Lett., 27, 2017
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5T28
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![BU of 5t28 by Molmil](/molmil-images/mine/5t28) | mPI3Kd IN COMPLEX WITH 5k | Descriptor: | 3-(benzotriazol-1-yl)-5-[1-methyl-5-(1-phenylcyclopropyl)-1,2,4-triazol-3-yl]pyrazin-2-amine, Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform | Authors: | Petersen, J, Terstige, I, Perry, M, Svensson, T, Tyrchan, C, Lindmark, H, Oster, L. | Deposit date: | 2016-08-23 | Release date: | 2017-04-12 | Last modified: | 2024-05-08 | Method: | X-RAY DIFFRACTION (2.8 Å) | Cite: | Discovery of triazole aminopyrazines as a highly potent and selective series of PI3K delta inhibitors. Bioorg. Med. Chem. Lett., 27, 2017
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5T2L
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![BU of 5t2l by Molmil](/molmil-images/mine/5t2l) | mPI3Kd IN COMPLEX WITH 7l | Descriptor: | 1-[3-azanyl-6-[1-methyl-5-(1-phenylcyclopropyl)-1,2,4-triazol-3-yl]pyrazin-2-yl]pyrazole-3-carboxamide, Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform | Authors: | Petersen, J, Terstige, I, Perry, M, Svensson, T, Tyrchan, C, Lindmark, H, Oster, L. | Deposit date: | 2016-08-23 | Release date: | 2017-04-19 | Last modified: | 2024-05-08 | Method: | X-RAY DIFFRACTION (2.55 Å) | Cite: | Discovery of triazole aminopyrazines as a highly potent and selective series of PI3K delta inhibitors. Bioorg. Med. Chem. Lett., 27, 2017
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1CFF
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![BU of 1cff by Molmil](/molmil-images/mine/1cff) | NMR SOLUTION STRUCTURE OF A COMPLEX OF CALMODULIN WITH A BINDING PEPTIDE OF THE CA2+-PUMP | Descriptor: | CALCIUM ION, CALCIUM PUMP, CALMODULIN | Authors: | Elshorst, B, Hennig, M, Foersterling, H, Diener, A, Maurer, M, Schulte, P, Schwalbe, H, Krebs, J, Schmid, H, Vorherr, T, Carafoli, E, Griesinger, C. | Deposit date: | 1999-03-18 | Release date: | 1999-09-24 | Last modified: | 2023-12-27 | Method: | SOLUTION NMR | Cite: | NMR solution structure of a complex of calmodulin with a binding peptide of the Ca2+ pump. Biochemistry, 38, 1999
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4MT6
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![BU of 4mt6 by Molmil](/molmil-images/mine/4mt6) | |
4MT7
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![BU of 4mt7 by Molmil](/molmil-images/mine/4mt7) | Crystal structure of collybistin I | Descriptor: | Rho guanine nucleotide exchange factor 9 | Authors: | Schneeberger, D, Schindelin, H. | Deposit date: | 2013-09-19 | Release date: | 2014-08-13 | Last modified: | 2024-02-28 | Method: | X-RAY DIFFRACTION (3.5 Å) | Cite: | A conformational switch in collybistin determines the differentiation of inhibitory postsynapses. Embo J., 33, 2014
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2NQN
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![BU of 2nqn by Molmil](/molmil-images/mine/2nqn) | MoeA T100W | Descriptor: | GLYCEROL, Molybdopterin biosynthesis protein moeA | Authors: | Nicolas, J, Xiang, S, Schindelin, H, Rajagopalan, K.V. | Deposit date: | 2006-10-31 | Release date: | 2007-01-16 | Last modified: | 2023-12-27 | Method: | X-RAY DIFFRACTION (2.2 Å) | Cite: | Mutational Analysis of Escherichia coli MoeA: Two Functional Activities Map to the Active Site Cleft. Biochemistry, 46, 2007
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2NQR
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![BU of 2nqr by Molmil](/molmil-images/mine/2nqr) | MoeA D142N | Descriptor: | GLYCEROL, Molybdopterin biosynthesis protein moeA | Authors: | Nicolas, J, Xiang, S, Schindelin, H, Rajagopalan, K.V. | Deposit date: | 2006-10-31 | Release date: | 2007-01-16 | Last modified: | 2023-12-27 | Method: | X-RAY DIFFRACTION (2.2 Å) | Cite: | Mutational Analysis of Escherichia coli MoeA: Two Functional Activities Map to the Active Site Cleft. Biochemistry, 46, 2007
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2NQV
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![BU of 2nqv by Molmil](/molmil-images/mine/2nqv) | MoeA D228A | Descriptor: | GLYCEROL, Molybdopterin biosynthesis protein moeA | Authors: | Nciolas, J, Xiang, S, Schindelin, H, Rajagopalan, K.V. | Deposit date: | 2006-10-31 | Release date: | 2007-01-16 | Last modified: | 2023-12-27 | Method: | X-RAY DIFFRACTION (2.82 Å) | Cite: | Mutational Analysis of Escherichia coli MoeA: Two Functional Activities Map to the Active Site Cleft. Biochemistry, 46, 2007
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2NQS
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![BU of 2nqs by Molmil](/molmil-images/mine/2nqs) | MoeA E188A | Descriptor: | GLYCEROL, Molybdopterin biosynthesis protein moeA | Authors: | Nicolas, J, Xiang, S, Schindelin, H, Rajagopalan, K.V. | Deposit date: | 2006-10-31 | Release date: | 2007-01-16 | Last modified: | 2023-12-27 | Method: | X-RAY DIFFRACTION (2.5 Å) | Cite: | Mutational Analysis of Escherichia coli MoeA: Two Functional Activities Map to the Active Site Cleft. Biochemistry, 46, 2007
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