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CRYSTAL STRUCTURE OF THE RAT ANDROGEN RECEPTOR LIGAND BINDING DOMAIN COMPLEX WITH DIHYDROTESTOSTERONE
Descriptor:	5-ALPHA-DIHYDROTESTOSTERONE, ANDROGEN RECEPTOR
Authors:	Sack, J.S.
Deposit date:	2001-02-13
Release date:	2001-03-21
Last modified:	2023-08-09
Method:	X-RAY DIFFRACTION (2 Å)
Cite:	Crystallographic structures of the ligand-binding domains of the androgen receptor and its T877A mutant complexed with the natural agonist dihydrotestosterone. Proc.Natl.Acad.Sci.USA, 98, 2001

P38 alpha kinase complexed with a pyrazolo-triazine based inhibitor
Descriptor:	3-[(6-benzoyl-5-methylpyrrolo[2,1-f][1,2,4]triazin-4-yl)amino]-N-cyclopropyl-4-methylbenzamide, Mitogen-activated protein kinase 14
Authors:	Sack, J.S.
Deposit date:	2011-05-20
Release date:	2012-02-01
Last modified:	2024-02-28
Method:	X-RAY DIFFRACTION (2.27 Å)
Cite:	Discovery of pyrrolo[2,1-f][1,2,4]triazine C6-ketones as potent, orally active p38α MAP kinase inhibitors. Bioorg.Med.Chem.Lett., 21, 2011