5SSM
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![BU of 5ssm by Molmil](/molmil-images/mine/5ssm) | PanDDA analysis group deposition -- Crystal structure of SARS-CoV-2 NSP3 macrodomain in complex with Z5459166256 - (R,R) and (S,S) isomers | Descriptor: | (1R,2R)-1-[(1H-benzimidazole-5-carbonyl)amino]-4-hydroxy-2,3-dihydro-1H-indene-2-carboxylic acid, (1S,2S)-1-[(1H-benzimidazole-5-carbonyl)amino]-4-hydroxy-2,3-dihydro-1H-indene-2-carboxylic acid, Non-structural protein 3 | Authors: | Correy, G.J, Fraser, J.S. | Deposit date: | 2022-06-09 | Release date: | 2022-07-06 | Last modified: | 2023-09-20 | Method: | X-RAY DIFFRACTION (1.15 Å) | Cite: | Iterative computational design and crystallographic screening identifies potent inhibitors targeting the Nsp3 macrodomain of SARS-CoV-2. Proc.Natl.Acad.Sci.USA, 120, 2023
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5SS9
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5SSR
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5SRC
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![BU of 5src by Molmil](/molmil-images/mine/5src) | PanDDA analysis group deposition -- Crystal structure of SARS-CoV-2 NSP3 macrodomain in complex with Z5198562500 - (R,R) and (R,S) isomers | Descriptor: | (2R)-[(3R)-1-(7-fluoro-9H-pyrimido[4,5-b]indol-4-yl)piperidin-3-yl](hydroxy)acetic acid, (2S)-[(3R)-1-(7-fluoro-9H-pyrimido[4,5-b]indol-4-yl)piperidin-3-yl](hydroxy)acetic acid, Non-structural protein 3 | Authors: | Correy, G.J, Fraser, J.S. | Deposit date: | 2022-06-09 | Release date: | 2022-07-06 | Last modified: | 2023-09-20 | Method: | X-RAY DIFFRACTION (1.05 Å) | Cite: | Iterative computational design and crystallographic screening identifies potent inhibitors targeting the Nsp3 macrodomain of SARS-CoV-2. Proc.Natl.Acad.Sci.USA, 120, 2023
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5SRD
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5SRE
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![BU of 5sre by Molmil](/molmil-images/mine/5sre) | |
5SRF
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![BU of 5srf by Molmil](/molmil-images/mine/5srf) | |
5SRG
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![BU of 5srg by Molmil](/molmil-images/mine/5srg) | |
5SRH
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![BU of 5srh by Molmil](/molmil-images/mine/5srh) | |
5SRI
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![BU of 5sri by Molmil](/molmil-images/mine/5sri) | |
5SRJ
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5SRK
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![BU of 5srk by Molmil](/molmil-images/mine/5srk) | |
5SRL
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![BU of 5srl by Molmil](/molmil-images/mine/5srl) | |
5SRO
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![BU of 5sro by Molmil](/molmil-images/mine/5sro) | |
5SRM
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![BU of 5srm by Molmil](/molmil-images/mine/5srm) | |
5SRN
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![BU of 5srn by Molmil](/molmil-images/mine/5srn) | |
5SRP
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5SRQ
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5SRS
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![BU of 5srs by Molmil](/molmil-images/mine/5srs) | PanDDA analysis group deposition -- Crystal structure of SARS-CoV-2 NSP3 macrodomain in complex with Z2614735107 - (R) and (S) isomers | Descriptor: | 3-[(3R)-1-(7-fluoro-9H-pyrimido[4,5-b]indol-4-yl)pyrrolidin-3-yl]-1,3-oxazolidin-2-one, 3-[(3S)-1-(7-fluoro-9H-pyrimido[4,5-b]indol-4-yl)pyrrolidin-3-yl]-1,3-oxazolidin-2-one, Non-structural protein 3 | Authors: | Correy, G.J, Fraser, J.S. | Deposit date: | 2022-06-09 | Release date: | 2022-07-06 | Last modified: | 2023-09-20 | Method: | X-RAY DIFFRACTION (1.05 Å) | Cite: | Iterative computational design and crystallographic screening identifies potent inhibitors targeting the Nsp3 macrodomain of SARS-CoV-2. Proc.Natl.Acad.Sci.USA, 120, 2023
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5SRV
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5SRU
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5SRT
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5SSA
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![BU of 5ssa by Molmil](/molmil-images/mine/5ssa) | |
5SSQ
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![BU of 5ssq by Molmil](/molmil-images/mine/5ssq) | |