5SRR
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![BU of 5srr by Molmil](/molmil-images/mine/5srr) | |
5SSC
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5SRY
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5SSD
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![BU of 5ssd by Molmil](/molmil-images/mine/5ssd) | PanDDA analysis group deposition -- Crystal structure of SARS-CoV-2 NSP3 macrodomain in complex with ZINCm4000007vvRA - (R,S) isomer | Descriptor: | (1R,2S)-2-({2-[(4S)-7-methyl-8-oxo-7,8-dihydro[1,2,4]triazolo[4,3-a]pyrazin-3-yl]ethyl}carbamoyl)cyclopropane-1-carboxylic acid, Non-structural protein 3 | Authors: | Correy, G.J, Fraser, J.S. | Deposit date: | 2022-06-09 | Release date: | 2022-07-06 | Last modified: | 2023-09-20 | Method: | X-RAY DIFFRACTION (1.15 Å) | Cite: | Iterative computational design and crystallographic screening identifies potent inhibitors targeting the Nsp3 macrodomain of SARS-CoV-2. Proc.Natl.Acad.Sci.USA, 120, 2023
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5SRX
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5SSE
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5SRZ
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![BU of 5srz by Molmil](/molmil-images/mine/5srz) | PanDDA analysis group deposition -- Crystal structure of SARS-CoV-2 NSP3 macrodomain in complex with Z5281440906 - (R,S) and (S,R) isomers | Descriptor: | (1R,2S)-2-[(7-fluoro-9H-pyrimido[4,5-b]indol-4-yl)amino]cyclohexane-1-carboxylic acid, (1S,2R)-2-[(7-fluoro-9H-pyrimido[4,5-b]indol-4-yl)amino]cyclohexane-1-carboxylic acid, Non-structural protein 3 | Authors: | Correy, G.J, Fraser, J.S. | Deposit date: | 2022-06-09 | Release date: | 2022-07-06 | Last modified: | 2023-09-20 | Method: | X-RAY DIFFRACTION (1.05 Å) | Cite: | Iterative computational design and crystallographic screening identifies potent inhibitors targeting the Nsp3 macrodomain of SARS-CoV-2. Proc.Natl.Acad.Sci.USA, 120, 2023
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5SSF
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5SS0
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5SSG
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![BU of 5ssg by Molmil](/molmil-images/mine/5ssg) | |
5SS2
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5SSH
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![BU of 5ssh by Molmil](/molmil-images/mine/5ssh) | |
5SS1
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5SSI
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5SS4
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5SSJ
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5SS3
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5SSK
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5SS5
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![BU of 5ss5 by Molmil](/molmil-images/mine/5ss5) | |
5SSL
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![BU of 5ssl by Molmil](/molmil-images/mine/5ssl) | |
5SS7
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5SSN
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5SS6
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5SSO
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![BU of 5sso by Molmil](/molmil-images/mine/5sso) | |
5SS8
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![BU of 5ss8 by Molmil](/molmil-images/mine/5ss8) | |