5MHQ
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![BU of 5mhq by Molmil](/molmil-images/mine/5mhq) | CCT068127 in complex with CDK2 | 分子名称: | (2~{R},3~{S})-3-[[9-propan-2-yl-6-(pyridin-3-ylmethylamino)purin-2-yl]amino]pentan-2-ol, Cyclin-dependent kinase 2 | 著者 | Whittaker, S.R, Barlow, C, Martin, M.P, Mancusi, C, Wagner, S, Barrie, E, te Poele, R, Sharp, S, Brown, N, Wilson, S, Clarke, P, Walton, M.I, MacDonald, E, Blagg, J, Noble, M.E.M, Garrett, M.D, Workman, P. | 登録日 | 2016-11-25 | 公開日 | 2017-12-20 | 最終更新日 | 2018-03-14 | 実験手法 | X-RAY DIFFRACTION (1.3 Å) | 主引用文献 | Molecular profiling and combinatorial activity of CCT068127: a potent CDK2 and CDK9 inhibitor. Mol Oncol, 12, 2018
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1YIY
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![BU of 1yiy by Molmil](/molmil-images/mine/1yiy) | Aedes aegypti kynurenine aminotransferase | 分子名称: | 4'-DEOXY-4'-AMINOPYRIDOXAL-5'-PHOSPHATE, BROMIDE ION, kynurenine aminotransferase; glutamine transaminase K | 著者 | Han, Q, Gao, Y.G, Robinson, H, Ding, H, Wilson, S, Li, J. | 登録日 | 2005-01-13 | 公開日 | 2005-05-10 | 最終更新日 | 2023-08-23 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | Crystal structures of Aedes aegypti kynurenine aminotransferase. FEBS J., 272, 2005
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1YIZ
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![BU of 1yiz by Molmil](/molmil-images/mine/1yiz) | Aedes aegypti kynurenine aminotrasferase | 分子名称: | BROMIDE ION, kynurenine aminotransferase; glutamine transaminase | 著者 | Han, Q, Gao, Y.G, Robinson, H, Ding, H, Wilson, S, Li, J. | 登録日 | 2005-01-13 | 公開日 | 2005-05-10 | 最終更新日 | 2024-04-03 | 実験手法 | X-RAY DIFFRACTION (1.55 Å) | 主引用文献 | Crystal structures of Aedes aegypti kynurenine aminotransferase. FEBS J., 272, 2005
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1PEA
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7AEL
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![BU of 7ael by Molmil](/molmil-images/mine/7ael) | alpha 1-antitrypsin (C232S) complexed with GSK716 | 分子名称: | Alpha-1-antitrypsin, SULFATE ION, ~{N}-[(1~{S},2~{R})-1-(3-fluoranyl-2-methyl-phenyl)-1-oxidanyl-pentan-2-yl]-2-oxidanylidene-1,3-dihydroindole-4-carboxamide | 著者 | Chung, C. | 登録日 | 2020-09-17 | 公開日 | 2021-03-10 | 最終更新日 | 2024-05-01 | 実験手法 | X-RAY DIFFRACTION (1.76 Å) | 主引用文献 | Development of a small molecule that corrects misfolding and increases secretion of Z alpha 1 -antitrypsin. Embo Mol Med, 13, 2021
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6I3G
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![BU of 6i3g by Molmil](/molmil-images/mine/6i3g) | Crystal structure of a putative peptide binding protein AppA from Clostridium difficile | 分子名称: | ABC transporter, substrate-binding protein, family 5, ... | 著者 | Hughes, A.M, Wilkinson, A, Dodson, E. | 登録日 | 2018-11-06 | 公開日 | 2019-04-10 | 最終更新日 | 2024-05-15 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Crystal structure of the putative peptide-binding protein AppA from Clostridium difficile. Acta Crystallogr.,Sect.F, 75, 2019
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6VZZ
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5VEH
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![BU of 5veh by Molmil](/molmil-images/mine/5veh) | Re-refinement OF THE PDB STRUCTURE 1yiz of Aedes aegypti kynurenine aminotransferase | 分子名称: | BROMIDE ION, GLYCEROL, Kynurenine aminotransferase | 著者 | Wlodawer, A, Dauter, Z, Minor, W, Stanfield, R, Porebski, P, Jaskolski, M, Pozharski, E, Weichenberger, C.X, Rupp, B. | 登録日 | 2017-04-04 | 公開日 | 2017-11-29 | 最終更新日 | 2022-04-13 | 実験手法 | X-RAY DIFFRACTION (1.55 Å) | 主引用文献 | Detect, correct, retract: How to manage incorrect structural models. FEBS J., 285, 2018
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