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2AIV
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BU of 2aiv by Molmil
Multiple conformations in the ligand-binding site of the yeast nuclear pore targeting domain of NUP116P
分子名称: fragment of Nucleoporin NUP116/NSP116
著者Robinson, M.A, Park, S, Sun, Z.-Y.J, Silver, P, Wagner, G, Hogle, J.
登録日2005-08-01
公開日2005-08-16
最終更新日2024-05-01
実験手法SOLUTION NMR
主引用文献Multiple Conformations in the Ligand-binding Site of the Yeast Nuclear Pore-targeting Domain of Nup116p
J.Biol.Chem., 280, 2005
1YHW
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BU of 1yhw by Molmil
Crystal Structure of PAK1 kinase domain with one point mutations (K299R)
分子名称: Serine/threonine-protein kinase PAK 1
著者Lei, M, Robinson, M.A, Harrison, S.C.
登録日2005-01-10
公開日2005-05-24
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献The Active Conformation of the PAK1 Kinase Domain
Structure, 13, 2005
1YHV
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BU of 1yhv by Molmil
Crystal Structure of PAK1 kinase domain with two point mutations (K299R, T423E)
分子名称: Serine/threonine-protein kinase PAK 1
著者Lei, M, Robinson, M.A, Harrison, S.C.
登録日2005-01-10
公開日2005-05-24
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献The Active Conformation of the PAK1 Kinase Domain
Structure, 13, 2005
1JI7
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BU of 1ji7 by Molmil
Crystal Structure of TEL SAM Polymer
分子名称: ETS-RELATED PROTEIN TEL1, SULFATE ION
著者Kim, C.A, Phillips, M.L, Kim, W, Gingery, M, Tran, H.H, Robinson, M.A, Faham, S, Bowie, J.U.
登録日2001-06-29
公開日2002-07-03
最終更新日2022-12-21
実験手法X-RAY DIFFRACTION (1.45 Å)
主引用文献Polymerization of the SAM domain of TEL in leukemogenesis and transcriptional repression.
EMBO J., 20, 2001
7SVP
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BU of 7svp by Molmil
Structure of compound 34 bound to human Phospholipase D2 catalytic domain
分子名称: 1-(1-{(2S)-1-[(3R,5R)-3,5-dimethylpiperazin-1-yl]-1-oxopropan-2-yl}piperidin-4-yl)-1,3-dihydro-2H-benzimidazol-2-one, Phospholipase D2
著者Metrick, C.M, Chodaparambil, J.V.
登録日2021-11-19
公開日2023-01-25
最終更新日2023-10-25
実験手法X-RAY DIFFRACTION (2.9 Å)
主引用文献Discovery of Phospholipase D Inhibitors with Improved Drug-like Properties and Central Nervous System Penetrance.
Acs Med.Chem.Lett., 13, 2022

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件を2024-07-31に公開中

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