6B2E
 
 | | Structure of full length human AMPK (a2b2g1) in complex with a small molecule activator SC4. | | 分子名称: | 5'-AMP-activated protein kinase catalytic subunit alpha-2, 5'-AMP-activated protein kinase subunit beta-2, 5'-AMP-activated protein kinase subunit gamma-1, ... | | 著者 | Ngoei, K.R.W, Langendorf, C.G, Ling, N.X.Y, Hoque, A, Johnson, S, Camerino, M.C, Walker, S.R, Bozikis, Y.E, Dite, T.A, Ovens, A.J, Smiles, W.J, Jacobs, R, Huang, H, Parker, M.W, Scott, J.W, Rider, M.H, Kemp, B.E, Foitzik, R.C, Baell, J.B, Oakhill, J.S. | | 登録日 | 2017-09-19 | | 公開日 | 2018-04-25 | | 最終更新日 | 2023-10-04 | | 実験手法 | X-RAY DIFFRACTION (3.8 Å) | | 主引用文献 | Structural Determinants for Small-Molecule Activation of Skeletal Muscle AMPK alpha 2 beta 2 gamma 1 by the Glucose Importagog SC4.
Cell Chem Biol, 25, 2018
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6B1U
 | | Structure of full-length human AMPK (a2b1g1) in complex with a small molecule activator SC4 | | 分子名称: | 5'-AMP-activated protein kinase catalytic subunit alpha-2, 5'-AMP-activated protein kinase subunit beta-1, 5'-AMP-activated protein kinase subunit gamma-1, ... | | 著者 | Ngoei, K.R.W, Langendorf, C.G, Ling, N.X.Y, Hoque, A, Johnson, S, Camerino, M.C, Walker, S.R, Bozikis, Y.E, Dite, T.A, Ovens, A.J, Smiles, W.J, Jacobs, R, Huang, H, Parker, M.W, Scott, J.W, Rider, M.H, Kemp, B.E, Foitzik, R.C, Baell, J.B, Oakhill, J.S. | | 登録日 | 2017-09-19 | | 公開日 | 2018-04-25 | | 最終更新日 | 2023-10-04 | | 実験手法 | X-RAY DIFFRACTION (2.77 Å) | | 主引用文献 | Structural Determinants for Small-Molecule Activation of Skeletal Muscle AMPK alpha 2 beta 2 gamma 1 by the Glucose Importagog SC4.
Cell Chem Biol, 25, 2018
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1OEP
 | | Structure of Trypanosoma brucei enolase reveals the inhibitory divalent metal site | | 分子名称: | 1,2-ETHANEDIOL, ENOLASE, SULFATE ION, ... | | 著者 | Da Silva giotto, M.T, Navarro, M.V.A.S, Garratt, R.C, Rigden, D.J. | | 登録日 | 2003-03-28 | | 公開日 | 2003-04-02 | | 最終更新日 | 2023-12-13 | | 実験手法 | X-RAY DIFFRACTION (2.3 Å) | | 主引用文献 | The Crystal Structure of Trypanosoma Brucei Enolase: Visualisation of the Inhibitory Metal Binding Site III and Potential as Target for Selective, Irreversible Inhibition
J.Mol.Biol., 331, 2003
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2PTW
 | | Crystal Structure of the T. brucei enolase complexed with sulphate, identification of a metal binding site IV | | 分子名称: | 1,2-ETHANEDIOL, Enolase, SULFATE ION, ... | | 著者 | Navarro, M.V.A.S, Rigden, D.J, Garratt, R.C, Dias, S.M.G. | | 登録日 | 2007-05-08 | | 公開日 | 2007-11-20 | | 最終更新日 | 2023-08-30 | | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | | 主引用文献 | Structural flexibility in Trypanosoma brucei enolase revealed by X-ray crystallography and molecular dynamics.
Febs J., 274, 2007
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2PTZ
 | | Crystal Structure of the T. brucei enolase complexed with phosphonoacetohydroxamate (PAH), His156-out conformation | | 分子名称: | 1,2-ETHANEDIOL, Enolase, PHOSPHONOACETOHYDROXAMIC ACID, ... | | 著者 | Navarro, M.V.A.S, Rigden, D.J, Garratt, R.C, Dias, S.M.G. | | 登録日 | 2007-05-08 | | 公開日 | 2007-11-20 | | 最終更新日 | 2023-08-30 | | 実験手法 | X-RAY DIFFRACTION (1.65 Å) | | 主引用文献 | Structural flexibility in Trypanosoma brucei enolase revealed by X-ray crystallography and molecular dynamics.
Febs J., 274, 2007
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2PU0
 | | Crystal Structure of the T. brucei enolase complexed with phosphonoacetohydroxamate (PAH), His156-in conformation | | 分子名称: | 1,2-ETHANEDIOL, Enolase, PHOSPHONOACETOHYDROXAMIC ACID, ... | | 著者 | Navarro, M.V.A.S, Rigden, D.J, Garratt, R.C, Dias, S.M.G. | | 登録日 | 2007-05-08 | | 公開日 | 2007-11-20 | | 最終更新日 | 2023-08-30 | | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | | 主引用文献 | Structural flexibility in Trypanosoma brucei enolase revealed by X-ray crystallography and molecular dynamics.
Febs J., 274, 2007
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2PTY
 | | Crystal Structure of the T. brucei enolase complexed with PEP | | 分子名称: | 1,2-ETHANEDIOL, Enolase, PHOSPHOENOLPYRUVATE, ... | | 著者 | Navarro, M.V.A.S, Rigden, D.J, Garratt, R.C, Dias, S.M.G. | | 登録日 | 2007-05-08 | | 公開日 | 2007-11-20 | | 最終更新日 | 2023-08-30 | | 実験手法 | X-RAY DIFFRACTION (2 Å) | | 主引用文献 | Structural flexibility in Trypanosoma brucei enolase revealed by X-ray crystallography and molecular dynamics.
Febs J., 274, 2007
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2PTX
 | | Crystal Structure of the T. brucei enolase complexed with sulphate in closed conformation | | 分子名称: | 1,2-ETHANEDIOL, Enolase, SULFATE ION, ... | | 著者 | Navarro, M.V.A.S, Rigden, D.J, Garratt, R.C, Dias, S.M.G. | | 登録日 | 2007-05-08 | | 公開日 | 2007-11-20 | | 最終更新日 | 2023-08-30 | | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | | 主引用文献 | Structural flexibility in Trypanosoma brucei enolase revealed by X-ray crystallography and molecular dynamics.
Febs J., 274, 2007
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2PU1
 | | Crystal Structure of the T. brucei enolase complexed with Fluoro-phosphonoacetohydroxamate (FPAH) | | 分子名称: | 1,2-ETHANEDIOL, Enolase, ZINC ION, ... | | 著者 | Navarro, M.V.A.S, Rigden, D.J, Garratt, R.C, Dias, S.M.G. | | 登録日 | 2007-05-08 | | 公開日 | 2007-11-20 | | 最終更新日 | 2023-08-30 | | 実験手法 | X-RAY DIFFRACTION (1.8 Å) | | 主引用文献 | Structural flexibility in Trypanosoma brucei enolase revealed by X-ray crystallography and molecular dynamics.
Febs J., 274, 2007
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