7MP8
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![BU of 7mp8 by Molmil](/molmil-images/mine/7mp8) | |
7MP9
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![BU of 7mp9 by Molmil](/molmil-images/mine/7mp9) | Crystal structure of the cytosolic domain of Tribolium castaneum PINK1 phosphorylated at Ser205 in complex with ADP analog | 分子名称: | AMP PHOSPHORAMIDATE, MAGNESIUM ION, SULFATE ION, ... | 著者 | Rasool, S, Veyron, S, Trempe, J.F. | 登録日 | 2021-05-04 | 公開日 | 2021-12-01 | 最終更新日 | 2023-10-18 | 実験手法 | X-RAY DIFFRACTION (2.8 Å) | 主引用文献 | Mechanism of PINK1 activation by autophosphorylation and insights into assembly on the TOM complex. Mol.Cell, 82, 2022
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8UDC
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![BU of 8udc by Molmil](/molmil-images/mine/8udc) | Crystal structure of TcPINK1 in complex with CYC116 | 分子名称: | (4P)-4-(2-amino-4-methyl-1,3-thiazol-5-yl)-N-[4-(morpholin-4-yl)phenyl]pyrimidin-2-amine, DI(HYDROXYETHYL)ETHER, SULFATE ION, ... | 著者 | Veyron, S, Rasool, S, Trempe, J.F. | 登録日 | 2023-09-28 | 公開日 | 2024-04-17 | 実験手法 | X-RAY DIFFRACTION (3.1 Å) | 主引用文献 | Structural Characterization of a small-molecule inhibitor of PINK1, a precursor tool compound for the study of Parkinson's disease To Be Published
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8UCT
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![BU of 8uct by Molmil](/molmil-images/mine/8uct) | Crystal structure of TcPINK1 in complex with PRT | 分子名称: | 2,3-DIHYDROXY-1,4-DITHIOBUTANE, 2-{[(1R,2S)-2-aminocyclohexyl]amino}-4-{[3-(2H-1,2,3-triazol-2-yl)phenyl]amino}pyrimidine-5-carboxamide, SULFATE ION, ... | 著者 | Veyron, S, Rasool, S, Trempe, J.F. | 登録日 | 2023-09-27 | 公開日 | 2024-05-08 | 実験手法 | X-RAY DIFFRACTION (2.93 Å) | 主引用文献 | Characterization of a new family of PINK1 inhibitors To Be Published
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4ZYN
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![BU of 4zyn by Molmil](/molmil-images/mine/4zyn) | Crystal Structure of Parkin E3 ubiquitin ligase (linker deletion; delta 86-130) | 分子名称: | E3 ubiquitin-protein ligase parkin, SULFATE ION, ZINC ION | 著者 | Lilov, A, Sauve, V, Trempe, J.F, Rodionov, D, Wang, J, Gehring, K. | 登録日 | 2015-05-21 | 公開日 | 2015-08-19 | 最終更新日 | 2023-09-27 | 実験手法 | X-RAY DIFFRACTION (2.54 Å) | 主引用文献 | A Ubl/ubiquitin switch in the activation of Parkin. Embo J., 34, 2015
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