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1BSJ
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BU of 1bsj by Molmil
COBALT DEFORMYLASE INHIBITOR COMPLEX FROM E.COLI
分子名称: (S)-2-(PHOSPHONOXY)CAPROYL-L-LEUCYL-P-NITROANILIDE, COBALT (II) ION, PHOSPHATE ION, ...
著者Hao, B, Gong, W, Rajagopalan, P.T, Hu, Y, Pei, D, Chan, M.K.
登録日1998-08-28
公開日2000-04-15
最終更新日2023-08-09
実験手法X-RAY DIFFRACTION (3 Å)
主引用文献Structural basis for the design of antibiotics targeting peptide deformylase.
Biochemistry, 38, 1999
1BSK
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BU of 1bsk by Molmil
ZINC DEFORMYLASE INHIBITOR COMPLEX FROM E.COLI
分子名称: (S)-2-(PHOSPHONOXY)CAPROYL-L-LEUCYL-P-NITROANILIDE, PHOSPHATE ION, PROTEIN (PEPTIDE DEFORMYLASE), ...
著者Hao, B, Gong, W, Rajagopalan, P.T, Hu, Y, Pei, D, Chan, M.K.
登録日1998-08-28
公開日2000-04-15
最終更新日2023-08-09
実験手法X-RAY DIFFRACTION (3 Å)
主引用文献Structural basis for the design of antibiotics targeting peptide deformylase.
Biochemistry, 38, 1999
1DFF
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BU of 1dff by Molmil
PEPTIDE DEFORMYLASE
分子名称: PEPTIDE DEFORMYLASE, ZINC ION
著者Chan, M.K, Gong, W, Rajagopalan, P.T.R, Hao, B, Tsai, C.M, Pei, D.
登録日1997-08-19
公開日1998-09-02
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (2.88 Å)
主引用文献Crystal structure of the Escherichia coli peptide deformylase.
Biochemistry, 36, 1997
3H98
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BU of 3h98 by Molmil
Crystal structure of HCV NS5b 1b with (1,1-dioxo-2H-[1,2,4]benzothiadiazin-3-yl) azolo[1,5-a]pyrimidine derivative
分子名称: GLYCEROL, N-{3-[5-hydroxy-8-(3-methylbutyl)-7-oxo-7,8-dihydroimidazo[1,2-a]pyrimidin-6-yl]-1,1-dioxido-4H-1,2,4-benzothiadiazin-7-yl}methanesulfonamide, RNA-directed RNA polymerase
著者Wang, G, Lei, H, Wang, X, Das, D, Mackinnon, C, Montalbetti, C.A.G, Mears, R, Gai, X, Bailey, S, Ruhrmund, D, Hooi, L, Misialek, S, Rajagopalan, R, Cheng, R.K.Y, Barker, J.L, Felicetti, B, Stoycheva, A, Buckman, B, Kossen, K, Seiwert, S, Beigelmana, L.
登録日2009-04-30
公開日2009-10-13
最終更新日2023-09-06
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献HCV NS5B polymerase inhibitors 2: Synthesis and in vitro activity of (1,1-dioxo-2H-[1,2,4]benzothiadiazin-3-yl) azolo[1,5-a]pyridine and azolo[1,5-a]pyrimidine derivatives.
Bioorg.Med.Chem.Lett., 19, 2009

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