Search by PDB author

Crystal structure of N-((2S)-5-(6-fluoro-3-pyridinyl)-2,3-dihydro-1H- inden-2-yl)-2-propanesulfonamide in complex with the ligand binding domain of the human GluA2 receptor
分子名称:	GLUTAMATE RECEPTOR 2, GLUTAMIC ACID, N-[(2S)-5-(6-FLUORO-3-PYRIDINYL)-2,3-DIHYDRO-1H-INDEN-2-YL]-2-PROPANESULFONAMIDE, ...
著者	Ward, S.E, Harries, M, Aldegheri, L, Andreotti, D, Ballantine, S, Bax, B.D, Harris, A.J, Harker, A.J, Lund, J, Melarange, R, Mingardi, A, Mookherjee, C, Mosley, J, Neve, M, Oliosi, B, Profeta, R, Smith, K.J, Smith, P.W, Spada, S, Thewlis, K.M, Yusaf, S.P.
登録日	2010-06-14
公開日	2010-07-21
最終更新日	2011-07-13
実験手法	X-RAY DIFFRACTION (1.8 Å)
主引用文献	Discovery of N-[(2S)-5-(6-Fluoro-3-Pyridinyl)-2,3-Dihydro-1H-Inden-2-Yl]-2-Propanesulfonamide, a Novel Clinical Ampa Receptor Positive Modulator. J.Med.Chem., 53, 2010

2.7A structure of benzoisoxazole 3 with S.aureus DNA gyrase and DNA.
分子名称:	(2~{R})-2-[[5-(2-chlorophenyl)-1,2-benzoxazol-3-yl]oxy]-2-phenyl-ethanamine, CHLORIDE ION, DNA (5'-D(APGPCPCPGPTPAPGPGPTPAPCPCPTPAPCPGPGPCPT)-3'), ...
著者	Bax, B.D.
登録日	2019-03-06
公開日	2019-04-17
最終更新日	2024-01-24
実験手法	X-RAY DIFFRACTION (2.65 Å)
主引用文献	Structure-guided design of antibacterials that allosterically inhibit DNA gyrase. Bioorg.Med.Chem.Lett., 29, 2019

3.4A structure of benzoisoxazole 3 with S.aureus DNA gyrase and DNA
分子名称:	(2~{R})-2-[[5-(2-chlorophenyl)-1,2-benzoxazol-3-yl]oxy]-2-phenyl-ethanamine, DNA (5'-D(GPAPGPCPGPTPAPCPGPGPCPCPGPTPAPCPGPCPTPT)-3'), DNA gyrase subunit A, ...
著者	Bax, B.D.
登録日	2019-03-06
公開日	2019-04-17
最終更新日	2024-01-24
実験手法	X-RAY DIFFRACTION (3.4 Å)
主引用文献	Structure-guided design of antibacterials that allosterically inhibit DNA gyrase. Bioorg.Med.Chem.Lett., 29, 2019