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7M16
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Triazole-based BET family bromodomain inhibitor bound to BRD4(D1)
分子名称: 4-{5-[6-(3,5-dimethylanilino)pyridin-2-yl]-4-methyl-1H-1,2,3-triazol-1-yl}piperidine-1-carboximidamide, Bromodomain-containing protein 4
著者Johnson, J.A, Pomerantz, W.
登録日2021-03-12
公開日2021-09-29
最終更新日2023-10-18
実験手法X-RAY DIFFRACTION (1.42 Å)
主引用文献Systematically Mitigating the p38alpha Activity of Triazole-based BET Inhibitors
ACS Med. Chem. Lett., 10, 2019

223790

件を2024-08-14に公開中

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