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5V68
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BU of 5v68 by Molmil
Crystal structure of cell division protein FtsZ from Mycobacterium tuberculosis bounded via the T9 loop
分子名称: Cell division protein FtsZ, GUANOSINE-5'-DIPHOSPHATE, PHOSPHATE ION
著者Lazo, E.O, Ojima, I, Chowdhury, S.R, Awasthi, D, Jakoncic, J.
登録日2017-03-16
公開日2017-03-29
最終更新日2023-10-04
実験手法X-RAY DIFFRACTION (3.46 Å)
主引用文献Novel T9 loop conformation of filamenting temperature-sensitive mutant Z from Mycobacterium tuberculosis.
Acta Crystallogr.,Sect.F, 75, 2019
4AZN
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BU of 4azn by Molmil
Murine epidermal fatty acid-binding protein (FABP5), apo form, poly- his tag-mediated crystal packing
分子名称: FATTY ACID-BINDING PROTEIN, EPIDERMAL
著者Sanson, B, Wang, T, Sun, J, Kaczocha, M, Ojima, I, Deutsch, D, Li, H.
登録日2012-06-26
公開日2013-08-07
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (2.51 Å)
主引用文献Crystallographic Study of Fabp5 as an Intracellular Endocannabinoid Transporter.
Acta Crystallogr.,Sect.D, 70, 2014
4AZO
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BU of 4azo by Molmil
Murine epidermal fatty acid-binding protein (FABP5), apo form, poly- his tag removed
分子名称: CHLORIDE ION, FATTY ACID-BINDING PROTEIN, EPIDERMAL
著者Sanson, B, Wang, T, Sun, J, Kaczocha, M, Ojima, I, Deutsch, D, Li, H.
登録日2012-06-26
公開日2013-08-07
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (2.33 Å)
主引用文献Crystallographic Study of Fabp5 as an Intracellular Endocannabinoid Transporter.
Acta Crystallogr.,Sect.D, 70, 2014
4AZQ
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BU of 4azq by Molmil
Murine epidermal fatty acid-binding protein (FABP5) in complex with the endocannabinoid 2-arachidonoylglycerol
分子名称: 2-hydroxy-1-(hydroxymethyl)ethyl icosanoate, CHLORIDE ION, FATTY ACID-BINDING PROTEIN, ...
著者Sanson, B, Wang, T, Sun, J, Kaczocha, M, Ojima, I, Deutsch, D, Li, H.
登録日2012-06-26
公開日2013-08-14
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Crystallographic Study of Fabp5 as an Intracellular Endocannabinoid Transporter.
Acta Crystallogr.,Sect.D, 70, 2014
4AZM
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BU of 4azm by Molmil
Human epidermal fatty acid-binding protein (FABP5) in complex with the inhibitor BMS-309413
分子名称: ((2'-(5-ETHYL-3,4-DIPHENYL-1H-PYRAZOL-1-YL)-3-BIPHENYLYL)OXY)ACETIC ACID, FATTY ACID-BINDING PROTEIN, EPIDERMAL, ...
著者Sanson, B, Wang, T, Sun, J, Kaczocha, M, Ojima, I, Deutsch, D, Li, H.
登録日2012-06-26
公開日2013-08-07
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (2.75 Å)
主引用文献Crystallographic Study of Fabp5 as an Intracellular Endocannabinoid Transporter.
Acta Crystallogr.,Sect.D, 70, 2014
4AZP
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BU of 4azp by Molmil
Murine epidermal fatty acid-binding protein (FABP5) in complex with the endocannabinoid anandamide
分子名称: CHLORIDE ION, FATTY ACID-BINDING PROTEIN, EPIDERMAL, ...
著者Sanson, B, Wang, T, Sun, J, Kaczocha, M, Ojima, I, Deutsch, D, Li, H.
登録日2012-06-26
公開日2013-08-07
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献Crystallographic Study of Fabp5 as an Intracellular Endocannabinoid Transporter.
Acta Crystallogr.,Sect.D, 70, 2014
4AZR
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BU of 4azr by Molmil
Human epidermal fatty acid-binding protein (FABP5) in complex with the endocannabinoid anandamide
分子名称: CHLORIDE ION, FATTY ACID-BINDING PROTEIN, EPIDERMAL, ...
著者Sanson, B, Wang, T, Sun, J, Kaczocha, M, Ojima, I, Deutsch, D, Li, H.
登録日2012-06-26
公開日2013-08-07
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (2.95 Å)
主引用文献Crystallographic Study of Fabp5 as an Intracellular Endocannabinoid Transporter.
Acta Crystallogr.,Sect.D, 70, 2014
5UR9
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BU of 5ur9 by Molmil
Enantiomer-Specific Binding of the Potent Antinociceptive Agent SBFI-26 to Anandamide transporters FABP5
分子名称: (1S,2S,3S,4S)-3-{[(naphthalen-1-yl)oxy]carbonyl}-2,4-diphenylcyclobutane-1-carboxylic acid, Fatty acid-binding protein, epidermal, ...
著者Hsu, H.-C, Li, H.
登録日2017-02-09
公開日2017-08-23
最終更新日2023-10-04
実験手法X-RAY DIFFRACTION (2.19800353 Å)
主引用文献The Antinociceptive Agent SBFI-26 Binds to Anandamide Transporters FABP5 and FABP7 at Two Different Sites.
Biochemistry, 56, 2017
8EXD
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BU of 8exd by Molmil
Crystal structure of Aspergillus fumigatus sterylglucosidase A
分子名称: Sterylglucosidase A (SglA)
著者Pereira de Sa, N, Del Poeta, M, Airola, M.V.
登録日2022-10-25
公開日2023-03-01
最終更新日2023-10-25
実験手法X-RAY DIFFRACTION (3.8 Å)
主引用文献Targeting Sterylglucosidase A to Treat Aspergillus fumigatus Infections.
Mbio, 14, 2023
6AQ1
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BU of 6aq1 by Molmil
The crystal structure of human FABP3
分子名称: Fatty acid-binding protein, heart, PALMITIC ACID, ...
著者Hsu, H.C, Li, H.
登録日2017-08-18
公開日2018-06-13
最終更新日2023-10-04
実験手法X-RAY DIFFRACTION (1.40000093 Å)
主引用文献SAR studies on truxillic acid mono esters as a new class of antinociceptive agents targeting fatty acid binding proteins.
Eur J Med Chem, 154, 2018
5URA
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BU of 5ura by Molmil
Enantiomer-Specific Binding of the Potent Antinociceptive Agent SBFI-26 to Anandamide transporters FABP7
分子名称: (1S,2S,3S,4S)-3-{[(naphthalen-1-yl)oxy]carbonyl}-2,4-diphenylcyclobutane-1-carboxylic acid, Fatty acid-binding protein, brain, ...
著者Hsu, H.-C, Li, H.
登録日2017-02-09
公開日2017-08-23
最終更新日2023-10-04
実験手法X-RAY DIFFRACTION (1.85002172 Å)
主引用文献The Antinociceptive Agent SBFI-26 Binds to Anandamide Transporters FABP5 and FABP7 at Two Different Sites.
Biochemistry, 56, 2017
7LPQ
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BU of 7lpq by Molmil
Crystal structure of Cryptococcus neoformans sterylglucosidase 1 with hit 9
分子名称: Cytoplasmic protein, GLYCEROL, MAGNESIUM ION, ...
著者Pereira de Sa, N, Del Poeta, M, Airola, M.V.
登録日2021-02-12
公開日2021-09-01
最終更新日2023-10-18
実験手法X-RAY DIFFRACTION (2.32 Å)
主引用文献Structure and inhibition of Cryptococcus neoformans sterylglucosidase to develop antifungal agents.
Nat Commun, 12, 2021
7LPO
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BU of 7lpo by Molmil
Crystal structure of Cryptococcus neoformans sterylglucosidase 1 with tris
分子名称: 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, Cytoplasmic protein, MAGNESIUM ION
著者Pereira de Sa, N, Del Poeta, M, Airola, M.V.
登録日2021-02-12
公開日2021-09-01
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (2.13 Å)
主引用文献Structure and inhibition of Cryptococcus neoformans sterylglucosidase to develop antifungal agents.
Nat Commun, 12, 2021
7LPP
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BU of 7lpp by Molmil
Crystal structure of Cryptococcus neoformans sterylglucosidase 1 with hit 1
分子名称: 4-(hydroxymethyl)-1-[[2-(3-methoxyphenyl)-1,3-thiazol-5-yl]methyl]piperidin-4-ol, Cytoplasmic protein, GLYCEROL, ...
著者Pereira de Sa, N, Del Poeta, M, Airola, M.V.
登録日2021-02-12
公開日2021-09-01
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (2.85 Å)
主引用文献Structure and inhibition of Cryptococcus neoformans sterylglucosidase to develop antifungal agents.
Nat Commun, 12, 2021
2Q1Y
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BU of 2q1y by Molmil
Crystal Structure of cell division protein FtsZ from Mycobacterium tuberculosis in complex with GTP-gamma-S
分子名称: 5'-GUANOSINE-DIPHOSPHATE-MONOTHIOPHOSPHATE, Cell division protein ftsZ
著者Truglio, J.J.
登録日2007-05-25
公開日2008-05-06
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Identification of FtsZ Polymerization Regulatory Elements Using a Mycobacterium tuberculosis FtsZ Temperature Sensitive Mutant
To be Published
2Q1X
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BU of 2q1x by Molmil
Crystal Structure of cell division protein FtsZ from Mycobacterium tuberculosis in complex with citrate.
分子名称: CITRIC ACID, Cell division protein ftsZ
著者Truglio, J.J.
登録日2007-05-25
公開日2008-05-06
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (2.35 Å)
主引用文献Identification of FtsZ Polymerization Regulatory Elements Using a Mycobacterium tuberculosis FtsZ Temperature Sensitive Mutant
To be Published
8WMD
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BU of 8wmd by Molmil
Structure of the SARS-CoV-2 EG.5.1 spike glycoprotein (closed-2 state)
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, Spike glycoprotein
著者Nomai, T, Anraku, Y, Kita, S, Hashiguchi, T, Maenaka, K.
登録日2023-10-03
公開日2024-04-24
最終更新日2024-07-17
実験手法ELECTRON MICROSCOPY (2.71 Å)
主引用文献Virological characteristics of the SARS-CoV-2 Omicron EG.5.1 variant.
Microbiol Immunol, 2024
8WMF
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BU of 8wmf by Molmil
Structure of the SARS-CoV-2 EG.5.1 spike glycoprotein (closed-1 state)
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, Spike glycoprotein
著者Nomai, T, Anraku, Y, Kita, S, Hashiguchi, T, Maenaka, K.
登録日2023-10-03
公開日2024-04-24
最終更新日2024-07-17
実験手法ELECTRON MICROSCOPY (2.51 Å)
主引用文献Virological characteristics of the SARS-CoV-2 Omicron EG.5.1 variant.
Microbiol Immunol, 2024
8XLM
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BU of 8xlm by Molmil
Structure of the SARS-CoV-2 EG.5.1 spike glycoprotein in complex with ACE2 (1-up state)
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, Processed angiotensin-converting enzyme 2, ...
著者Nomai, T, Anraku, Y, Kita, S, Hashiguchi, T, Maenaka, K.
登録日2023-12-26
公開日2024-05-01
最終更新日2024-07-17
実験手法ELECTRON MICROSCOPY (3.22 Å)
主引用文献Virological characteristics of the SARS-CoV-2 Omicron EG.5.1 variant.
Microbiol Immunol, 2024
8XLN
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BU of 8xln by Molmil
Structure of the SARS-CoV-2 EG.5.1 spike RBD in complex with ACE2
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, Processed angiotensin-converting enzyme 2, ...
著者Nomai, T, Anraku, Y, Kita, S, Hashiguchi, T, Maenaka, K.
登録日2023-12-26
公開日2024-05-01
最終更新日2024-07-17
実験手法ELECTRON MICROSCOPY (3.78 Å)
主引用文献Virological characteristics of the SARS-CoV-2 Omicron EG.5.1 variant.
Microbiol Immunol, 2024

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件を2024-07-24に公開中

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