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5XSO
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BU of 5xso by Molmil
Crystal structure of full-length FixJ from B. japonicum crystallized in space group C2221
分子名称: FORMIC ACID, GLYCEROL, Response regulator FixJ
著者Nishizono, Y, Hisano, T, Sawai, H, Shiro, Y, Nakamura, H, Wright, G.S.A, Saeki, A, Hikima, T, Yamamoto, M, Antonyuk, S.V, Hasnain, S.S.
登録日2017-06-14
公開日2018-05-23
最終更新日2024-03-27
実験手法X-RAY DIFFRACTION (1.778 Å)
主引用文献Architecture of the complete oxygen-sensing FixL-FixJ two-component signal transduction system.
Sci Signal, 11, 2018
5XT2
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BU of 5xt2 by Molmil
Crystal structures of full-length FixJ from B. japonicum crystallized in space group P212121
分子名称: FORMIC ACID, GLYCEROL, MAGNESIUM ION, ...
著者Nishizono, Y, Hisano, T, Shiro, Y, Sawai, H, Wright, G.S.A, Saeki, A, Hikima, T, Nakamura, H, Yamamoto, M, Antonyuk, S.V, Hasnain, S.S.
登録日2017-06-16
公開日2018-05-23
最終更新日2024-03-27
実験手法X-RAY DIFFRACTION (2.652 Å)
主引用文献Architecture of the complete oxygen-sensing FixL-FixJ two-component signal transduction system.
Sci Signal, 11, 2018
8X6R
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BU of 8x6r by Molmil
KRasG12C in complex with inhibitor
分子名称: 1-[7-[6-ethenyl-8-ethoxy-7-(5-methyl-1~{H}-indazol-4-yl)-2-(1-methylpiperidin-4-yl)oxy-quinazolin-4-yl]-2,7-diazaspiro[3.5]nonan-2-yl]propan-1-one, GUANOSINE-5'-DIPHOSPHATE, Isoform 2B of GTPase KRas, ...
著者Amano, Y, Tateishi, Y.
登録日2023-11-21
公開日2024-01-17
実験手法X-RAY DIFFRACTION (1.85 Å)
主引用文献Discovery of ASP6918, a KRAS G12C inhibitor: Synthesis and structure-activity relationships of 1-{2,7-diazaspiro[3.5]non-2-yl}prop-2-en-1-one derivatives as covalent inhibitors with good potency and oral activity for the treatment of solid tumors.
Bioorg.Med.Chem., 98, 2023
8JS7
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BU of 8js7 by Molmil
Dimeric PAS domains of oxygen sensor FixL in complex with imidazole-bound heme
分子名称: GLYCEROL, IMIDAZOLE, PROTOPORPHYRIN IX CONTAINING FE, ...
著者Kamaya, M, Koteishi, H, Sawai, H, Sugimoto, H, Shiro, Y.
登録日2023-06-19
公開日2024-06-26
実験手法X-RAY DIFFRACTION (2.85 Å)
主引用文献Dimeric PAS domains of oxygen sensor FixL in complex with imidazole-bound heme.
To be published
8JS5
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BU of 8js5 by Molmil
Dimeric PAS domains of oxygen sensor FixL with ferric unliganded heme
分子名称: GLYCEROL, PROTOPORPHYRIN IX CONTAINING FE, Sensor protein FixL
著者Kamaya, M, Koteishi, H, Sawai, H, Sugimoto, H, Shiro, Y.
登録日2023-06-19
公開日2024-06-26
実験手法X-RAY DIFFRACTION (2.95 Å)
主引用文献Dimeric PAS domains of oxygen sensor FixL in complex with imidazole-bound heme.
To be published
8JS6
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BU of 8js6 by Molmil
Dimeric PAS domains of oxygen sensor FixL in complex with cyanide-bound ferric heme
分子名称: CYANIDE ION, GLYCEROL, PROTOPORPHYRIN IX CONTAINING FE, ...
著者Kamaya, M, Koteishi, H, Sawai, H, Sugimoto, H, Shiro, Y.
登録日2023-06-19
公開日2024-06-26
実験手法X-RAY DIFFRACTION (2.7 Å)
主引用文献Dimeric PAS domains of oxygen sensor FixL in complex with imidazole-bound heme.
To be published

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件を2024-07-24に公開中

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