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5U9N
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BU of 5u9n by Molmil
Second Bromodomain of cdg4_1340 from Cryptosporidium parvum, complexed with bromosporine
分子名称: Bromo domain containing protein, Bromosporine, SULFATE ION
著者Hou, C.F.D, Lin, Y.H, Loppnau, P, Hutchinson, A, Dong, A, Bountra, C, Edwards, A.M, Arrowsmith, C.H, Hui, R, Walker, J.R, Structural Genomics Consortium (SGC)
登録日2016-12-16
公開日2017-01-18
最終更新日2023-10-04
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献Second Bromodomain of cdg4_1340 from Cryptosporidium parvum, complexed with bromosporine
To be published
5VS7
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BU of 5vs7 by Molmil
Bromodomain of PF3D7_1475600 from Plasmodium falciparum complexed with peptide H4K5ac
分子名称: Bromodomain protein, putative, CHLORIDE ION, ...
著者Hou, C.F.D, Loppnau, P, Dong, A, Bountra, C, Edwards, A.M, Arrowsmith, C.H, Hui, R, Walker, J.R, Structural Genomics Consortium (SGC)
登録日2017-05-11
公開日2017-05-31
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (2.04 Å)
主引用文献Bromodomain of PF3D7_1475600 from Plasmodium falciparum complexed with peptide H4K5ac
To be published
5FEA
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BU of 5fea by Molmil
Domain Swapped Bromodomain from Leishmania donovani
分子名称: BROMIDE ION, Bromosporine, Uncharacterized protein
著者Walker, J.R, Hou, C.F.D, Lin, Y.H, LOPPNAU, P, Dong, A, El Bakkouri, M, Bountra, C, Edwards, A.M, Arrowsmith, C.H, Hui, R, Structural Genomics Consortium (SGC)
登録日2015-12-16
公開日2016-01-13
最終更新日2023-09-27
実験手法X-RAY DIFFRACTION (2.6 Å)
主引用文献Domain Swapped Bromodomain from Leishmania donovani
To be published
5K29
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BU of 5k29 by Molmil
Trypanosoma brucei bromodomain BDF5 (Tb427tmp.01.5000)
分子名称: UNKNOWN ATOM OR ION, uncharacterized protein BDF5
著者Lin, Y.H, Tempel, W, Walker, J.R, Loppnau, P, Amani, M, Hou, C.F.D, Arrowsmith, C.H, Edwards, A.M, Bountra, C, Weigelt, J, Hui, R, Structural Genomics Consortium (SGC)
登録日2016-05-18
公開日2016-07-13
最終更新日2016-11-02
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献Trypanosoma brucei bromodomain BDF5 (Tb427tmp.01.5000)
To Be Published
5KO4
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BU of 5ko4 by Molmil
Bromodomain from Trypanosoma brucei Tb427.10.8150
分子名称: Putative uncharacterized protein, SULFATE ION
著者El Bakkouri, M, Walker, J.R, Hou, C.F.D, Lin, Y.H, Bountra, C, Edwards, A.M, Arrowsmith, C.H, Hui, R, Structural Genomics Consortium (SGC)
登録日2016-06-29
公開日2016-08-31
最終更新日2023-09-27
実験手法X-RAY DIFFRACTION (1.44 Å)
主引用文献Bromodomain from Trypanosoma brucei Tb427.10.8150
To be published
5TCM
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BU of 5tcm by Molmil
First Bromodomain from Leishmania donovani LdBPK.091320 complexed with BI-2536
分子名称: 1,2-ETHANEDIOL, 4-{[(7R)-8-cyclopentyl-7-ethyl-5-methyl-6-oxo-5,6,7,8-tetrahydropteridin-2-yl]amino}-3-methoxy-N-(1-methylpiperidin-4-yl)benzamide, Uncharacterized protein
著者Lin, Y.H, Hou, C.F.D, Loppnau, P, Dong, A, Bountra, C, Edwards, A.M, Arrowsmith, C.H, Hui, R, Walker, J.R, Structural Genomics Consortium (SGC)
登録日2016-09-15
公開日2016-10-05
最終更新日2023-10-04
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献First Bromodomain from Leishmania donovani LdBPK.091320 complexed with BI-2536
To be published
5TCK
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BU of 5tck by Molmil
Second Bromodomain from Leishmania donovani LdBPK.091320 complexed with Bromosporine
分子名称: 1,2-ETHANEDIOL, BETA-MERCAPTOETHANOL, Bromosporine, ...
著者Lin, L.-H, Hou, C.F.D, Loppnau, P, Dong, A, Bountra, C, Edwards, A.M, Arrowsmith, C.H, Hui, R, Walker, J.R, Structural Genomics Consortium (SGC)
登録日2016-09-15
公開日2016-11-09
最終更新日2018-01-24
実験手法X-RAY DIFFRACTION (1.95 Å)
主引用文献Second Bromodomain from Leishmania donovani LdBPK.091320 complexed with Bromosporine
To Be Published
5C8G
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BU of 5c8g by Molmil
Crystal Structure Analysis of PP-BRD20 from Tb427tmp complexed with BI-2536
分子名称: 4-{[(7R)-8-cyclopentyl-7-ethyl-5-methyl-6-oxo-5,6,7,8-tetrahydropteridin-2-yl]amino}-3-methoxy-N-(1-methylpiperidin-4-yl)benzamide, PP-BRD20, UNKNOWN ATOM OR ION
著者Jiang, D.Q, Tempel, W, Loppnau, P, Graslund, S, Hou, C.F.D, El Bakkouri, M, Arrowsmith, C.H, Edwards, A.M, Bountra, C, Hui, R, Amain, M, Lin, Y.H, Structural Genomics Consortium (SGC)
登録日2015-06-25
公開日2015-07-22
最終更新日2023-09-27
実験手法X-RAY DIFFRACTION (1.95 Å)
主引用文献Crystal Structure Analysis of PP-BRD20 from Tb427tmp
to be published
5C4Q
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BU of 5c4q by Molmil
Crystal Structure Analysis of bromodomain from Leishmania donovani complexed with bromosporine
分子名称: Bromodomain, Bromosporine, UNKNOWN ATOM OR ION
著者Jiang, D.Q, Tempel, W, Loppnau, P, Graslund, S, Arrowsmith, C.H, Edwards, A.M, Bountra, C, Hui, R, Amani, M, Hou, C.F.D, Structural Genomics Consortium (SGC)
登録日2015-06-18
公開日2015-07-08
最終更新日2023-09-27
実験手法X-RAY DIFFRACTION (1.932 Å)
主引用文献Crystal Structure Analysis of bromodomain from Leishmania donovani complexed with bromosporine
to be published
5CZG
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BU of 5czg by Molmil
Crystal Structure Analysis of hypothetical bromodomain Tb427.10.7420 from Trypanosoma brucei in complex with bromosporine
分子名称: Bromosporine, Hypothetical Bromodomain, SODIUM ION, ...
著者Jiang, D.Q, Tempel, W, Loppnau, P, Graslund, S, Arrowsmith, C.H, Edwards, A.M, Bountra, C, Hui, R, Amani, M, Hou, C.F.D, Structural Genomics Consortium (SGC)
登録日2015-07-31
公開日2015-08-12
最終更新日2023-09-27
実験手法X-RAY DIFFRACTION (1.451 Å)
主引用文献Crystal Structure Analysis of hypothetical bromodomain from Trypanosoma brucei
to be published
7SYA
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BU of 7sya by Molmil
Kinetically trapped Pseudomonas-phage PaP3 portal protein - Full Length
分子名称: Portal protein
著者Hou, C.F.D, Swanson, N.A, Li, F, Yang, R, Lokareddy, R.K, Cingolani, G.
登録日2021-11-24
公開日2022-04-20
最終更新日2024-02-28
実験手法ELECTRON MICROSCOPY (3.5 Å)
主引用文献Cryo-EM Structure of a Kinetically Trapped Dodecameric Portal Protein from the Pseudomonas-phage PaP3.
J.Mol.Biol., 434, 2022
7SXK
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BU of 7sxk by Molmil
Kinetically trapped Pseudomonas-phage PaP3 portal protein - Full Length
分子名称: Portal protein
著者Hou, C.F.D, Swanson, N.A, Li, F, Yang, R, Lokareddy, R.K, Cingolani, G.
登録日2021-11-23
公開日2022-04-20
実験手法ELECTRON MICROSCOPY (3.4 Å)
主引用文献Cryo-EM Structure of a Kinetically Trapped Dodecameric Portal Protein from the Pseudomonas-phage PaP3.
J.Mol.Biol., 434, 2022
5TPX
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BU of 5tpx by Molmil
Bromodomain from Plasmodium Faciparum Gcn5, complexed with compound
分子名称: (1S,2S)-N~1~,N~1~-dimethyl-N~2~-(3-methyl[1,2,4]triazolo[3,4-a]phthalazin-6-yl)-1-phenylpropane-1,2-diamine, CHLORIDE ION, Histone acetyltransferase GCN5, ...
著者Lin, Y.H, Hou, C.F.D, MOUSTAKIM, M, DIXON, D.J, Loppnau, P, Tempel, W, Bountra, C, Edwards, A.M, Arrowsmith, C.H, Hui, R, BRENNAN, P.E, Walker, J.R, Structural Genomics Consortium (SGC)
登録日2016-10-21
公開日2017-01-04
最終更新日2023-10-04
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献Discovery of a PCAF Bromodomain Chemical Probe.
Angew. Chem. Int. Ed. Engl., 56, 2017

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件を2024-07-03に公開中

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