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4Z7Y
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BU of 4z7y by Molmil
diphosphomevalonate decarboxylase from the Sulfolobus solfataricus, space group P21
分子名称: Diphosphomevalonate decarboxylase, SULFATE ION
著者Hattori, A, Unno, H, Hemmi, H.
登録日2015-04-08
公開日2015-09-16
最終更新日2023-11-08
実験手法X-RAY DIFFRACTION (2.7 Å)
主引用文献In Vivo Formation of the Protein Disulfide Bond That Enhances the Thermostability of Diphosphomevalonate Decarboxylase, an Intracellular Enzyme from the Hyperthermophilic Archaeon Sulfolobus solfataricus
J.Bacteriol., 197, 2015
4Z7C
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BU of 4z7c by Molmil
Diphosphomevalonate decarboxylase from the Sulfolobus solfataricus, space group h32
分子名称: Diphosphomevalonate decarboxylase, GLYCEROL, PHOSPHATE ION, ...
著者Unno, H, Hattori, A, Hemmi, H.
登録日2015-04-07
公開日2015-09-16
最終更新日2023-11-08
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献In Vivo Formation of the Protein Disulfide Bond That Enhances the Thermostability of Diphosphomevalonate Decarboxylase, an Intracellular Enzyme from the Hyperthermophilic Archaeon Sulfolobus solfataricus
J.Bacteriol., 197, 2015
5GMD
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BU of 5gmd by Molmil
Crystal structure of Sulfolobus solfataricus diphosphomevalonate decarboxylase in complex with ATP-gamma-S
分子名称: (3R)-3-HYDROXY-5-{[(R)-HYDROXY(PHOSPHONOOXY)PHOSPHORYL]OXY}-3-METHYLPENTANOIC ACID, ADENOSINE MONOPHOSPHATE, Diphosphomevalonate decarboxylase, ...
著者Unno, H, Hemmi, H, Hattori, A.
登録日2016-07-13
公開日2016-12-28
最終更新日2023-11-08
実験手法X-RAY DIFFRACTION (1.5 Å)
主引用文献A Single Amino Acid Mutation Converts (R)-5-Diphosphomevalonate Decarboxylase into a Kinase
J. Biol. Chem., 292, 2017
5GME
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BU of 5gme by Molmil
Crystal structure of Sulfolobus solfataricus Diphosphomevalonate decarboxylase in complex with ADP
分子名称: (3R)-3-HYDROXY-5-{[(R)-HYDROXY(PHOSPHONOOXY)PHOSPHORYL]OXY}-3-METHYLPENTANOIC ACID, ADENOSINE MONOPHOSPHATE, ADENOSINE-5'-DIPHOSPHATE, ...
著者Unno, H, Hemmi, H, Hattori, A.
登録日2016-07-13
公開日2016-12-28
最終更新日2023-11-08
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献A Single Amino Acid Mutation Converts (R)-5-Diphosphomevalonate Decarboxylase into a Kinase
J. Biol. Chem., 292, 2017
6IO0
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BU of 6io0 by Molmil
Human IDH1 R132C mutant complexed with compound A.
分子名称: (2E)-3-{3-[3-(2,6-dichlorophenyl)-5-(propan-2-yl)-1,2-oxazole-4-carbonyl]-1-methyl-1H-indol-7-yl}prop-2-enoic acid, CITRIC ACID, GLYCEROL, ...
著者Suzuki, M, Baba, D, Hanzawa, H.
登録日2018-10-29
公開日2019-10-30
最終更新日2024-03-27
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献A Potent Blood-Brain Barrier-Permeable Mutant IDH1 Inhibitor Suppresses the Growth of Glioblastoma with IDH1 Mutation in a Patient-Derived Orthotopic Xenograft Model.
Mol.Cancer Ther., 19, 2020

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件を2024-06-12に公開中

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