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Crystal structure of p38alpha with an allosteric inhibitor 2
分子名称:	Mitogen-activated protein kinase 14, ~{N}-(5,6-dimethoxy-1,3-benzothiazol-2-yl)-2-[(4-fluoranylphenoxy)methyl]-1,3-thiazole-4-carboxamide
著者	Hasegawa, S, Kinoshita, T.
登録日	2023-11-14
公開日	2024-11-20
最終更新日	2025-03-05
実験手法	X-RAY DIFFRACTION (1.85 Å)
主引用文献	Distinct binding modes of a benzothiazole derivative confer structural bases for increasing ERK2 or p38 alpha MAPK selectivity. Biochem.Biophys.Res.Commun., 704, 2024

Crystal structure of p38alpha with an allosteric inhibitor 3
分子名称:	13-[4-({Imidazo[1,2-a]pyridin-2-yl}methoxy)phenyl]-4,8-dioxa-12,14,16,18-tetraazatetracyclo[9.7.0.0^{3,9}.0^{12,17}]octadeca-1(11),2,9,15,17-pentaen-15-amine, GLYCEROL, Mitogen-activated protein kinase 14
著者	Hasegawa, S, Kinoshita, T.
登録日	2024-02-19
公開日	2025-02-26
実験手法	X-RAY DIFFRACTION (1.66 Å)
主引用文献	Identification of a novel target site for ATP-independent p38 alpha inhibitors To Be Published