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1SCD
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BU of 1scd by Molmil
X-RAY CRYSTAL STRUCTURE OF CROSS-LINKED SUBTILISM CARLSBERG IN WATER VS. ACETONITRILE
分子名称: CALCIUM ION, SUBTILISIN CARLSBERG
著者Fitzpatrick, P.A, Ringe, D, Klibanov, A.M.
登録日1993-08-23
公開日1994-01-31
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献X-ray crystal structure of cross-linked subtilisin Carlsberg in water vs. acetonitrile.
Biochem.Biophys.Res.Commun., 198, 1994
1SCA
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BU of 1sca by Molmil
ENZYME CRYSTAL STRUCTURE IN A NEAT ORGANIC SOLVENT
分子名称: CALCIUM ION, SODIUM ION, SUBTILISIN CARLSBERG
著者Fitzpatrick, P.A, Steinmetz, A.C.U, Ringe, D, Klibanov, A.M.
登録日1993-07-19
公開日1994-01-31
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Enzyme crystal structure in a neat organic solvent.
Proc.Natl.Acad.Sci.USA, 90, 1993
1SCB
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BU of 1scb by Molmil
ENZYME CRYSTAL STRUCTURE IN A NEAT ORGANIC SOLVENT
分子名称: ACETONITRILE, CALCIUM ION, SUBTILISIN CARLSBERG
著者Fitzpatrick, P.A, Steinmetz, A.C.U, Ringe, D, Klibanov, A.M.
登録日1993-07-13
公開日1994-01-31
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Enzyme crystal structure in a neat organic solvent.
Proc.Natl.Acad.Sci.USA, 90, 1993
3VSB
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BU of 3vsb by Molmil
SUBTILISIN CARLSBERG D-NAPHTHYL-1-ACETAMIDO BORONIC ACID INHIBITOR COMPLEX
分子名称: SODIUM ION, SUBTILISIN CARLSBERG, TYPE VIII
著者Stoll, V.S, Eger, B.T, Hynes, R.C, Martichonok, V, Jones, J.B, Pai, E.F.
登録日1997-09-25
公開日1998-03-25
最終更新日2023-08-09
実験手法X-RAY DIFFRACTION (2.6 Å)
主引用文献Differences in binding modes of enantiomers of 1-acetamido boronic acid based protease inhibitors: crystal structures of gamma-chymotrypsin and subtilisin Carlsberg complexes.
Biochemistry, 37, 1998
4PJV
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BU of 4pjv by Molmil
Structure of PARP2 catalytic domain bound to inhibitor BMN 673
分子名称: (8S,9R)-5-fluoro-8-(4-fluorophenyl)-9-(1-methyl-1H-1,2,4-triazol-5-yl)-2,7,8,9-tetrahydro-3H-pyrido[4,3,2-de]phthalazin-3-one, GLYCEROL, Poly [ADP-ribose] polymerase 2
著者Aoyagi-Scharber, M, Gardberg, A.S, Edwards, T.L.
登録日2014-05-12
公開日2014-09-24
最終更新日2023-09-27
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献Structural basis for the inhibition of poly(ADP-ribose) polymerases 1 and 2 by BMN 673, a potent inhibitor derived from dihydropyridophthalazinone.
Acta Crystallogr.,Sect.F, 70, 2014
4PJT
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BU of 4pjt by Molmil
Structure of PARP1 catalytic domain bound to inhibitor BMN 673
分子名称: (8S,9R)-5-fluoro-8-(4-fluorophenyl)-9-(1-methyl-1H-1,2,4-triazol-5-yl)-2,7,8,9-tetrahydro-3H-pyrido[4,3,2-de]phthalazin-3-one, GLYCEROL, Poly [ADP-ribose] polymerase 1, ...
著者Aoyagi-Scharber, M, Gardberg, A.S, Arakaki, T.L.
登録日2014-05-12
公開日2014-09-24
最終更新日2023-09-27
実験手法X-RAY DIFFRACTION (2.35 Å)
主引用文献Structural basis for the inhibition of poly(ADP-ribose) polymerases 1 and 2 by BMN 673, a potent inhibitor derived from dihydropyridophthalazinone.
Acta Crystallogr.,Sect.F, 70, 2014
1AVT
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BU of 1avt by Molmil
SUBTILISIN CARLSBERG D-PARA-CHLOROPHENYL-1-ACETAMIDO BORONIC ACID INHIBITOR COMPLEX
分子名称: SODIUM ION, SUBTILISIN CARLSBERG, TYPE VIII
著者Stoll, V.S, Eger, B.T, Hynes, R.C, Martichonok, V, Jones, J.B, Pai, E.F.
登録日1997-09-19
公開日1998-03-25
最終更新日2023-08-02
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Differences in binding modes of enantiomers of 1-acetamido boronic acid based protease inhibitors: crystal structures of gamma-chymotrypsin and subtilisin Carlsberg complexes.
Biochemistry, 37, 1998
1AV7
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BU of 1av7 by Molmil
SUBTILISIN CARLSBERG L-NAPHTHYL-1-ACETAMIDO BORONIC ACID INHIBITOR COMPLEX
分子名称: SODIUM ION, SUBTILISIN CARLSBERG, TYPE VIII
著者Stoll, V.S, Eger, B.T, Hynes, R.C, Martichonok, V, Jones, J.B, Pai, E.F.
登録日1997-09-29
公開日1998-04-01
最終更新日2023-08-02
実験手法X-RAY DIFFRACTION (2.6 Å)
主引用文献Differences in binding modes of enantiomers of 1-acetamido boronic acid based protease inhibitors: crystal structures of gamma-chymotrypsin and subtilisin Carlsberg complexes.
Biochemistry, 37, 1998
1VSB
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BU of 1vsb by Molmil
SUBTILISIN CARLSBERG L-PARA-CHLOROPHENYL-1-ACETAMIDO BORONIC ACID INHIBITOR COMPLEX
分子名称: SUBTILISIN CARLSBERG, TYPE VIII
著者Stoll, V.S, Eger, B.T, Hynes, R.C, Martichonok, V, Jones, J.B, Pai, E.F.
登録日1997-09-17
公開日1998-03-18
最終更新日2023-08-09
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献Differences in binding modes of enantiomers of 1-acetamido boronic acid based protease inhibitors: crystal structures of gamma-chymotrypsin and subtilisin Carlsberg complexes.
Biochemistry, 37, 1998

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