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7UEK
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BU of 7uek by Molmil
Crystal structure of a de novo designed ovoid TIM barrel OT3
分子名称: OT3
著者Chu, A.E, Fernandez, D, Huang, P.-S.
登録日2022-03-21
公開日2023-01-18
最終更新日2024-04-03
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献De Novo Design of a Highly Stable Ovoid TIM Barrel: Unlocking Pocket Shape towards Functional Design.
Biodes Res, 2022, 2022
7RAA
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BU of 7raa by Molmil
Designed StabIL-2 seq15
分子名称: Interleukin-2, MAGNESIUM ION
著者Jude, K.M, Chu, A.E, Huang, P.-S, Garcia, K.C.
登録日2021-06-30
公開日2022-03-16
最終更新日2024-04-03
実験手法X-RAY DIFFRACTION (2.69 Å)
主引用文献Interleukin-2 superkines by computational design.
Proc.Natl.Acad.Sci.USA, 119, 2022
7RA9
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BU of 7ra9 by Molmil
Designed StabIL-2 seq1
分子名称: 4-(2-HYDROXYETHYL)-1-PIPERAZINE ETHANESULFONIC ACID, Interleukin-2, PHOSPHATE ION
著者Jude, K.M, Chu, A.E, Huang, P.-S, Garcia, K.C.
登録日2021-06-30
公開日2022-03-16
最終更新日2023-10-25
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Interleukin-2 superkines by computational design.
Proc.Natl.Acad.Sci.USA, 119, 2022
7KCH
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BU of 7kch by Molmil
Myosin XI-F-actin complex
分子名称: ADENOSINE-5'-DIPHOSPHATE, Actin, alpha skeletal muscle, ...
著者Gong, R, Alushin, G.M.
登録日2020-10-05
公開日2021-01-13
最終更新日2024-03-06
実験手法ELECTRON MICROSCOPY (4.33 Å)
主引用文献Optical control of fast and processive engineered myosins in vitro and in living cells.
Nat.Chem.Biol., 17, 2021
8TCE
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BU of 8tce by Molmil
Lipoprotein(a) Kringle IV domain 8 - Lp(a) KIV8 in complex with LY3353871
分子名称: (2S)-3-phenyl-2-[(3R)-pyrrolidin-3-yl]propanoic acid, Apolipoprotein(a)
著者Hendle, J, Weichert, K, Sauder, J.M.
登録日2023-06-30
公開日2024-05-08
最終更新日2024-06-19
実験手法X-RAY DIFFRACTION (1.07 Å)
主引用文献Discovery of potent small-molecule inhibitors of lipoprotein(a) formation.
Nature, 629, 2024
8V9B
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BU of 8v9b by Molmil
Lipoprotein(a) Kringle IV domain 7 - Lp(a) KIV7 in complex with LY3441732
分子名称: (2S,2'S)-3,3'-[carbonylbis(azanediyl-3,1-phenylene)]bis{2-[(3R)-pyrrolidin-1-ium-3-yl]propanoate}, Apolipoprotein(a), MAGNESIUM ION, ...
著者Hendle, J, Weichert, K, Sauder, J.M.
登録日2023-12-07
公開日2024-05-08
最終更新日2024-06-19
実験手法X-RAY DIFFRACTION (1.19 Å)
主引用文献Discovery of potent small-molecule inhibitors of lipoprotein(a) formation.
Nature, 629, 2024
8V8Z
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BU of 8v8z by Molmil
Lipoprotein(a) Kringle IV domain 8 - Lp(a) KIV8 in complex with LY3473329
分子名称: Apolipoprotein(a), muvalaplin
著者Hendle, J, Weichert, K, Sauder, J.M.
登録日2023-12-06
公開日2024-05-08
最終更新日2024-06-19
実験手法X-RAY DIFFRACTION (2.01 Å)
主引用文献Discovery of potent small-molecule inhibitors of lipoprotein(a) formation.
Nature, 629, 2024

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件を2024-09-11に公開中

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