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1ME4
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BU of 1me4 by Molmil
High Resolution Crystal Structure Analysis Of Cruzain non-covalently Bound To A Hydroxymethyl Ketone Inhibitor (I)
分子名称: CRUZIPAIN, [1-(1-BENZYL-3-HYDROXY-2-OXO-PROPYLCARBAMOYL)-2-PHENYL-ETHYL]-CARBAMIC ACID BENZYL ESTER
著者Brinen, L.S, Huang, L, Ellman, J.A.
登録日2002-08-07
公開日2002-12-18
最終更新日2017-10-11
実験手法X-RAY DIFFRACTION (1.2 Å)
主引用文献Crystal Structures of Reversible Ketone-based Inhibitors of the Cysteine Protease Cruzain
Bioorg.Med.Chem., 11, 2003
1ST3
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BU of 1st3 by Molmil
THE CRYSTAL STRUCTURE OF THE BACILLUS LENTUS ALKALINE PROTEASE, SUBTILISIN BL, AT 1.4 ANGSTROMS RESOLUTION
分子名称: CALCIUM ION, SUBTILISIN BL
著者Goddette, D.W.
登録日1991-11-22
公開日1994-01-31
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (1.4 Å)
主引用文献The crystal structure of the Bacillus lentus alkaline protease, subtilisin BL, at 1.4 A resolution.
J.Mol.Biol., 228, 1992
1AK5
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BU of 1ak5 by Molmil
INOSINE MONOPHOSPHATE DEHYDROGENASE (IMPDH) FROM TRITRICHOMONAS FOETUS
分子名称: INOSINE-5'-MONOPHOSPHATE DEHYDROGENASE, SULFATE ION
著者Whitby, F.G.
登録日1997-05-28
公開日1997-09-17
最終更新日2011-07-13
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Crystal structure of Tritrichomonas foetus inosine-5'-monophosphate dehydrogenase and the enzyme-product complex.
Biochemistry, 36, 1997
1EWP
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BU of 1ewp by Molmil
CRUZAIN BOUND TO MOR-LEU-HPQ
分子名称: CRUZAIN, N-[(3S)-1-fluoro-2-oxo-5-phenylpentan-3-yl]-N~2~-(morpholin-4-ylcarbonyl)-L-leucinamide
著者Gillmor, S.A.
登録日2000-04-26
公開日2000-05-17
最終更新日2024-03-13
実験手法X-RAY DIFFRACTION (1.75 Å)
主引用文献Chapter 3: X-ray Structures of Complexes of Cruzain with Designed Covalent Inhibitors
Enzyme-ligand Interactions, Inhibition and Specificity, 1998
1AMH
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BU of 1amh by Molmil
UNCOMPLEXED RAT TRYPSIN MUTANT WITH ASP 189 REPLACED WITH SER (D189S)
分子名称: ANIONIC TRYPSIN, CALCIUM ION
著者Szabo, E, Bocskei, Z.S, Naray-Szabo, G, Graf, L.
登録日1997-06-17
公開日1997-12-24
最終更新日2023-08-02
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献The three-dimensional structure of Asp189Ser trypsin provides evidence for an inherent structural plasticity of the protease.
Eur.J.Biochem., 263, 1999
1DPO
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BU of 1dpo by Molmil
STRUCTURE OF RAT TRYPSIN
分子名称: BENZAMIDINE, CALCIUM ION, SULFATE ION, ...
著者Stroud, R.M.
登録日1997-03-31
公開日1997-07-07
最終更新日2021-11-03
実験手法X-RAY DIFFRACTION (1.59 Å)
主引用文献1.59 A structure of trypsin at 120 K: comparison of low temperature and room temperature structures.
Proteins, 10, 1991

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