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5S9E
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BU of 5s9e by Molmil
PanDDA analysis group deposition -- Crystal Structure of PHIP in complex with Z198194396 synthetic derivative
分子名称: 4-(5-methylfuran-2-carbonyl)-N-[(pyridin-3-yl)methyl]piperazine-1-carboxamide, PH-interacting protein
著者Grosjean, H, Aimon, A, Hassel-Hart , S, Krojer, T, Talon, R, Douangamath, A, Koekemoer, L, Biggin, P.C, Spencer, J, von Delft, F.
登録日2021-01-22
公開日2021-02-17
最終更新日2024-03-06
実験手法X-RAY DIFFRACTION (1.18 Å)
主引用文献Crystal Structures of the second bromodomain of Pleckstrin homology domain interacting protein (PHIP) in space group C2 soaked with crude reaction mixtures
To Be Published
5S9C
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BU of 5s9c by Molmil
PanDDA analysis group deposition -- Crystal Structure of PHIP in complex with Z198194396 synthetic derivative
分子名称: N-(cyclopropylmethyl)-4-(thiophene-2-carbonyl)piperazine-1-carboxamide, PH-interacting protein
著者Grosjean, H, Aimon, A, Hassel-Hart , S, Krojer, T, Talon, R, Douangamath, A, Koekemoer, L, Biggin, P.C, Spencer, J, von Delft, F.
登録日2021-01-22
公開日2021-02-17
最終更新日2024-03-06
実験手法X-RAY DIFFRACTION (1.14 Å)
主引用文献Crystal Structures of the second bromodomain of Pleckstrin homology domain interacting protein (PHIP) in space group C2 soaked with crude reaction mixtures
To Be Published
5S99
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BU of 5s99 by Molmil
PanDDA analysis group deposition -- Crystal Structure of PHIP in complex with starting material
分子名称: 2,3-dihydrothieno[3,4-b][1,4]dioxine-5-carboxylic acid, PH-interacting protein
著者Grosjean, H, Aimon, A, Hassel-Hart , S, Krojer, T, Talon, R, Douangamath, A, Koekemoer, L, Biggin, P.C, Spencer, J, von Delft, F.
登録日2021-01-22
公開日2021-02-17
最終更新日2024-03-06
実験手法X-RAY DIFFRACTION (1.18 Å)
主引用文献Crystal Structures of the second bromodomain of Pleckstrin homology domain interacting protein (PHIP) in space group C2 soaked with crude reaction mixtures
To Be Published
5S9B
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BU of 5s9b by Molmil
PanDDA analysis group deposition -- Crystal Structure of PHIP in complex withstarting material
分子名称: 3-methoxybenzoic acid, PH-interacting protein
著者Grosjean, H, Aimon, A, Hassel-Hart , S, Krojer, T, Talon, R, Douangamath, A, Koekemoer, L, Biggin, P.C, Spencer, J, von Delft, F.
登録日2021-01-22
公開日2021-02-17
最終更新日2024-03-06
実験手法X-RAY DIFFRACTION (1.153 Å)
主引用文献Crystal Structures of the second bromodomain of Pleckstrin homology domain interacting protein (PHIP) in space group C2 soaked with crude reaction mixtures
To Be Published
5S9A
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BU of 5s9a by Molmil
PanDDA analysis group deposition -- Crystal Structure of PHIP in complex with Z198194396 synthetic derivative
分子名称: 4-(5-chlorofuran-2-carbonyl)-N-(2,2,2-trifluoroethyl)piperazine-1-carboxamide, PH-interacting protein
著者Grosjean, H, Aimon, A, Hassel-Hart , S, Krojer, T, Talon, R, Douangamath, A, Koekemoer, L, Biggin, P.C, Spencer, J, von Delft, F.
登録日2021-01-22
公開日2021-02-17
最終更新日2024-03-06
実験手法X-RAY DIFFRACTION (1.36 Å)
主引用文献Crystal Structures of the second bromodomain of Pleckstrin homology domain interacting protein (PHIP) in space group C2 soaked with crude reaction mixtures
To Be Published
5S9G
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BU of 5s9g by Molmil
PanDDA analysis group deposition -- Crystal Structure of PHIP in complex with starting material
分子名称: 1,3-benzothiazole-6-carboxylic acid, PH-interacting protein
著者Grosjean, H, Aimon, A, Hassel-Hart , S, Krojer, T, Talon, R, Douangamath, A, Koekemoer, L, Biggin, P.C, Spencer, J, von Delft, F.
登録日2021-01-22
公開日2021-02-17
最終更新日2024-03-06
実験手法X-RAY DIFFRACTION (1.091 Å)
主引用文献Crystal Structures of the second bromodomain of Pleckstrin homology domain interacting protein (PHIP) in space group C2 soaked with crude reaction mixtures
To Be Published
5S9J
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BU of 5s9j by Molmil
PanDDA analysis group deposition -- Crystal Structure of PHIP in complex with starting material
分子名称: 2-azanyl-3-methyl-benzoic acid, PH-interacting protein
著者Grosjean, H, Aimon, A, Hassel-Hart , S, Krojer, T, Talon, R, Douangamath, A, Koekemoer, L, Biggin, P.C, Spencer, J, von Delft, F.
登録日2021-01-22
公開日2021-02-17
最終更新日2024-03-06
実験手法X-RAY DIFFRACTION (1.15 Å)
主引用文献Crystal Structures of the second bromodomain of Pleckstrin homology domain interacting protein (PHIP) in space group C2 soaked with crude reaction mixtures
To Be Published
7FV1
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BU of 7fv1 by Molmil
PanDDA analysis group deposition -- PHIP in complex with Z4912742920
分子名称: PH-interacting protein, tert-butyl [3-({[4-(furan-2-carbonyl)piperazine-1-carbonyl]amino}methyl)phenyl]carbamate
著者Grosjean, H, Tomlinson, C, Bradshaw, W.J, Koekemoer, L, Krojer, T, Fearon, D, Biggin, P.C, von Delft, F.
登録日2023-03-09
公開日2023-03-29
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (1.19 Å)
主引用文献PanDDA analysis group deposition
To Be Published
7FVG
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BU of 7fvg by Molmil
PanDDA analysis group deposition -- PHIP in complex with Z992453336
分子名称: N-(4-methoxyphenyl)-4-(5-methylfuran-2-carbonyl)piperazine-1-carboxamide, PH-interacting protein
著者Grosjean, H, Tomlinson, C, Bradshaw, W.J, Koekemoer, L, Krojer, T, Fearon, D, Biggin, P.C, von Delft, F.
登録日2023-03-09
公開日2023-03-29
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (1.15 Å)
主引用文献PanDDA analysis group deposition
To Be Published
7FVL
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BU of 7fvl by Molmil
PanDDA analysis group deposition -- PHIP in complex with Z4140355932
分子名称: N-{[(2S)-5,5-dimethyl-1,4-dioxan-2-yl]methyl}-4-(3-hydroxybenzoyl)piperazine-1-carboxamide, PH-interacting protein
著者Grosjean, H, Tomlinson, C, Bradshaw, W.J, Koekemoer, L, Krojer, T, Fearon, D, Biggin, P.C, von Delft, F.
登録日2023-03-09
公開日2023-03-29
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (1.15 Å)
主引用文献PanDDA analysis group deposition
To Be Published
7FV2
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BU of 7fv2 by Molmil
PanDDA analysis group deposition -- PHIP in complex with Z445899798
分子名称: N-(2-methoxyethyl)-4-(thiophene-2-carbonyl)piperazine-1-carboxamide, PH-interacting protein
著者Grosjean, H, Tomlinson, C, Bradshaw, W.J, Koekemoer, L, Krojer, T, Fearon, D, Biggin, P.C, von Delft, F.
登録日2023-03-09
公開日2023-03-29
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (1.15 Å)
主引用文献PanDDA analysis group deposition
To Be Published
7FVI
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BU of 7fvi by Molmil
PanDDA analysis group deposition -- PHIP in complex with Z183306756
分子名称: N-[(2H-1,3-benzodioxol-5-yl)methyl]-4-(furan-2-carbonyl)piperazine-1-carboxamide, PH-interacting protein
著者Grosjean, H, Tomlinson, C, Bradshaw, W.J, Koekemoer, L, Krojer, T, Fearon, D, Biggin, P.C, von Delft, F.
登録日2023-03-09
公開日2023-03-29
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (1.18 Å)
主引用文献PanDDA analysis group deposition
To Be Published
7FVJ
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BU of 7fvj by Molmil
PanDDA analysis group deposition -- PHIP in complex with Z4913873236
分子名称: (2S)-4-(furan-2-carbonyl)-2-methyl-N-(2,2,2-trifluoroethyl)piperazine-1-carboxamide, PH-interacting protein
著者Grosjean, H, Tomlinson, C, Bradshaw, W.J, Koekemoer, L, Krojer, T, Fearon, D, Biggin, P.C, von Delft, F.
登録日2023-03-09
公開日2023-03-29
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (1.19 Å)
主引用文献PanDDA analysis group deposition
To Be Published
7FVA
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BU of 7fva by Molmil
PanDDA analysis group deposition -- PHIP in complex with Z4913872963
分子名称: (2S)-N-(cyclopropylmethyl)-4-(furan-2-carbonyl)-2-methylpiperazine-1-carboxamide, PH-interacting protein
著者Grosjean, H, Tomlinson, C, Bradshaw, W.J, Koekemoer, L, Krojer, T, Fearon, D, Biggin, P.C, von Delft, F.
登録日2023-03-09
公開日2023-03-29
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (1.19 Å)
主引用文献PanDDA analysis group deposition
To Be Published
7FV9
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BU of 7fv9 by Molmil
PanDDA analysis group deposition -- PHIP in complex with Z1004253138
分子名称: 4-(5-methylfuran-2-carbonyl)-N-[(thiophen-2-yl)methyl]piperazine-1-carboxamide, PH-interacting protein
著者Grosjean, H, Tomlinson, C, Bradshaw, W.J, Koekemoer, L, Krojer, T, Fearon, D, Biggin, P.C, von Delft, F.
登録日2023-03-09
公開日2023-03-29
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (1.17 Å)
主引用文献PanDDA analysis group deposition
To Be Published
7FVM
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BU of 7fvm by Molmil
PanDDA analysis group deposition -- PHIP in complex with Z1590917771
分子名称: 4-(furan-2-carbonyl)-N-(1,2-oxazol-3-yl)piperazine-1-carboxamide, PH-interacting protein
著者Grosjean, H, Tomlinson, C, Bradshaw, W.J, Koekemoer, L, Krojer, T, Fearon, D, Biggin, P.C, von Delft, F.
登録日2023-03-09
公開日2023-03-29
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (1.26 Å)
主引用文献PanDDA analysis group deposition
To Be Published
7FVQ
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BU of 7fvq by Molmil
PanDDA analysis group deposition -- PHIP in complex with Z68576046
分子名称: N-butyl-4-(thiophene-2-carbonyl)piperazine-1-carboxamide, PH-interacting protein
著者Grosjean, H, Tomlinson, C, Bradshaw, W.J, Koekemoer, L, Krojer, T, Fearon, D, Biggin, P.C, von Delft, F.
登録日2023-03-09
公開日2023-03-29
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (1.15 Å)
主引用文献PanDDA analysis group deposition
To Be Published
7FVP
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BU of 7fvp by Molmil
PanDDA analysis group deposition -- PHIP in complex with Z1004277578
分子名称: N-butyl-4-(5-methylfuran-2-carbonyl)piperazine-1-carboxamide, PH-interacting protein
著者Grosjean, H, Tomlinson, C, Bradshaw, W.J, Koekemoer, L, Krojer, T, Fearon, D, Biggin, P.C, von Delft, F.
登録日2023-03-09
公開日2023-03-29
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (1.15 Å)
主引用文献PanDDA analysis group deposition
To Be Published
7FVC
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BU of 7fvc by Molmil
PanDDA analysis group deposition -- PHIP in complex with Z495704106
分子名称: N-(cyclopropylmethyl)-4-(3,4-dichlorobenzoyl)piperazine-1-carboxamide, PH-interacting protein
著者Grosjean, H, Tomlinson, C, Bradshaw, W.J, Koekemoer, L, Krojer, T, Fearon, D, Biggin, P.C, von Delft, F.
登録日2023-03-09
公開日2023-03-29
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (1.18 Å)
主引用文献PanDDA analysis group deposition
To Be Published
7FVN
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BU of 7fvn by Molmil
PanDDA analysis group deposition -- PHIP in complex with Z371875396
分子名称: N-(propan-2-yl)-4-(thiophene-2-carbonyl)piperazine-1-carboxamide, PH-interacting protein
著者Grosjean, H, Tomlinson, C, Bradshaw, W.J, Koekemoer, L, Krojer, T, Fearon, D, Biggin, P.C, von Delft, F.
登録日2023-03-09
公開日2023-03-29
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (1.15 Å)
主引用文献PanDDA analysis group deposition
To Be Published
7FUT
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BU of 7fut by Molmil
PanDDA analysis group deposition -- PHIP in complex with Z44602357
分子名称: 4-(furan-2-carbonyl)-N-propylpiperazine-1-carboxamide, PH-interacting protein
著者Grosjean, H, Tomlinson, C, Bradshaw, W.J, Koekemoer, L, Krojer, T, Fearon, D, Biggin, P.C, von Delft, F.
登録日2023-03-09
公開日2023-03-29
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (1.18 Å)
主引用文献PanDDA analysis group deposition
To Be Published
7FVO
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BU of 7fvo by Molmil
PanDDA analysis group deposition -- PHIP in complex with Z1435810807
分子名称: N-[2-(4,5-dimethyl-1,3-thiazol-2-yl)ethyl]-4-(thiophene-2-carbonyl)piperazine-1-carboxamide, PH-interacting protein
著者Grosjean, H, Tomlinson, C, Bradshaw, W.J, Koekemoer, L, Krojer, T, Fearon, D, Biggin, P.C, von Delft, F.
登録日2023-03-09
公開日2023-03-29
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (1.19 Å)
主引用文献PanDDA analysis group deposition
To Be Published
7FVR
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BU of 7fvr by Molmil
PanDDA analysis group deposition -- PHIP in complex with Z166737374
分子名称: 4-(thiophene-2-carbonyl)-N-[(thiophen-2-yl)methyl]piperazine-1-carboxamide, PH-interacting protein
著者Grosjean, H, Tomlinson, C, Bradshaw, W.J, Koekemoer, L, Krojer, T, Fearon, D, Biggin, P.C, von Delft, F.
登録日2023-03-09
公開日2023-03-29
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (1.19 Å)
主引用文献PanDDA analysis group deposition
To Be Published
7FUV
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BU of 7fuv by Molmil
PanDDA analysis group deposition -- PHIP in complex with Z183376720
分子名称: N-cyclopropyl-4-(furan-2-carbonyl)piperazine-1-carboxamide, PH-interacting protein
著者Grosjean, H, Tomlinson, C, Bradshaw, W.J, Koekemoer, L, Krojer, T, Fearon, D, Biggin, P.C, von Delft, F.
登録日2023-03-09
公開日2023-03-29
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (1.19 Å)
主引用文献PanDDA analysis group deposition
To Be Published
7FUZ
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BU of 7fuz by Molmil
PanDDA analysis group deposition -- PHIP in complex with Z4307421429
分子名称: N-tert-butyl-4-(2,3,3-trimethyl-3H-indole-5-carbonyl)piperazine-1-carboxamide, PH-interacting protein
著者Grosjean, H, Tomlinson, C, Bradshaw, W.J, Koekemoer, L, Krojer, T, Fearon, D, Biggin, P.C, von Delft, F.
登録日2023-03-09
公開日2023-03-29
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (1.43 Å)
主引用文献PanDDA analysis group deposition
To Be Published

224004

件を2024-08-21に公開中

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