8IQ5
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![BU of 8iq5 by Molmil](/molmil-images/mine/8iq5) | Crystal structure of trimeric K2-2 TSP | 分子名称: | 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, BICINE, GLYCEROL, ... | 著者 | Ye, T.J, Huang, K.F, Ko, T.P. | 登録日 | 2023-03-15 | 公開日 | 2024-02-21 | 最終更新日 | 2024-04-03 | 実験手法 | X-RAY DIFFRACTION (1.38 Å) | 主引用文献 | Klebsiella pneumoniae K2 capsular polysaccharide degradation by a bacteriophage depolymerase does not require trimer formation. Mbio, 15, 2024
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6M5N
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![BU of 6m5n by Molmil](/molmil-images/mine/6m5n) | Apo-Form Structure of Borneol Dehydrogenase | 分子名称: | ACETATE ION, Borneol dehydrogenase, SULFATE ION | 著者 | Khine, A.A, Huang, K.F, Ko, T.P, Chen, H.P. | 登録日 | 2020-03-11 | 公開日 | 2020-07-15 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (1.84 Å) | 主引用文献 | Structural characterization of borneol dehydrogenase from Pseudomonas sp. TCU-HL1 Acta Crystallogr.,Sect.F, 76, 2020
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4J4M
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![BU of 4j4m by Molmil](/molmil-images/mine/4j4m) | Crystal structure of TM-1, a Trimeresurus mucrosquamatus venom metalloproteinase | 分子名称: | ZINC ION, zinc-dependent metalloproteinase | 著者 | Chou, T.L, Wu, C.H, Huang, K.F, Wang, A.H. | 登録日 | 2013-02-07 | 公開日 | 2013-07-10 | 最終更新日 | 2023-11-08 | 実験手法 | X-RAY DIFFRACTION (1.8 Å) | 主引用文献 | Crystal structure of a Trimeresurus mucrosquamatus venom metalloproteinase providing new insights into the inhibition by endogenous tripeptide inhibitors. Toxicon, 71C, 2013
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8K7I
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![BU of 8k7i by Molmil](/molmil-images/mine/8k7i) | Crystal structure of human lysosomal alpha-galactosidase A in complex with (2R,3S,4R,5R)-2-(hydroxymethyl)-5-((methylamino)methyl)pyrrolidine-3,4-diol | 分子名称: | (2~{R},3~{S},4~{R},5~{R})-2-(hydroxymethyl)-5-(methylaminomethyl)pyrrolidine-3,4-diol, 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, ... | 著者 | Li, H.Y, Huang, K.F, Ko, T.P, Cheng, W.C. | 登録日 | 2023-07-26 | 公開日 | 2024-04-10 | 実験手法 | X-RAY DIFFRACTION (2.12 Å) | 主引用文献 | Mechanistic Insights into Dibasic Iminosugars as pH-Selective Pharmacological Chaperones to Stabilize Human alpha-Galactosidase. Jacs Au, 4, 2024
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8K7J
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![BU of 8k7j by Molmil](/molmil-images/mine/8k7j) | Crystal structure of human lysosomal alpha-galactosidase A in complex with (2R,3R,4S,5R)-2-((dimethylamino)methyl)-5-(hydroxymethyl)pyrrolidine-3,4-diol | 分子名称: | (2~{R},3~{R},4~{S},5~{R})-2-[(dimethylamino)methyl]-5-(hydroxymethyl)pyrrolidine-3,4-diol, 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, ... | 著者 | Li, H.Y, Huang, K.F, Ko, T.P, Cheng, W.C. | 登録日 | 2023-07-26 | 公開日 | 2024-04-10 | 実験手法 | X-RAY DIFFRACTION (2.01 Å) | 主引用文献 | Mechanistic Insights into Dibasic Iminosugars as pH-Selective Pharmacological Chaperones to Stabilize Human alpha-Galactosidase. Jacs Au, 4, 2024
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8K7H
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![BU of 8k7h by Molmil](/molmil-images/mine/8k7h) | Crystal structure of human lysosomal alpha-galactosidase A in complex with (2R,3S,4R)-2-(hydroxymethyl)-1-methylpyrrolidine-3,4-diol | 分子名称: | (2~{R},3~{S},4~{R})-2-(hydroxymethyl)-1-methyl-pyrrolidine-3,4-diol, 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, ... | 著者 | Li, H.Y, Huang, K.F, Ko, T.P, Cheng, W.C. | 登録日 | 2023-07-26 | 公開日 | 2024-04-10 | 実験手法 | X-RAY DIFFRACTION (2.28 Å) | 主引用文献 | Mechanistic Insights into Dibasic Iminosugars as pH-Selective Pharmacological Chaperones to Stabilize Human alpha-Galactosidase. Jacs Au, 4, 2024
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8K7L
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![BU of 8k7l by Molmil](/molmil-images/mine/8k7l) | Crystal structure of human lysosomal alpha-galactosidase A in complex with (2R,3R,4S,5R)-2-(aminomethyl)-5-(hydroxymethyl)-1-methylpyrrolidine-3,4-diol | 分子名称: | (2~{R},3~{R},4~{S},5~{R})-2-(aminomethyl)-5-(hydroxymethyl)-1-methyl-pyrrolidine-3,4-diol, 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, ... | 著者 | Li, H.Y, Huang, K.F, Ko, T.P, Cheng, W.C. | 登録日 | 2023-07-26 | 公開日 | 2024-04-10 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Mechanistic Insights into Dibasic Iminosugars as pH-Selective Pharmacological Chaperones to Stabilize Human alpha-Galactosidase. Jacs Au, 4, 2024
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8K7D
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![BU of 8k7d by Molmil](/molmil-images/mine/8k7d) | Crystal structure of human lysosomal alpha-galactosidase A in complex with (2R,3R,4S,5R)-2-(aminomethyl)-5-(hydroxymethyl)pyrrolidine-3,4-diol | 分子名称: | (2~{R},3~{R},4~{S},5~{R})-2-(aminomethyl)-5-(hydroxymethyl)pyrrolidine-3,4-diol, 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, ... | 著者 | Li, H.Y, Huang, K.F, Ko, T.P, Cheng, W.C. | 登録日 | 2023-07-26 | 公開日 | 2024-04-10 | 実験手法 | X-RAY DIFFRACTION (2.61 Å) | 主引用文献 | Mechanistic Insights into Dibasic Iminosugars as pH-Selective Pharmacological Chaperones to Stabilize Human alpha-Galactosidase. Jacs Au, 4, 2024
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8K7F
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![BU of 8k7f by Molmil](/molmil-images/mine/8k7f) | Crystal structure of human lysosomal alpha-galactosidase A in complex with (2R,3S,4R,5R)-2,5-bis(hydroxymethyl)pyrrolidine-3,4-diol | 分子名称: | (2~{R},3~{R},4~{S},5~{R})-2,5-bis(hydroxymethyl)pyrrolidine-3,4-diol, 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, ... | 著者 | Li, H.Y, Huang, K.F, Ko, T.P, Cheng, W.C. | 登録日 | 2023-07-26 | 公開日 | 2024-04-10 | 実験手法 | X-RAY DIFFRACTION (1.98 Å) | 主引用文献 | Mechanistic Insights into Dibasic Iminosugars as pH-Selective Pharmacological Chaperones to Stabilize Human alpha-Galactosidase. Jacs Au, 4, 2024
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8K7G
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![BU of 8k7g by Molmil](/molmil-images/mine/8k7g) | Crystal structure of human lysosomal alpha-galactosidase A in complex with (2R,3S,4R,5R)-2,5-bis(hydroxymethyl)pyrrolidine-3,4-diol | 分子名称: | (2~{R},3~{R},4~{S},5~{R})-2,5-bis(hydroxymethyl)pyrrolidine-3,4-diol, 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, ... | 著者 | Li, H.Y, Huang, K.F, Ko, T.P, Cheng, W.C. | 登録日 | 2023-07-26 | 公開日 | 2024-04-10 | 実験手法 | X-RAY DIFFRACTION (2.32 Å) | 主引用文献 | Mechanistic Insights into Dibasic Iminosugars as pH-Selective Pharmacological Chaperones to Stabilize Human alpha-Galactosidase. Jacs Au, 4, 2024
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8K7E
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![BU of 8k7e by Molmil](/molmil-images/mine/8k7e) | Crystal structure of human lysosomal alpha-galactosidase A in complex with (2R,3R,4S,5R)-2-(aminomethyl)-5-(hydroxymethyl)pyrrolidine-3,4-diol | 分子名称: | (2~{R},3~{R},4~{S},5~{R})-2-(aminomethyl)-5-(hydroxymethyl)pyrrolidine-3,4-diol, 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, ... | 著者 | Li, H.Y, Huang, K.F, Ko, T.P, Cheng, W.C. | 登録日 | 2023-07-26 | 公開日 | 2024-04-10 | 実験手法 | X-RAY DIFFRACTION (2.2 Å) | 主引用文献 | Mechanistic Insights into Dibasic Iminosugars as pH-Selective Pharmacological Chaperones to Stabilize Human alpha-Galactosidase. Jacs Au, 4, 2024
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8K7K
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![BU of 8k7k by Molmil](/molmil-images/mine/8k7k) | Crystal structure of human lysosomal alpha-galactosidase A in complex with (2R,3S,4R,5R)-2,5-bis(hydroxymethyl)-1-methylpyrrolidine-3,4-diol | 分子名称: | (2~{R},3~{S},4~{R},5~{R})-2,5-bis(hydroxymethyl)-1-methyl-pyrrolidine-3,4-diol, 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, ... | 著者 | Li, H.Y, Huang, K.F, Ko, T.P, Cheng, W.C. | 登録日 | 2023-07-26 | 公開日 | 2024-04-10 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Mechanistic Insights into Dibasic Iminosugars as pH-Selective Pharmacological Chaperones to Stabilize Human alpha-Galactosidase. Jacs Au, 4, 2024
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3VA4
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![BU of 3va4 by Molmil](/molmil-images/mine/3va4) | Crystal structure of the mammalian MDC1 FHA domain complexed with CHK2 pThr68 peptide | 分子名称: | Mediator of DNA damage checkpoint protein 1, Serine/threonine-protein kinase Chk2 | 著者 | Wu, H.H, Wu, P.Y, Huang, K.F, Kao, Y.Y, Tsai, M.D. | 登録日 | 2011-12-28 | 公開日 | 2012-02-01 | 実験手法 | X-RAY DIFFRACTION (1.54 Å) | 主引用文献 | Structural Delineation of MDC1-FHA Domain Binding with CHK2-pThr68. Biochemistry, 2012
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5XFT
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![BU of 5xft by Molmil](/molmil-images/mine/5xft) | |
5ZYO
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![BU of 5zyo by Molmil](/molmil-images/mine/5zyo) | |
6JC5
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![BU of 6jc5 by Molmil](/molmil-images/mine/6jc5) | |
6JC6
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![BU of 6jc6 by Molmil](/molmil-images/mine/6jc6) | |
7EI3
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![BU of 7ei3 by Molmil](/molmil-images/mine/7ei3) | |
7EI4
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![BU of 7ei4 by Molmil](/molmil-images/mine/7ei4) | Crystal structure of MasL in complex with a novel covalent inhibitor, collimonin C | 分子名称: | (6S,7R,9E)-6,7-bis(oxidanyl)hexadeca-9,15-dien-11,13-diynoic acid, Acetyl-CoA C-acyltransferase | 著者 | Lin, C.C, Huang, K.F, Yang, Y.L. | 登録日 | 2021-03-30 | 公開日 | 2022-04-06 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (1.66 Å) | 主引用文献 | Integrated omics approach to unveil antifungal bacterial polyynes as acetyl-CoA acetyltransferase inhibitors. Commun Biol, 5, 2022
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7EV4
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![BU of 7ev4 by Molmil](/molmil-images/mine/7ev4) | Crystal structure of the Lon-like protease MtaLonC with S582A mutation in complex with F-b20-Q | 分子名称: | Endopeptidase La, F-b20-Q peptide {ortho-aminobenzoic acid (Abz)- QLRSLNGEWRFAWFPAPEAV[Tyr(3-NO2)]A}, PHOSPHATE ION | 著者 | Hsieh, K.Y, Kuo, C.I, Su, S.C, Huang, K.F, Chang, C.I. | 登録日 | 2021-05-20 | 公開日 | 2021-11-24 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (2.12 Å) | 主引用文献 | Processive cleavage of substrate at individual proteolytic active sites of the Lon protease complex. Sci Adv, 7, 2021
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7EV6
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![BU of 7ev6 by Molmil](/molmil-images/mine/7ev6) | Crystal structure of the Lon-like protease MtaLonC with D581A mutation in complex with F-b20-Q | 分子名称: | Endopeptidase La, F-b20-Q peptide {ortho-aminobenzoic acid (Abz)- QLRSLNGEWRFAWFPAPEAV[Tyr(3-NO2)]A}, PHOSPHATE ION | 著者 | Hsieh, K.Y, Kuo, C.I, Su, S.C, Huang, K.F, Chang, C.I. | 登録日 | 2021-05-20 | 公開日 | 2021-11-24 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (2.1 Å) | 主引用文献 | Processive cleavage of substrate at individual proteolytic active sites of the Lon protease complex. Sci Adv, 7, 2021
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7EUY
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![BU of 7euy by Molmil](/molmil-images/mine/7euy) | Crystal structure of the Lon-like protease MtaLonC with D582A mutation in complex with substrate polypeptide | 分子名称: | ALA-PRO-GLU-ALA-VAL, Endopeptidase La, PHOSPHATE ION | 著者 | Hsieh, K.Y, Kuo, C.I, Su, S.C, Huang, K.F, Chang, C.I. | 登録日 | 2021-05-19 | 公開日 | 2021-11-24 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (2.2 Å) | 主引用文献 | Processive cleavage of substrate at individual proteolytic active sites of the Lon protease complex. Sci Adv, 7, 2021
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7EUX
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![BU of 7eux by Molmil](/molmil-images/mine/7eux) | Crystal structure of the Lon-like protease MtaLonC with D581A mutation in complex with substrate polypeptide | 分子名称: | ALA-PRO-GLU-ALA-VAL, Endopeptidase La, PHOSPHATE ION | 著者 | Hsieh, K.Y, Kuo, C.I, Su, S.C, Huang, K.F, Chang, C.I. | 登録日 | 2021-05-19 | 公開日 | 2021-11-24 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (2.25 Å) | 主引用文献 | Processive cleavage of substrate at individual proteolytic active sites of the Lon protease complex. Sci Adv, 7, 2021
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7FEA
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![BU of 7fea by Molmil](/molmil-images/mine/7fea) | PY14 in complex with Col-D | 分子名称: | (6~{R},7~{R},9~{E})-6,7-bis(oxidanyl)hexadeca-9,15-dien-11,13-diynoic acid, Acetyl-CoA C-acyltransferase | 著者 | Lin, C.C, Ko, T.P, Huang, K.F, Yang, Y.L. | 登録日 | 2021-07-19 | 公開日 | 2022-07-27 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (1.4 Å) | 主引用文献 | Integrated omics approach to unveil antifungal bacterial polyynes as acetyl-CoA acetyltransferase inhibitors. Commun Biol, 5, 2022
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7VT7
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![BU of 7vt7 by Molmil](/molmil-images/mine/7vt7) | Crystal structure of CBM deleted MtGlu5 in complex with CBI | 分子名称: | Endoglucanase H, GLYCEROL, TRYPTOPHAN, ... | 著者 | Ye, T.J, Ko, P.T, Huang, K.F, Wu, S.H. | 登録日 | 2021-10-28 | 公開日 | 2022-09-07 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (1.53 Å) | 主引用文献 | Synergic action of an inserted carbohydrate-binding module in a glycoside hydrolase family 5 endoglucanase. Acta Crystallogr D Struct Biol, 78, 2022
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