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Crystal structure of D1228V c-MET bound by compound 16
分子名称:	1-[(1S)-1-[3-(1H-imidazol-4-yl)phenyl]ethyl]-5-(1H-indazol-7-yl)pyrimidine-2,4-dione, Hepatocyte growth factor receptor, IODIDE ION
著者	Collie, G.W.
登録日	2023-04-26
公開日	2023-07-05
最終更新日	2023-09-20
実験手法	X-RAY DIFFRACTION (2.206 Å)
主引用文献	Discovery and Optimization of the First ATP Competitive Type-III c-MET Inhibitor. J.Med.Chem., 66, 2023

Crystal structure of the kinase domain of human PAK1 in complex with compound 15
分子名称:	Serine/threonine-protein kinase PAK 1, [2-chloro-5-(hydroxymethyl)phenyl]{5-[1-(piperidin-4-yl)-1H-pyrazol-4-yl]-1H-pyrrolo[2,3-b]pyridin-3-yl}methanone
著者	Ferguson, A.D.
登録日	2014-04-01
公開日	2014-09-10
最終更新日	2023-09-27
実験手法	X-RAY DIFFRACTION (2.49 Å)
主引用文献	Identification and optimisation of 7-azaindole PAK1 inhibitors with improved potency and kinase selectivity. MEDCHEMCOMM, 2014