4F7D
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![BU of 4f7d by Molmil](/molmil-images/mine/4f7d) | |
3TMQ
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![BU of 3tmq by Molmil](/molmil-images/mine/3tmq) | |
3TK1
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![BU of 3tk1 by Molmil](/molmil-images/mine/3tk1) | |
3U7J
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![BU of 3u7j by Molmil](/molmil-images/mine/3u7j) | |
3TSC
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![BU of 3tsc by Molmil](/molmil-images/mine/3tsc) | |
3U0I
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![BU of 3u0i by Molmil](/molmil-images/mine/3u0i) | |
3UE9
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![BU of 3ue9 by Molmil](/molmil-images/mine/3ue9) | |
3UK1
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![BU of 3uk1 by Molmil](/molmil-images/mine/3uk1) | |
4NW7
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![BU of 4nw7 by Molmil](/molmil-images/mine/4nw7) | PDE4 catalytic domain | 分子名称: | (4-{[4-(3-chlorophenyl)-6-cyclopropyl-1,3,5-triazin-2-yl]amino}phenyl)acetic acid, 1,2-ETHANEDIOL, MAGNESIUM ION, ... | 著者 | Fox III, D, Edwards, T.E. | 登録日 | 2013-12-05 | 公開日 | 2014-10-15 | 最終更新日 | 2024-02-28 | 実験手法 | X-RAY DIFFRACTION (2.15 Å) | 主引用文献 | Discovery of triazines as selective PDE4B versus PDE4D inhibitors. Bioorg.Med.Chem.Lett., 24, 2014
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4GK6
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4HDT
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![BU of 4hdt by Molmil](/molmil-images/mine/4hdt) | |
4HR3
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![BU of 4hr3 by Molmil](/molmil-images/mine/4hr3) | |
4I1Y
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![BU of 4i1y by Molmil](/molmil-images/mine/4i1y) | |
4IJN
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![BU of 4ijn by Molmil](/molmil-images/mine/4ijn) | |
4WTF
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![BU of 4wtf by Molmil](/molmil-images/mine/4wtf) | CRYSTAL STRUCTURE OF HCV NS5B GENOTYPE 2A JFH-1 ISOLATE WITH S15G E86Q E87Q C223H V321I MUTATIONS AND DELTA8 BETA HAIRPIN LOOP DELETION IN COMPLEX WITH GS-639475, MN2+ AND SYMMETRICAL PRIMER TEMPLATE 5'-CAAAAUUU | 分子名称: | 2'-C-methyluridine 5'-(trihydrogen diphosphate), CHLORIDE ION, MANGANESE (II) ION, ... | 著者 | Edwards, T.E, Appleby, T.C, Mcgrath, M.E. | 登録日 | 2014-10-30 | 公開日 | 2015-02-11 | 最終更新日 | 2023-09-27 | 実験手法 | X-RAY DIFFRACTION (2.65 Å) | 主引用文献 | Structural basis for RNA replication by the hepatitis C virus polymerase. Science, 347, 2015
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4WTJ
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![BU of 4wtj by Molmil](/molmil-images/mine/4wtj) | CRYSTAL STRUCTURE OF HCV NS5B GENOTYPE 2A JFH-1 ISOLATE WITH S15G E86Q E87Q C223H V321I MUTATIONS IN COMPLEX WITH RNA TEMPLATE 5'-AUCC, RNA PRIMER 5'-PGG, MN2+, AND ADP | 分子名称: | 1,2-ETHANEDIOL, 1-(2-METHOXY-ETHOXY)-2-{2-[2-(2-METHOXY-ETHOXY]-ETHOXY}-ETHANE, 2-[3-(2-HYDROXY-1,1-DIHYDROXYMETHYL-ETHYLAMINO)-PROPYLAMINO]-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, ... | 著者 | Edwards, T.E, Appleby, T.C. | 登録日 | 2014-10-30 | 公開日 | 2015-02-11 | 最終更新日 | 2023-09-27 | 実験手法 | X-RAY DIFFRACTION (2.2 Å) | 主引用文献 | Structural basis for RNA replication by the hepatitis C virus polymerase. Science, 347, 2015
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4WT9
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![BU of 4wt9 by Molmil](/molmil-images/mine/4wt9) | |
4WTA
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![BU of 4wta by Molmil](/molmil-images/mine/4wta) | |
4WTC
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![BU of 4wtc by Molmil](/molmil-images/mine/4wtc) | |
4WTE
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![BU of 4wte by Molmil](/molmil-images/mine/4wte) | |
4WTG
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![BU of 4wtg by Molmil](/molmil-images/mine/4wtg) | |
4WTI
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![BU of 4wti by Molmil](/molmil-images/mine/4wti) | CRYSTAL STRUCTURE OF HCV NS5B GENOTYPE 2A JFH-1 ISOLATE WITH S15G E86Q E87Q C223H V321I MUTATIONS IN COMPLEX WITH RNA TEMPLATE 5'-ACGG, RNA PRIMER 5'-PCC, MN2+, AND GDP | 分子名称: | 2-[3-(2-HYDROXY-1,1-DIHYDROXYMETHYL-ETHYLAMINO)-PROPYLAMINO]-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, CHLORIDE ION, GUANOSINE-5'-DIPHOSPHATE, ... | 著者 | Edwards, T.E, Appleby, T.C. | 登録日 | 2014-10-30 | 公開日 | 2015-02-11 | 最終更新日 | 2023-09-27 | 実験手法 | X-RAY DIFFRACTION (2.8 Å) | 主引用文献 | Structural basis for RNA replication by the hepatitis C virus polymerase. Science, 347, 2015
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4WTK
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![BU of 4wtk by Molmil](/molmil-images/mine/4wtk) | CRYSTAL STRUCTURE OF HCV NS5B GENOTYPE 2A JFH-1 ISOLATE WITH S15G E86Q E87Q C223H V321I MUTATIONS IN COMPLEX WITH RNA TEMPLATE 5'-AGCC, RNA PRIMER 5'-PGG, MN2+, AND CDP | 分子名称: | 1,2-ETHANEDIOL, 1-(2-METHOXY-ETHOXY)-2-{2-[2-(2-METHOXY-ETHOXY]-ETHOXY}-ETHANE, 2-[3-(2-HYDROXY-1,1-DIHYDROXYMETHYL-ETHYLAMINO)-PROPYLAMINO]-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, ... | 著者 | Edwards, T.E, Appleby, T.C. | 登録日 | 2014-10-30 | 公開日 | 2015-02-11 | 最終更新日 | 2023-09-27 | 実験手法 | X-RAY DIFFRACTION (2.5 Å) | 主引用文献 | Structural basis for RNA replication by the hepatitis C virus polymerase. Science, 347, 2015
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4WTL
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![BU of 4wtl by Molmil](/molmil-images/mine/4wtl) | CRYSTAL STRUCTURE OF HCV NS5B GENOTYPE 2A JFH-1 ISOLATE WITH S15G E86Q E87Q C223H V321I MUTATIONS IN COMPLEX WITH RNA TEMPLATE 5'-UACC, RNA PRIMER 5'-PGG, MN2+, AND UDP | 分子名称: | 1-(2-METHOXY-ETHOXY)-2-{2-[2-(2-METHOXY-ETHOXY]-ETHOXY}-ETHANE, 2-[3-(2-HYDROXY-1,1-DIHYDROXYMETHYL-ETHYLAMINO)-PROPYLAMINO]-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, CHLORIDE ION, ... | 著者 | Edwards, T.E, Appleby, T.C. | 登録日 | 2014-10-30 | 公開日 | 2015-02-11 | 最終更新日 | 2023-09-27 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Structural basis for RNA replication by the hepatitis C virus polymerase. Science, 347, 2015
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4IZ9
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![BU of 4iz9 by Molmil](/molmil-images/mine/4iz9) | |