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6ZL3
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BU of 6zl3 by Molmil
CRYSTAL STRUCTURE OF HRAS IN COMPLEX WITH COMPOUND 18 and GDP
分子名称: (3~{S})-3-[2-[(dimethylamino)methyl]-1~{H}-indol-3-yl]-5-oxidanyl-2,3-dihydroisoindol-1-one, GTPase HRas, GUANOSINE-5'-DIPHOSPHATE, ...
著者Kessler, D, Fischer, G, Boettcher, J.
登録日2020-06-30
公開日2020-08-19
最終更新日2024-01-31
実験手法X-RAY DIFFRACTION (2.031 Å)
主引用文献Drugging all RAS isoforms with one pocket.
Future Med Chem, 12, 2020
6ZJ0
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BU of 6zj0 by Molmil
CRYSTAL STRUCTURE OF HRAS-G12D IN COMPLEX WITH GCP AND COMPOUND 18
分子名称: (3~{S})-3-[2-[(dimethylamino)methyl]-1~{H}-indol-3-yl]-5-oxidanyl-2,3-dihydroisoindol-1-one, GTPase HRas, MAGNESIUM ION, ...
著者Kessler, D, Fischer, G, Boettcher, J.
登録日2020-06-26
公開日2020-08-19
最終更新日2024-01-31
実験手法X-RAY DIFFRACTION (1.763 Å)
主引用文献Drugging all RAS isoforms with one pocket.
Future Med Chem, 12, 2020
6ZLI
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BU of 6zli by Molmil
CRYSTAL STRUCTURE OF KRAS-G12D IN COMPLEX WITH COMPOUND 13 AND GCP
分子名称: 2-[(2~{R})-piperidin-2-yl]-1~{H}-indole, GTPase KRas, MAGNESIUM ION, ...
著者Kessler, D, Fischer, G, Boettcher, J.
登録日2020-06-30
公開日2020-08-19
最終更新日2024-01-31
実験手法X-RAY DIFFRACTION (1.73 Å)
主引用文献Drugging all RAS isoforms with one pocket.
Future Med Chem, 12, 2020
6ZIR
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BU of 6zir by Molmil
CRYSTAL STRUCTURE OF NRAS (C118S) IN COMPLEX WITH GDP AND COMPOUND 18
分子名称: (3~{S})-3-[2-[(dimethylamino)methyl]-1~{H}-indol-3-yl]-5-oxidanyl-2,3-dihydroisoindol-1-one, GTPase NRas, GUANOSINE-5'-DIPHOSPHATE, ...
著者Kessler, D, Fischer, G, Boettcher, J.
登録日2020-06-26
公開日2020-08-19
最終更新日2024-01-31
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Drugging all RAS isoforms with one pocket.
Future Med Chem, 12, 2020
1QRZ
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BU of 1qrz by Molmil
CATALYTIC DOMAIN OF PLASMINOGEN
分子名称: PLASMINOGEN
著者Peisach, E, Wang, J, de los Santos, T, Reich, E, Ringe, D.
登録日1999-06-16
公開日1999-10-14
最終更新日2021-11-03
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Crystal structure of the proenzyme domain of plasminogen.
Biochemistry, 38, 1999
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