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4BX0
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BU of 4bx0 by Molmil
Crystal Structure of a Monomeric Variant of murine Chronophin (Pyridoxal Phosphate phosphatase)
分子名称: GLYCEROL, MAGNESIUM ION, PYRIDOXAL PHOSPHATE PHOSPHATASE
著者Kestler, C, Knobloch, G, Gohla, A, Schindelin, H.
登録日2013-07-08
公開日2013-12-25
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (1.75 Å)
主引用文献Chronophin Dimerization is Required for Proper Positioning of its Substrate Specificity Loop
J.Biol.Chem., 289, 2014
4FBT
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BU of 4fbt by Molmil
Dpo4 post-insertion complex with the N-(deoxyguanosin-8-yl)-1-aminopyrene lesion
分子名称: 2'-DEOXYGUANOSINE-5'-TRIPHOSPHATE, CALCIUM ION, DNA polymerase IV, ...
著者Kirouac, K, Ling, H.
登録日2012-05-23
公開日2013-06-12
最終更新日2024-02-28
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Structural mechanism of replication stalling on a bulky amino-polycyclic aromatic hydrocarbon DNA adduct by a y family DNA polymerase.
J.Mol.Biol., 425, 2013
1JW9
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BU of 1jw9 by Molmil
Structure of the Native MoeB-MoaD Protein Complex
分子名称: MOLYBDOPTERIN BIOSYNTHESIS MOEB PROTEIN, MOLYBDOPTERIN [MPT] CONVERTING FACTOR, SUBUNIT 1, ...
著者Lake, M.W, Wuebbens, M.M, Rajagopalan, K.V, Schindelin, H.
登録日2001-09-03
公開日2001-11-21
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献Mechanism of ubiquitin activation revealed by the structure of a bacterial MoeB-MoaD complex.
Nature, 414, 2001
4D81
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BU of 4d81 by Molmil
Metallosphera sedula Vps4 crystal structure
分子名称: AAA ATPase, central domain protein, ADENOSINE-5'-DIPHOSPHATE
著者Caillat, C, Macheboeuf, P, Wu, Y, McCarthy, A.A, Boeri-Erba, E, Effantin, G, Gottlinger, H.G, Weissenhorn, W, Renesto, P.
登録日2014-12-02
公開日2015-11-25
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献Asymmetric Ring Structure of Vps4 Required for Escrt-III Disassembly.
Nat.Commun., 6, 2015
1DMS
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BU of 1dms by Molmil
STRUCTURE OF DMSO REDUCTASE
分子名称: 2-AMINO-5,6-DIMERCAPTO-7-METHYL-3,7,8A,9-TETRAHYDRO-8-OXA-1,3,9,10-TETRAAZA-ANTHRACEN-4-ONE GUANOSINE DINUCLEOTIDE, DMSO REDUCTASE, MOLYBDENUM (IV)OXIDE
著者Schneider, F, Loewe, J, Huber, R, Schindelin, H, Kisker, C, Knaeblein, J.
登録日1996-09-03
公開日1998-07-01
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (1.88 Å)
主引用文献Crystal structure of dimethyl sulfoxide reductase from Rhodobacter capsulatus at 1.88 A resolution.
J.Mol.Biol., 263, 1996
4FBU
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BU of 4fbu by Molmil
Dpo4 polymerase pre-insertion binary complex with the N-(deoxyguanosin-8-yl)-1-aminopyrene lesion
分子名称: CALCIUM ION, DNA polymerase IV, DNA primer, ...
著者Kirouac, K, Basu, A, Ling, H.
登録日2012-05-23
公開日2013-06-12
最終更新日2024-02-28
実験手法X-RAY DIFFRACTION (2.6 Å)
主引用文献Structural mechanism of replication stalling on a bulky amino-polycyclic aromatic hydrocarbon DNA adduct by a y family DNA polymerase.
J.Mol.Biol., 425, 2013
4D80
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BU of 4d80 by Molmil
Metallosphera sedula Vps4 crystal structure
分子名称: AAA ATPASE, CENTRAL DOMAIN PROTEIN
著者Caillat, C, Macheboeuf, P, Wu, Y, McCarthy, A.A, Boeri-Erba, E, Effantin, G, Gottlinger, H.G, Weissenhorn, W, Renesto, P.
登録日2014-12-02
公開日2015-10-28
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (3.6 Å)
主引用文献Asymmetric Ring Structure of Vps4 Required for Escrt-III Disassembly.
Nat.Commun., 6, 2015
4EYI
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BU of 4eyi by Molmil
Human DNA polymerase iota incorporating dATP opposite N-(deoxyguanosin-8-yl)-1-aminopyrene lesion
分子名称: 2'-DEOXYADENOSINE 5'-TRIPHOSPHATE, DNA polymerase iota, DNA primer, ...
著者Kirouac, K, Ling, H.
登録日2012-05-01
公開日2013-01-09
最終更新日2024-02-28
実験手法X-RAY DIFFRACTION (2.9 Å)
主引用文献Replication of a carcinogenic nitropyrene DNA lesion by human Y-family DNA polymerase.
Nucleic Acids Res., 41, 2013
5T14
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BU of 5t14 by Molmil
DNA polymerase kappa extending beyond a bulky major benzo[a]pyrene adduct
分子名称: 2'-deoxy-5'-O-[(R)-hydroxy{[(R)-hydroxy(phosphonooxy)phosphoryl]amino}phosphoryl]adenosine, DNA, DNA polymerase kappa, ...
著者Jha, V.K, Ling, H.
登録日2016-08-17
公開日2016-12-21
最終更新日2024-03-06
実験手法X-RAY DIFFRACTION (3 Å)
主引用文献Structural basis of accurate replication beyond a bulky major benzo[a]pyrene adduct by human DNA polymerase kappa.
DNA Repair (Amst.), 49, 2017
1DI7
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BU of 1di7 by Molmil
1.60 ANGSTROM CRYSTAL STRUCTURE OF THE MOLYBDENUM COFACTOR BIOSYNTHESIS PROTEIN MOGA FROM ESCHERICHIA COLI
分子名称: MOLYBDENUM COFACTOR BIOSYNTHETIC ENZYME, SULFATE ION
著者Liu, M.T.W, Wuebbens, M.M, Rajagopalan, K.V, Schindelin, H.
登録日1999-11-29
公開日2000-01-19
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (1.6 Å)
主引用文献Crystal structure of the gephyrin-related molybdenum cofactor biosynthesis protein MogA from Escherichia coli.
J.Biol.Chem., 275, 2000
1DI6
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BU of 1di6 by Molmil
1.45 A CRYSTAL STRUCTURE OF THE MOLYBDENUMM COFACTOR BIOSYNTHESIS PROTEIN MOGA FROM ESCHERICHIA COLI
分子名称: MOLYBDENUM COFACTOR BIOSYNTHETIC ENZYME, SULFATE ION
著者Liu, M.T.W, Wuebbens, M.M, Rajagopalan, K.V, Schindelin, H.
登録日1999-11-29
公開日2000-01-19
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (1.45 Å)
主引用文献Crystal structure of the gephyrin-related molybdenum cofactor biosynthesis protein MogA from Escherichia coli.
J.Biol.Chem., 275, 2000
2NTI
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BU of 2nti by Molmil
Crystal structure of PCNA123 heterotrimer.
分子名称: 2,5,8,11,14,17,20,23-OCTAOXAPENTACOSAN-25-OL, BROMIDE ION, DNA polymerase sliding clamp A, ...
著者Hlinkova, V, Ling, H.
登録日2006-11-07
公開日2007-12-18
最終更新日2024-04-03
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献Structures of monomeric, dimeric and trimeric PCNA: PCNA-ring assembly and opening.
Acta Crystallogr.,Sect.D, 64, 2008
1FM0
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BU of 1fm0 by Molmil
MOLYBDOPTERIN SYNTHASE (MOAD/MOAE)
分子名称: CHLORIDE ION, MOLYBDOPTERIN CONVERTING FACTOR, SUBUNIT 1, ...
著者Rudolph, M.J, Wuebbens, M.M, Rajagolpalan, K.V, Schindelin, H.
登録日2000-08-15
公開日2001-01-17
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (1.45 Å)
主引用文献Crystal structure of molybdopterin synthase and its evolutionary relationship to ubiquitin activation.
Nat.Struct.Biol., 8, 2001
1K6Y
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BU of 1k6y by Molmil
Crystal Structure of a Two-Domain Fragment of HIV-1 Integrase
分子名称: Integrase, PHOSPHATE ION, POTASSIUM ION, ...
著者Wang, J, Ling, H, Yang, W, Craigie, R.
登録日2001-10-17
公開日2001-12-21
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献Structure of a two-domain fragment of HIV-1 integrase: implications for domain organization in the intact protein.
EMBO J., 20, 2001
1FMA
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BU of 1fma by Molmil
MOLYBDOPTERIN SYNTHASE (MOAD/MOAE)
分子名称: CHLORIDE ION, MOLYBDOPTERIN CONVERTING FACTOR, SUBUNIT 1, ...
著者Rudolph, M.J, Wuebbens, M.M, Rajagolpalan, K.V, Schindelin, H.
登録日2000-08-16
公開日2001-01-17
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (1.58 Å)
主引用文献Crystal structure of molybdopterin synthase and its evolutionary relationship to ubiquitin activation.
Nat.Struct.Biol., 8, 2001
1FR9
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BU of 1fr9 by Molmil
STRUCTURE OF E. COLI MOBA
分子名称: ACETATE ION, MOLYBDOPTERIN-GUANINE DINUCLEOTIDE BIOSYNTHESIS PROTEIN, ZINC ION
著者Lake, M.W, Temple, C.A, Rajagopalan, K.V, Schindelin, H.
登録日2000-09-07
公開日2001-01-10
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (1.65 Å)
主引用文献The crystal structure of the Escherichia coli MobA protein provides insight into molybdopterin guanine dinucleotide biosynthesis.
J.Biol.Chem., 275, 2000
1FRW
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BU of 1frw by Molmil
STRUCTURE OF E. COLI MOBA WITH BOUND GTP AND MANGANESE
分子名称: ACETATE ION, GUANOSINE-5'-TRIPHOSPHATE, MANGANESE (II) ION, ...
著者Lake, M.W, Temple, C.A, Rajagopalan, K.V, Schindelin, H.
登録日2000-09-07
公開日2001-01-10
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (1.75 Å)
主引用文献The crystal structure of the Escherichia coli MobA protein provides insight into molybdopterin guanine dinucleotide biosynthesis.
J.Biol.Chem., 275, 2000
4GLJ
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BU of 4glj by Molmil
Crystal structure of methylthioadenosine phosphorylase in complex with rhodamine B
分子名称: CHLORIDE ION, N-[9-(2-carboxyphenyl)-6-(diethylamino)-3H-xanthen-3-ylidene]-N-ethylethanaminium, PHOSPHATE ION, ...
著者Bujacz, A, Bujacz, G, Cieslinski, H, Bartasun, P.
登録日2012-08-14
公開日2013-02-20
最終更新日2023-09-13
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献A study on the interaction of rhodamine B with methylthioadenosine phosphorylase protein sourced from an antarctic soil metagenomic library.
Plos One, 8, 2013
4GLF
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BU of 4glf by Molmil
Crystal structure of methylthioadenosine phosphorylase sourced from an antarctic soil metagenomic library
分子名称: RsfP
著者Bujacz, A, Bujacz, G, Cieslinski, H, Bartasun, P.
登録日2012-08-14
公開日2013-02-20
最終更新日2023-09-13
実験手法X-RAY DIFFRACTION (1.98 Å)
主引用文献A study on the interaction of rhodamine B with methylthioadenosine phosphorylase protein sourced from an antarctic soil metagenomic library.
Plos One, 8, 2013
5T28
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BU of 5t28 by Molmil
mPI3Kd IN COMPLEX WITH 5k
分子名称: 3-(benzotriazol-1-yl)-5-[1-methyl-5-(1-phenylcyclopropyl)-1,2,4-triazol-3-yl]pyrazin-2-amine, Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform
著者Petersen, J, Terstige, I, Perry, M, Svensson, T, Tyrchan, C, Lindmark, H, Oster, L.
登録日2016-08-23
公開日2017-04-12
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (2.8 Å)
主引用文献Discovery of triazole aminopyrazines as a highly potent and selective series of PI3K delta inhibitors.
Bioorg. Med. Chem. Lett., 27, 2017
1JWA
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BU of 1jwa by Molmil
Structure of the ATP-bound MoeB-MoaD Protein Complex
分子名称: ADENOSINE-5'-TRIPHOSPHATE, MOLYBDOPTERIN BIOSYNTHESIS MOEB PROTEIN, MOLYBDOPTERIN [MPT] CONVERTING FACTOR, ...
著者Lake, M.W, Wuebbens, M.M, Rajagopalan, K.V, Schindelin, H.
登録日2001-09-03
公開日2001-11-21
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (2.9 Å)
主引用文献Mechanism of ubiquitin activation revealed by the structure of a bacterial MoeB-MoaD complex.
Nature, 414, 2001
5T2L
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BU of 5t2l by Molmil
mPI3Kd IN COMPLEX WITH 7l
分子名称: 1-[3-azanyl-6-[1-methyl-5-(1-phenylcyclopropyl)-1,2,4-triazol-3-yl]pyrazin-2-yl]pyrazole-3-carboxamide, Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform
著者Petersen, J, Terstige, I, Perry, M, Svensson, T, Tyrchan, C, Lindmark, H, Oster, L.
登録日2016-08-23
公開日2017-04-19
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (2.55 Å)
主引用文献Discovery of triazole aminopyrazines as a highly potent and selective series of PI3K delta inhibitors.
Bioorg. Med. Chem. Lett., 27, 2017
5T27
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BU of 5t27 by Molmil
mPI3Kd IN COMPLEX WITH 5d
分子名称: 3-(benzotriazol-1-yl)-5-[1-methyl-5-[(1~{S})-1-morpholin-4-ylethyl]-1,2,4-triazol-3-yl]pyrazin-2-amine, Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform
著者Petersen, J, Terstige, I, Perry, M, Svensson, T, Tyrchan, C, Lindmark, H, Oster, L.
登録日2016-08-23
公開日2017-04-19
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (2.6 Å)
主引用文献Discovery of triazole aminopyrazines as a highly potent and selective series of PI3K delta inhibitors.
Bioorg. Med. Chem. Lett., 27, 2017
5T23
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BU of 5t23 by Molmil
PI3Kg IN COMPLEX WITH 5d
分子名称: 3-(benzotriazol-1-yl)-5-[1-methyl-5-[(1~{S})-1-morpholin-4-ylethyl]-1,2,4-triazol-3-yl]pyrazin-2-amine, Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform
著者Petersen, J, Terstige, I, Perry, M, Svensson, T, Tyrchan, C, Lindmark, H, Oster, L.
登録日2016-08-23
公開日2017-04-19
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (2.78 Å)
主引用文献Discovery of triazole aminopyrazines as a highly potent and selective series of PI3K delta inhibitors.
Bioorg. Med. Chem. Lett., 27, 2017
5T2I
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BU of 5t2i by Molmil
mPI3Kd IN COMPLEX WITH 7k
分子名称: 1-[3-azanyl-6-[1-methyl-5-(1-phenylcyclopropyl)-1,2,4-triazol-3-yl]pyrazin-2-yl]pyrazole-4-carboxamide, Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform
著者Petersen, J, Terstige, I, Perry, M, Svensson, T, Tyrchan, C, Lindmark, H, Oster, L.
登録日2016-08-23
公開日2017-04-19
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Discovery of triazole aminopyrazines as a highly potent and selective series of PI3K delta inhibitors.
Bioorg. Med. Chem. Lett., 27, 2017

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