7XOV
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![BU of 7xov by Molmil](/molmil-images/mine/7xov) | Structural insights into human brain gut peptide cholecystokinin receptors | 分子名称: | 2-[2-[[4-(4-chloranyl-2,5-dimethoxy-phenyl)-5-(2-cyclohexylethyl)-1,3-thiazol-2-yl]carbamoyl]-5,7-dimethyl-indol-1-yl]ethanoic acid, Cholecystokinin receptor type A, Guanine nucleotide-binding protein G(I)/G(S)/G(O) subunit gamma-2, ... | 著者 | Ding, Y, Zhang, H, Liao, Y, Chen, L, Ji, S. | 登録日 | 2022-05-01 | 公開日 | 2022-07-20 | 実験手法 | ELECTRON MICROSCOPY (3 Å) | 主引用文献 | Structural insights into human brain-gut peptide cholecystokinin receptors. Cell Discov, 8, 2022
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7XYD
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![BU of 7xyd by Molmil](/molmil-images/mine/7xyd) | Crystal structure of TMPRSS2 in complex with Nafamostat | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, 4-carbamimidamidobenzoic acid, CALCIUM ION, ... | 著者 | Wang, H, Liu, X, Duan, Y, Liu, X, Sun, L, Yang, H. | 登録日 | 2022-06-01 | 公開日 | 2023-12-06 | 最終更新日 | 2024-06-19 | 実験手法 | X-RAY DIFFRACTION (2.58 Å) | 主引用文献 | Structure-based discovery of dual pathway inhibitors for SARS-CoV-2 entry. Nat Commun, 14, 2023
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7Y0F
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![BU of 7y0f by Molmil](/molmil-images/mine/7y0f) | Crystal structure of TMPRSS2 in complex with UK-371804 | 分子名称: | 2-[(1-carbamimidamido-4-chloranyl-isoquinolin-7-yl)sulfonylamino]-2-methyl-propanoic acid, 2-acetamido-2-deoxy-beta-D-glucopyranose, CALCIUM ION, ... | 著者 | Wang, H, Duan, Y, Liu, X, Sun, L, Yang, H. | 登録日 | 2022-06-04 | 公開日 | 2023-12-06 | 最終更新日 | 2024-06-19 | 実験手法 | X-RAY DIFFRACTION (2.6 Å) | 主引用文献 | Structure-based discovery of dual pathway inhibitors for SARS-CoV-2 entry. Nat Commun, 14, 2023
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7Y0E
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![BU of 7y0e by Molmil](/molmil-images/mine/7y0e) | Crystal structure of TMPRSS2 in complex with Camostat | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, 4-carbamimidamidobenzoic acid, CALCIUM ION, ... | 著者 | Wang, H, Duan, Y, Liu, X, Sun, L, Yang, H. | 登録日 | 2022-06-04 | 公開日 | 2023-12-06 | 最終更新日 | 2024-06-19 | 実験手法 | X-RAY DIFFRACTION (2.39 Å) | 主引用文献 | Structure-based discovery of dual pathway inhibitors for SARS-CoV-2 entry. Nat Commun, 14, 2023
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4KAM
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![BU of 4kam by Molmil](/molmil-images/mine/4kam) | |
4K3E
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![BU of 4k3e by Molmil](/molmil-images/mine/4k3e) | Crystal structure of bovine antibody BLV5B8 with ultralong CDR H3 | 分子名称: | BOVINE ANTIBODY WITH ULTRALONG CDR H3, HEAVY CHAIN, LIGHT CHAIN, ... | 著者 | Ekiert, D.C, Wang, F, Wilson, I.A. | 登録日 | 2013-04-10 | 公開日 | 2013-06-19 | 最終更新日 | 2023-09-20 | 実験手法 | X-RAY DIFFRACTION (2.2 Å) | 主引用文献 | Reshaping antibody diversity. Cell(Cambridge,Mass.), 153, 2013
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6A92
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![BU of 6a92 by Molmil](/molmil-images/mine/6a92) | Crystal structure of a cyclase Filc1 from Fischerella sp. | 分子名称: | 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, CALCIUM ION, TETRAETHYLENE GLYCOL, ... | 著者 | Hu, X.Y, Liu, W.D, Chen, C.C, Guo, R.T. | 登録日 | 2018-07-11 | 公開日 | 2018-12-19 | 最終更新日 | 2023-11-22 | 実験手法 | X-RAY DIFFRACTION (1.58 Å) | 主引用文献 | The Crystal Structure of a Class of Cyclases that Catalyze the Cope Rearrangement Angew. Chem. Int. Ed. Engl., 57, 2018
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4J1U
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![BU of 4j1u by Molmil](/molmil-images/mine/4j1u) | Crystal structure of antibody 93F3 unstable variant | 分子名称: | antibody 93F3 Heavy chain, antibody 93F3 Light chain | 著者 | Wang, F. | 登録日 | 2013-02-02 | 公開日 | 2013-03-13 | 最終更新日 | 2013-05-22 | 実験手法 | X-RAY DIFFRACTION (2.58 Å) | 主引用文献 | Somatic hypermutation maintains antibody thermodynamic stability during affinity maturation. Proc.Natl.Acad.Sci.USA, 110, 2013
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4I88
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![BU of 4i88 by Molmil](/molmil-images/mine/4i88) | R107G HSP16.5 | 分子名称: | Small heat shock protein HSP16.5 | 著者 | Pohl, E, Williamson, I.R, Quinlan, R.A. | 登録日 | 2012-12-03 | 公開日 | 2013-11-13 | 最終更新日 | 2024-02-28 | 実験手法 | X-RAY DIFFRACTION (2.85 Å) | 主引用文献 | Changes in the quaternary structure and function of MjHSP16.5 attributable to deletion of the IXI motif and introduction of the substitution, R107G, in the alpha-crystallin domain. PHILOS.TRANS.R.SOC.LOND.B BIOL.SCI., 368, 2013
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4KW5
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![BU of 4kw5 by Molmil](/molmil-images/mine/4kw5) | M. tuberculosis DprE1 in complex with inhibitor TCA1 | 分子名称: | FLAVIN-ADENINE DINUCLEOTIDE, GLYCEROL, IMIDAZOLE, ... | 著者 | Batt, S.M, Besra, G.S, Futterer, K. | 登録日 | 2013-05-23 | 公開日 | 2013-07-10 | 最終更新日 | 2023-09-20 | 実験手法 | X-RAY DIFFRACTION (2.612 Å) | 主引用文献 | Identification of a small molecule with activity against drug-resistant and persistent tuberculosis. Proc.Natl.Acad.Sci.USA, 110, 2013
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6IRA
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![BU of 6ira by Molmil](/molmil-images/mine/6ira) | Structure of the human GluN1/GluN2A NMDA receptor in the glutamate/glycine-bound state at pH 7.8 | 分子名称: | Glutamate receptor ionotropic, NMDA 1, NMDA 2A | 著者 | Zhang, J, Chang, S, Zhang, X, Zhu, S. | 登録日 | 2018-11-12 | 公開日 | 2019-01-16 | 最終更新日 | 2019-06-05 | 実験手法 | ELECTRON MICROSCOPY (4.5 Å) | 主引用文献 | Structural Basis of the Proton Sensitivity of Human GluN1-GluN2A NMDA Receptors Cell Rep, 25, 2018
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6IV3
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![BU of 6iv3 by Molmil](/molmil-images/mine/6iv3) | |
2YU2
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![BU of 2yu2 by Molmil](/molmil-images/mine/2yu2) | |
3QDR
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![BU of 3qdr by Molmil](/molmil-images/mine/3qdr) | |
2YU1
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3QHA
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![BU of 3qha by Molmil](/molmil-images/mine/3qha) | |
5XVW
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![BU of 5xvw by Molmil](/molmil-images/mine/5xvw) | |
3R7K
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3R1J
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6IV0
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![BU of 6iv0 by Molmil](/molmil-images/mine/6iv0) | |
6IVW
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![BU of 6ivw by Molmil](/molmil-images/mine/6ivw) | |
3R6H
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7E53
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![BU of 7e53 by Molmil](/molmil-images/mine/7e53) | |
6IRH
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![BU of 6irh by Molmil](/molmil-images/mine/6irh) | Structure of the human GluN1/GluN2A NMDA receptor in the glutamate/glycine-bound state at pH 6.3, Class III | 分子名称: | Glutamate receptor ionotropic, NMDA 1, NMDA 2A | 著者 | Zhang, J, Chang, S, Zhang, X, Zhu, S. | 登録日 | 2018-11-12 | 公開日 | 2019-01-16 | 最終更新日 | 2019-06-05 | 実験手法 | ELECTRON MICROSCOPY (7.8 Å) | 主引用文献 | Structural Basis of the Proton Sensitivity of Human GluN1-GluN2A NMDA Receptors Cell Rep, 25, 2018
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3TDE
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![BU of 3tde by Molmil](/molmil-images/mine/3tde) | |