5SRC
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![BU of 5src by Molmil](/molmil-images/mine/5src) | PanDDA analysis group deposition -- Crystal structure of SARS-CoV-2 NSP3 macrodomain in complex with Z5198562500 - (R,R) and (R,S) isomers | 分子名称: | (2R)-[(3R)-1-(7-fluoro-9H-pyrimido[4,5-b]indol-4-yl)piperidin-3-yl](hydroxy)acetic acid, (2S)-[(3R)-1-(7-fluoro-9H-pyrimido[4,5-b]indol-4-yl)piperidin-3-yl](hydroxy)acetic acid, Non-structural protein 3 | 著者 | Correy, G.J, Fraser, J.S. | 登録日 | 2022-06-09 | 公開日 | 2022-07-06 | 最終更新日 | 2023-09-20 | 実験手法 | X-RAY DIFFRACTION (1.05 Å) | 主引用文献 | Iterative computational design and crystallographic screening identifies potent inhibitors targeting the Nsp3 macrodomain of SARS-CoV-2. Proc.Natl.Acad.Sci.USA, 120, 2023
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5SRM
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![BU of 5srm by Molmil](/molmil-images/mine/5srm) | |
5SRR
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![BU of 5srr by Molmil](/molmil-images/mine/5srr) | |
5SS2
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![BU of 5ss2 by Molmil](/molmil-images/mine/5ss2) | |
5SS9
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![BU of 5ss9 by Molmil](/molmil-images/mine/5ss9) | |
5SRQ
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![BU of 5srq by Molmil](/molmil-images/mine/5srq) | |
5SSE
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![BU of 5sse by Molmil](/molmil-images/mine/5sse) | |
5SSJ
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![BU of 5ssj by Molmil](/molmil-images/mine/5ssj) | |
5SSQ
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![BU of 5ssq by Molmil](/molmil-images/mine/5ssq) | |
5SSR
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![BU of 5ssr by Molmil](/molmil-images/mine/5ssr) | |
5SRD
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![BU of 5srd by Molmil](/molmil-images/mine/5srd) | |
5SRV
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![BU of 5srv by Molmil](/molmil-images/mine/5srv) | |
5SS5
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![BU of 5ss5 by Molmil](/molmil-images/mine/5ss5) | |
5SSD
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![BU of 5ssd by Molmil](/molmil-images/mine/5ssd) | PanDDA analysis group deposition -- Crystal structure of SARS-CoV-2 NSP3 macrodomain in complex with ZINCm4000007vvRA - (R,S) isomer | 分子名称: | (1R,2S)-2-({2-[(4S)-7-methyl-8-oxo-7,8-dihydro[1,2,4]triazolo[4,3-a]pyrazin-3-yl]ethyl}carbamoyl)cyclopropane-1-carboxylic acid, Non-structural protein 3 | 著者 | Correy, G.J, Fraser, J.S. | 登録日 | 2022-06-09 | 公開日 | 2022-07-06 | 最終更新日 | 2023-09-20 | 実験手法 | X-RAY DIFFRACTION (1.15 Å) | 主引用文献 | Iterative computational design and crystallographic screening identifies potent inhibitors targeting the Nsp3 macrodomain of SARS-CoV-2. Proc.Natl.Acad.Sci.USA, 120, 2023
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5SSM
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![BU of 5ssm by Molmil](/molmil-images/mine/5ssm) | PanDDA analysis group deposition -- Crystal structure of SARS-CoV-2 NSP3 macrodomain in complex with Z5459166256 - (R,R) and (S,S) isomers | 分子名称: | (1R,2R)-1-[(1H-benzimidazole-5-carbonyl)amino]-4-hydroxy-2,3-dihydro-1H-indene-2-carboxylic acid, (1S,2S)-1-[(1H-benzimidazole-5-carbonyl)amino]-4-hydroxy-2,3-dihydro-1H-indene-2-carboxylic acid, Non-structural protein 3 | 著者 | Correy, G.J, Fraser, J.S. | 登録日 | 2022-06-09 | 公開日 | 2022-07-06 | 最終更新日 | 2023-09-20 | 実験手法 | X-RAY DIFFRACTION (1.15 Å) | 主引用文献 | Iterative computational design and crystallographic screening identifies potent inhibitors targeting the Nsp3 macrodomain of SARS-CoV-2. Proc.Natl.Acad.Sci.USA, 120, 2023
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5SRN
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![BU of 5srn by Molmil](/molmil-images/mine/5srn) | |
5SRX
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![BU of 5srx by Molmil](/molmil-images/mine/5srx) | |
5SRU
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![BU of 5sru by Molmil](/molmil-images/mine/5sru) | |
5SS6
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![BU of 5ss6 by Molmil](/molmil-images/mine/5ss6) | |
5SSC
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![BU of 5ssc by Molmil](/molmil-images/mine/5ssc) | |
5SSO
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![BU of 5sso by Molmil](/molmil-images/mine/5sso) | |