9QB5

AP2-associated protein kinase 1 (AAK1) bound to CKJB68

Summary for 9QB5

• Entry DOI: 10.2210/pdb9qb5/pdb
• Descriptor: AP2-associated protein kinase 1, ~{N}-(phenylmethyl)-7,10-dioxa-13,17,18,21-tetrazatetracyclo[12.5.2.1^{2,6}.0^{17,20}]docosa-1(20),2(22),3,5,14(21),15,18-heptaene-5-carboxamide, SULFATE ION, ... (4 entities in total)
• Functional Keywords: kinase inhibitor macrocycle, transferase
• Biological source: Homo sapiens (human)
• Total number of polymer chains: 2
• Total formula weight: 73089.84

Authors

Preuss, F.,Mensing, T.E.,Hanke, T.,Knapp, S.,Mathea, S. (deposition date: 2025-02-28, release date: 2025-04-09)

• Primary citation: Preuss, F.,Mensing, T.E.,Hanke, T.,Knapp, S.,Mathea, S.; AP2-associated protein kinase 1 (AAK1) bound to CKJB68; To Be Published,

Experimental method

X-RAY DIFFRACTION (2 Å)