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8WB1

Crystal Structure of small molecule KN2H covalently bound to K-Ras(G12D)

Summary for 8WB1
Entry DOI10.2210/pdb8wb1/pdb
DescriptorGTPase KRas, GUANOSINE-5'-DIPHOSPHATE, MAGNESIUM ION, ... (6 entities in total)
Functional Keywordscovalent inhibitor, kras g12d, hydrolase
Biological sourceHomo sapiens (human)
Total number of polymer chains1
Total formula weight20559.09
Authors
Zhou, L.,Zhang, R.,Shuai, T.B. (deposition date: 2023-09-08, release date: 2024-09-11, Last modification date: 2024-10-09)
Primary citationZhou, L.,Zhang, R.,Shuai, T.B.
Crystal Structure of small molecule KN2H covalently bound to K-Ras(G12D)
To Be Published,
Experimental method
X-RAY DIFFRACTION (1.72 Å)
Structure validation

225946

数据于2024-10-09公开中

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