8WB1
Crystal Structure of small molecule KN2H covalently bound to K-Ras(G12D)
Summary for 8WB1
Entry DOI | 10.2210/pdb8wb1/pdb |
Descriptor | GTPase KRas, GUANOSINE-5'-DIPHOSPHATE, MAGNESIUM ION, ... (6 entities in total) |
Functional Keywords | covalent inhibitor, kras g12d, hydrolase |
Biological source | Homo sapiens (human) |
Total number of polymer chains | 1 |
Total formula weight | 20559.09 |
Authors | Zhou, L.,Zhang, R.,Shuai, T.B. (deposition date: 2023-09-08, release date: 2024-09-11, Last modification date: 2024-10-09) |
Primary citation | Zhou, L.,Zhang, R.,Shuai, T.B. Crystal Structure of small molecule KN2H covalently bound to K-Ras(G12D) To Be Published, |
Experimental method | X-RAY DIFFRACTION (1.72 Å) |
Structure validation
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