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8V70

Crystal structure of the core catalytic domain of human inositol phosphate multikinase in complex with compound 6

8V70 の概要
エントリーDOI10.2210/pdb8v70/pdb
分子名称Inositol polyphosphate multikinase, (5P)-3-phenyl-5-(1H-tetrazol-5-yl)-2,1-benzoxazole, SULFATE ION, ... (4 entities in total)
機能のキーワードstructure-based inhibitor development, kinase, inhibitor, inositol polyphosphate, inositol polyphosphate kinase, transferase, transferase-transferase inhibitor complex, transferase/transferase inhibitor
由来する生物種Homo sapiens (human)
詳細
タンパク質・核酸の鎖数1
化学式量合計30187.23
構造登録者
Wang, H.,Shears, S.B. (登録日: 2023-12-04, 公開日: 2024-12-11)
主引用文献Wang, H.,Shears, S.B.
Structure-based development of IPMK kinase inhibitors.
To Be Published,
実験手法
X-RAY DIFFRACTION (1.85 Å)
構造検証レポート
Validation report summary of 8v70
検証レポート(詳細版)ダウンロードをダウンロード

239149

件を2025-07-23に公開中

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