8P11
X-ray structure of acetylcholine-binding protein (AChBP) in complex with FL003044.
Summary for 8P11
Entry DOI | 10.2210/pdb8p11/pdb |
Descriptor | Acetylcholine-binding protein, CHLORIDE ION, 4-(4-chlorophenyl)piperidin-4-ol, ... (5 entities in total) |
Functional Keywords | fragment based drug design, acetylcholine-binding protein, choline-binding proteins, choline-binding protein |
Biological source | Lymnaea stagnalis (great pond snail) |
Total number of polymer chains | 10 |
Total formula weight | 271896.58 |
Authors | Cederfelt, D.,Boronat, P.,Dobritzsch, D.,Hennig, S.,Fitzgerald, E.A.,de Esch, I.J.P.,Danielson, U.H. (deposition date: 2023-05-11, release date: 2024-05-08) |
Primary citation | Fitzgerald, E.A.,Cederfelt, D.,Boronat, P.,Aarmo Lund, B.,Dobritzsch, D.,de Esch, I.J.P.,Danielson, U.H. Elucidating the regulation of ligand gated ion channels via biophysical studies of ligand-induced conformational dynamics of acetylcholine binding proteins To Be Published, |
Experimental method | X-RAY DIFFRACTION (1.9 Å) |
Structure validation
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