8P06
Crystal structure of human Casein Kinase II subunit alpha (CK2a1) in complex with 5-((2-(4H-1,2,4-triazol-4-yl)pyridin-4-yl)amino)-7-(cyclopropylamino)pyrazolo[1,5-a]pyrimidine-3-carbonitrile
8P06 の概要
エントリーDOI | 10.2210/pdb8p06/pdb |
分子名称 | CSNK2A1 protein, SULFATE ION, 7-(cyclopropylamino)-5-[[2-(1,2,4-triazol-4-yl)pyridin-4-yl]amino]pyrazolo[1,5-a]pyrimidine-3-carbonitrile, ... (4 entities in total) |
機能のキーワード | kinase, ck2, typi inhibitor, transferase |
由来する生物種 | Homo sapiens (human) |
タンパク質・核酸の鎖数 | 2 |
化学式量合計 | 82141.18 |
構造登録者 | Kraemer, A.,Ong, H.W.,Yang, X.,Brown, J.W.,Chang, E.,Willson, T.,Knapp, S.,Structural Genomics Consortium (SGC) (登録日: 2023-05-09, 公開日: 2023-06-21) |
主引用文献 | Kraemer, A.,Ong, H.W.,Yang, X.,Brown, J.W.,Chang, E.,Willson, T.,Knapp, S.,Structural Genomics Consortium (SGC) Crystal structure of human Casein Kinase II subunit alpha (CK2a1) in complex with 5-((2-(4H-1,2,4-triazol-4-yl)pyridin-4-yl)amino)-7-(cyclopropylamino)pyrazolo[1,5-a]pyrimidine-3-carbonitrile To Be Published, |
実験手法 | X-RAY DIFFRACTION (2.4 Å) |
構造検証レポート
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