8ORC
Mus Musculus Acetylcholinesterase in complex with AL237
Summary for 8ORC
Entry DOI | 10.2210/pdb8orc/pdb |
Descriptor | Acetylcholinesterase, 1-[2-(dimethylamino)ethyl]-3-(2-methoxyphenyl)thiourea, 2-(2-METHOXYETHOXY)ETHANOL, ... (7 entities in total) |
Functional Keywords | neurotransmission, cholinesterase, inhibitor, hydrolase |
Biological source | Mus musculus (house mouse) |
Total number of polymer chains | 2 |
Total formula weight | 121609.62 |
Authors | Ekstrom, F.E.,Linusson, A. (deposition date: 2023-04-13, release date: 2024-04-24, Last modification date: 2024-10-02) |
Primary citation | Kumari, R.,Lindgren, C.,Kumar, R.,Forsgren, N.,Andersson, C.D.,Ekstrom, F.,Linusson, A. Enzyme Dynamics Determine the Potency and Selectivity of Inhibitors Targeting Disease-Transmitting Mosquitoes. Acs Infect Dis., 2024 Cited by PubMed: 39291389DOI: 10.1021/acsinfecdis.4c00531 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (2.1 Å) |
Structure validation
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