8K6D
Crystal structure of SARS-CoV-2 3CLpro M49K/S301P mutant in complex with WU-04
Summary for 8K6D
Entry DOI | 10.2210/pdb8k6d/pdb |
Descriptor | 3C-like proteinase nsp5, ~{N}-[(1~{S},2~{R})-2-[[4-bromanyl-2-(methylcarbamoyl)-6-nitro-phenyl]amino]cyclohexyl]isoquinoline-4-carboxamide (3 entities in total) |
Functional Keywords | sars-cov-2 3clpro, mutant, wu-04, inhibitor, viral protein |
Biological source | Severe acute respiratory syndrome coronavirus 2 (2019-nCoV, SARS-CoV-2) |
Total number of polymer chains | 1 |
Total formula weight | 34359.95 |
Authors | |
Primary citation | Zhang, L.,Xie, X.,Luo, H.,Qian, R.,Yang, Y.,Yu, H.,Huang, J.,Shi, P.Y.,Hu, Q. Resistance mechanisms of SARS-CoV-2 3CLpro to the non-covalent inhibitor WU-04. Cell Discov, 10:40-40, 2024 Cited by PubMed: 38594245DOI: 10.1038/s41421-024-00673-0 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (1.65 Å) |
Structure validation
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